DK150477C - ANALOGY PROCEDURE FOR PREPARING 4- (4- (NAPHTHALENYLOXY) -1-PIPERIDINYL) -1-PHENYL-1-BUTANON DERIVATIVES AND INTERMEDIATES FOR USING THE PROCEDURE - Google Patents

ANALOGY PROCEDURE FOR PREPARING 4- (4- (NAPHTHALENYLOXY) -1-PIPERIDINYL) -1-PHENYL-1-BUTANON DERIVATIVES AND INTERMEDIATES FOR USING THE PROCEDURE

Info

Publication number
DK150477C
DK150477C DK337280A DK337280A DK150477C DK 150477 C DK150477 C DK 150477C DK 337280 A DK337280 A DK 337280A DK 337280 A DK337280 A DK 337280A DK 150477 C DK150477 C DK 150477C
Authority
DK
Denmark
Prior art keywords
procedure
butanon
naphthalenyloxy
piperidinyl
intermediates
Prior art date
Application number
DK337280A
Other languages
Danish (da)
Other versions
DK337280A (en
DK150477B (en
Inventor
Albert A Carr
Robert A Farr
Original Assignee
Richardson Merrell Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Richardson Merrell Inc filed Critical Richardson Merrell Inc
Publication of DK337280A publication Critical patent/DK337280A/en
Publication of DK150477B publication Critical patent/DK150477B/en
Application granted granted Critical
Publication of DK150477C publication Critical patent/DK150477C/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D211/00Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/36Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D211/40Oxygen atoms
    • C07D211/44Oxygen atoms attached in position 4
    • C07D211/46Oxygen atoms attached in position 4 having a hydrogen atom as the second substituent in position 4
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/20Hypnotics; Sedatives

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Anesthesiology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Biomedical Technology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Hydrogenated Pyridines (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
DK337280A 1979-08-06 1980-08-05 ANALOGY PROCEDURE FOR PREPARING 4- (4- (NAPHTHALENYLOXY) -1-PIPERIDINYL) -1-PHENYL-1-BUTANON DERIVATIVES AND INTERMEDIATES FOR USING THE PROCEDURE DK150477C (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US6430579A 1979-08-06 1979-08-06
US6430579 1979-08-06

Publications (3)

Publication Number Publication Date
DK337280A DK337280A (en) 1981-02-07
DK150477B DK150477B (en) 1987-03-09
DK150477C true DK150477C (en) 1987-10-12

Family

ID=22055014

Family Applications (1)

Application Number Title Priority Date Filing Date
DK337280A DK150477C (en) 1979-08-06 1980-08-05 ANALOGY PROCEDURE FOR PREPARING 4- (4- (NAPHTHALENYLOXY) -1-PIPERIDINYL) -1-PHENYL-1-BUTANON DERIVATIVES AND INTERMEDIATES FOR USING THE PROCEDURE

Country Status (18)

Country Link
JP (1) JPS5626875A (en)
AU (1) AU534398B2 (en)
BE (1) BE884581A (en)
CA (1) CA1123440A (en)
CH (1) CH644364A5 (en)
DE (1) DE3028064A1 (en)
DK (1) DK150477C (en)
ES (1) ES493591A0 (en)
FR (1) FR2463129A1 (en)
GB (1) GB2056447B (en)
IE (1) IE49998B1 (en)
IL (1) IL60593A (en)
IT (1) IT1146966B (en)
NL (1) NL8004147A (en)
NO (1) NO153726C (en)
NZ (1) NZ194248A (en)
SE (1) SE448728B (en)
ZA (1) ZA804112B (en)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2508445A1 (en) * 1981-06-29 1982-12-31 Sori Soc Rech Ind NOVEL BENZOYL-PHENYL-PIPERIDINE DERIVATIVES, PROCESS FOR PREPARING THEM AND THEIR USE, IN PARTICULAR THERAPEUTICS
ATE13425T1 (en) * 1981-10-15 1985-06-15 Synthelabo PIPERIDINE DERIVATIVES, PROCESSES FOR THEIR PRODUCTION AND THEIR USE AS MEDICINAL PRODUCTS.
GB8321157D0 (en) * 1983-08-05 1983-09-07 Fordonal Sa Piperidine derivatives
JP2751346B2 (en) * 1989-03-15 1998-05-18 ミノルタ株式会社 Printer
JP5373104B2 (en) * 2008-11-17 2013-12-18 エフ.ホフマン−ラ ロシュ アーゲー Naphthyl acetic acid used as CRTH2 antagonist or partial agonist

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB895309A (en) * 1959-11-18 1962-05-02 Res Lab Dr C Janssen Nv Pyrrolidine and piperidine derivatives
BE637978A (en) * 1963-02-15
US3743645A (en) * 1970-10-19 1973-07-03 Robins Co Inc A H 1-substituted-4-phenoxypiperidines
ZA717147B (en) * 1970-11-27 1972-07-26 Richardson Merrell Inc 4-(4-(alpha-hydroxybenzyl)piperidino)-4'-fluorobutyrophenone derivatives
US3806526A (en) * 1972-01-28 1974-04-23 Richardson Merrell Inc 1-aroylalkyl-4-diphenylmethyl piperidines
SE7409245L (en) * 1973-07-19 1975-01-20 Robins Co Inc A H
DE2718405A1 (en) * 1977-04-26 1978-11-02 Boehringer Sohn Ingelheim NEW N-NECK CLAMP ON 1- (3-BENZOYLPROPYL) -4-PIPERIDYL NECK CLAMP ON -SULPHONIC ACID AMIDES AND METHOD FOR THE PRODUCTION THEREOF
US4134982A (en) * 1977-09-26 1979-01-16 Warner-Lambert Company Antipsychotic 1-[4,4-Bis(4-fluorophenyl) butyl]-4-phenoxy-1,2,3,6-tetrahydropyridines

Also Published As

Publication number Publication date
IE49998B1 (en) 1986-01-22
NZ194248A (en) 1984-07-06
IL60593A (en) 1984-03-30
IT1146966B (en) 1986-11-19
IT8049394A0 (en) 1980-07-31
GB2056447B (en) 1983-07-06
DK337280A (en) 1981-02-07
AU534398B2 (en) 1984-01-26
CA1123440A (en) 1982-05-11
IE801382L (en) 1981-02-06
NO153726C (en) 1986-05-14
DE3028064C2 (en) 1989-11-09
AU6039480A (en) 1981-02-12
NO153726B (en) 1986-02-03
JPS5626875A (en) 1981-03-16
GB2056447A (en) 1981-03-18
JPS6341390B2 (en) 1988-08-17
CH644364A5 (en) 1984-07-31
ES8105981A1 (en) 1981-07-01
DE3028064A1 (en) 1981-02-26
ZA804112B (en) 1981-07-29
IL60593A0 (en) 1980-09-16
NL8004147A (en) 1981-02-10
ES493591A0 (en) 1981-07-01
SE448728B (en) 1987-03-16
DK150477B (en) 1987-03-09
BE884581A (en) 1980-11-17
FR2463129A1 (en) 1981-02-20
FR2463129B1 (en) 1983-04-22
SE8005493L (en) 1981-02-07
NO802346L (en) 1981-02-09

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