DK416888D0 - CEPHALOSPORINE COMPOUNDS, CRYSTALLINIC DERIVATIVES THEREOF, INTERMEDIATES FOR USE IN THE PRODUCTION OF CEPHALOSPORINE COMPOUNDS AND PROCEDURES FOR THE PRODUCTION OF CEPHALOSPORINE COMPOUNDS - Google Patents
CEPHALOSPORINE COMPOUNDS, CRYSTALLINIC DERIVATIVES THEREOF, INTERMEDIATES FOR USE IN THE PRODUCTION OF CEPHALOSPORINE COMPOUNDS AND PROCEDURES FOR THE PRODUCTION OF CEPHALOSPORINE COMPOUNDSInfo
- Publication number
- DK416888D0 DK416888D0 DK416888A DK416888A DK416888D0 DK 416888 D0 DK416888 D0 DK 416888D0 DK 416888 A DK416888 A DK 416888A DK 416888 A DK416888 A DK 416888A DK 416888 D0 DK416888 D0 DK 416888D0
- Authority
- DK
- Denmark
- Prior art keywords
- production
- cephalosporine compounds
- cephalosporine
- compounds
- crystallinic
- Prior art date
Links
- HOKIDJSKDBPKTQ-UHFFFAOYSA-N 3-(acetyloxymethyl)-7-[(5-amino-5-carboxypentanoyl)amino]-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid Chemical class S1CC(COC(=O)C)=C(C(O)=O)N2C(=O)C(NC(=O)CCCC(N)C(O)=O)C12 HOKIDJSKDBPKTQ-UHFFFAOYSA-N 0.000 title 3
- 239000000543 intermediate Substances 0.000 title 1
- 238000000034 method Methods 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
- C07D501/14—Compounds having a nitrogen atom directly attached in position 7
- C07D501/16—Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
- C07D501/20—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids
- C07D501/24—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids with hydrocarbon radicals, substituted by hetero atoms or hetero rings, attached in position 3
- C07D501/36—Methylene radicals, substituted by sulfur atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/587—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with aliphatic hydrocarbon radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms, said aliphatic radicals being substituted in the alpha-position to the ring by a hetero atom, e.g. with m >= 0, Z being a singly or a doubly bound hetero atom
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Communicable Diseases (AREA)
- Pharmacology & Pharmacy (AREA)
- Oncology (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Cephalosporin Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP61280019A JPS63132893A (en) | 1986-11-25 | 1986-11-25 | Novel cephalosporin derivative, production thereof and antibacterial agent containing said derivative as active ingredient |
PCT/JP1987/000902 WO1988003924A1 (en) | 1986-11-25 | 1987-11-20 | Novel cephalosporin derivatives and their crystalline derivatives |
Publications (2)
Publication Number | Publication Date |
---|---|
DK416888A DK416888A (en) | 1988-07-25 |
DK416888D0 true DK416888D0 (en) | 1988-07-25 |
Family
ID=17619166
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
DK416888A DK416888D0 (en) | 1986-11-25 | 1988-07-25 | CEPHALOSPORINE COMPOUNDS, CRYSTALLINIC DERIVATIVES THEREOF, INTERMEDIATES FOR USE IN THE PRODUCTION OF CEPHALOSPORINE COMPOUNDS AND PROCEDURES FOR THE PRODUCTION OF CEPHALOSPORINE COMPOUNDS |
Country Status (13)
Country | Link |
---|---|
US (1) | US4866055A (en) |
EP (1) | EP0272487A1 (en) |
JP (1) | JPS63132893A (en) |
KR (1) | KR890700128A (en) |
AU (2) | AU598607B2 (en) |
DK (1) | DK416888D0 (en) |
FI (1) | FI883496A (en) |
IL (1) | IL84580A0 (en) |
NZ (1) | NZ222670A (en) |
PH (1) | PH24993A (en) |
WO (1) | WO1988003924A1 (en) |
ZA (1) | ZA878835B (en) |
ZW (1) | ZW21787A1 (en) |
Families Citing this family (12)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FI872879A (en) * | 1986-07-21 | 1988-01-22 | Sankei Yakuhin Kk | --LAKTAMFOERENING, FOERFARANDE FOER DESS FRAMSTAELLNING, DENNA INNEHAOLLANDE LAEKEMEDELSKOMPOSITION FOER BEHANDLING AV SJUKDOM MED BAKTERIEINFEKTION SAMT MELLANPRODUKTER FOER DESS SYNTES. |
US4880798A (en) * | 1986-11-25 | 1989-11-14 | Mochida Pharmaceutical Co., Ltd. | Cephalosporin derivatives |
NZ225383A (en) * | 1987-08-07 | 1990-03-27 | Sankei Yakuhin Kk | Cephalosporin derivatives and pharmaceutical compositions |
JPH0418056A (en) * | 1990-05-09 | 1992-01-22 | Sanwa Kagaku Kenkyusho Co Ltd | Polyisoprene compound, its salt, production thereof and remedy for peptic ulcer containing the same as active ingredient |
US5095012A (en) * | 1990-08-23 | 1992-03-10 | Bristol-Myers Squibb Company | Antibiotic c-7 catechol-substituted cephalosporin compounds, compositions, and method of use thereof |
US5234920A (en) * | 1990-08-23 | 1993-08-10 | Bristol-Myers Squibb Company | Antibiotic C-7 catechol-substituted cephalosporin compounds, compositions, and method of use thereof |
EP0544166A3 (en) * | 1991-11-26 | 1993-11-03 | Hoffmann La Roche | Cephalosporinderivatives |
HU221478B (en) * | 1991-12-12 | 2002-10-28 | Hoechst Marion Roussel Inc | Cephalosporine derivatives substituted in 7th position by benzyl-oxi-imino group, pharmaceutical compositions containing the same, method for producing them and intermediates |
IL105191A (en) * | 1992-04-04 | 1998-08-16 | Basf Ag | 0-Iminooxymethylbenzoic acids and their preparation |
KR100257129B1 (en) * | 1993-09-11 | 2000-05-15 | 성재갑 | Novel cephalosphorine antibiotics |
DE102004024010A1 (en) * | 2004-05-14 | 2005-12-01 | Bayer Chemicals Ag | Process for the preparation of difluorobenzo-1,3-dioxole-5-carboxylic acid derivatives |
US8698184B2 (en) | 2011-01-21 | 2014-04-15 | Cree, Inc. | Light emitting diodes with low junction temperature and solid state backlight components including light emitting diodes with low junction temperature |
Family Cites Families (36)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
BE566543A (en) * | 1957-04-09 | |||
JPS503170B1 (en) * | 1970-06-11 | 1975-01-31 | ||
GB1399086A (en) * | 1971-05-14 | 1975-06-25 | Glaxo Lab Ltd | Cephalosporin compounds |
NZ189245A (en) * | 1976-01-23 | 1979-12-11 | Roussel Uclaf | Substituted 2-(2-amino-4-thiazoyl)-2-hydroxyimino-acetic acid derivatives |
GB1576625A (en) * | 1976-04-12 | 1980-10-08 | Fujisawa Pharmaceutical Co | Syn isomer 3,7 disubstituted 3 cephem 4 carboxylic acid compounds and processes for the preparation thereof |
US4082912A (en) * | 1976-06-30 | 1978-04-04 | Bristol-Myers Company | Certain 7-acylamido-3-(2-carboxyalkyl-2,3-dihydro-s-triazolo[4,3-b]pyridazin-3-on-6-ylmethyl)-3-cephem-4-carboxylic acids their salts and easily hydrolyzed esters |
US4103085A (en) * | 1977-02-24 | 1978-07-25 | Bristol-Myers Company | 7-(Syn-α-alkoxy-iminofurylacetamido-3-(2-carboxyalkyl-2,3-dihydro-s-triazolo[4,3-b]pyridazin-3-on-6-ylthiomethyl)-3-cephem-4-carboxylic acids |
US4104469A (en) * | 1977-04-15 | 1978-08-01 | Bristol-Myers Company | 7-(Syn-α-alkoxy-iminofuryl)acetamido-3-(2-methyl-2,3-dihydro-s-triazolo[4,3-b]pyridazin-3-on-6-ylthiomethyl)-3-cephem-4-carboxylic acids |
DE2714880A1 (en) * | 1977-04-02 | 1978-10-26 | Hoechst Ag | CEPHEMDER DERIVATIVES AND PROCESS FOR THEIR PRODUCTION |
DE2716677C2 (en) * | 1977-04-15 | 1985-10-10 | Hoechst Ag, 6230 Frankfurt | Cephem derivatives and processes for their preparation |
FR2400519A1 (en) * | 1977-08-17 | 1979-03-16 | Roussel Uclaf | CRYSTALLINE FORM OF SODIUM SALT OF AN OXIMIN DERIVATIVE OF 7-AMINO-THIAZOLYL ACETAMIDO CEPHALOSPORANIC, ITS PREPARATION PROCESS AND ITS APPLICATION AS A MEDICINAL PRODUCT |
FR2432521A1 (en) * | 1978-03-31 | 1980-02-29 | Roussel Uclaf | NOVEL O-SUBSTITUTED OXIMES DERIVED FROM 7-AMINO THIAZOLYL ACETAMIDO CEPHALOSPORANIC ACID, THEIR PREPARATION PROCESS AND THEIR USE AS MEDICAMENTS |
AR231986A1 (en) * | 1978-05-26 | 1985-04-30 | Glaxo Group Ltd | PROCEDURE FOR PREPARING CEPHALOSPORIN ANTIBIOTICS |
US4331666A (en) * | 1979-05-11 | 1982-05-25 | Farmitalia Carlo Erba S.P.A. | 3-[(8-Carboxy-6-tetrazolo[1,5-b]pyridazinyl)-thiomethyl]-7-[2-(2-amino-4-thiazolyl)-2-methoxyimino-acetamido]-3-cephem-4-carboxylic acid |
EP0037380B1 (en) * | 1980-03-28 | 1984-09-12 | BIOCHEMIE Gesellschaft m.b.H. | New process for the production of cephalosporin antibiotics, and novel intermediates used in such process and their production |
US4316024A (en) * | 1980-09-15 | 1982-02-16 | Bristol-Myers Company | Dioxo piperazine compounds |
JPS6011917B2 (en) * | 1981-04-09 | 1985-03-28 | 山之内製薬株式会社 | Novel cephalosporin compounds |
US4436912A (en) * | 1981-09-08 | 1984-03-13 | Eli Lilly And Company | 7-[2-(2-Aminooxazol-4-yl)-2-(oximino)acetamido cephalosporin antibiotics and intermediates therefor |
JPS5849382A (en) * | 1981-09-18 | 1983-03-23 | Kyowa Hakko Kogyo Co Ltd | Beta-lactam compound |
US4526977A (en) * | 1981-10-07 | 1985-07-02 | American Home Products Corporation | 2-(3-Amino-5-isoxazolyl)-2-oxyimino-acetic acids |
US4594417A (en) * | 1981-10-30 | 1986-06-10 | Eli Lilly Company | Crystalline antibiotic salt |
DE3143537A1 (en) * | 1981-11-03 | 1983-05-11 | Hoechst Ag, 6230 Frankfurt | CRYSTALLINE SALTS FROM CEFODIZIM AND METHOD FOR THE PRODUCTION THEREOF |
FR2517309A1 (en) * | 1981-12-01 | 1983-06-03 | Sanofi Sa | NOVEL DERIVATIVES OF CEPHALOSPORINS SUBSTITUTED IN POSITION 3 BY A HETEROCYCLE THIOMETHYL GROUP; PROCESS FOR THE PREPARATION OF SAID COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME |
DE3207840A1 (en) * | 1982-03-04 | 1983-09-15 | Hoechst Ag, 6230 Frankfurt | "CEPHALOSPORINE DERIVATIVES AND METHOD FOR THE PRODUCTION THEREOF" |
US4500526A (en) * | 1982-06-28 | 1985-02-19 | Bristol-Myers Company | Cephalosporin derivatives |
JPS5946292A (en) * | 1982-09-09 | 1984-03-15 | Otsuka Chem Co Ltd | 2-substituted cephem derivative and its preparation |
JPS5973575A (en) * | 1982-10-05 | 1984-04-25 | Shionogi & Co Ltd | Propynylaminoisoxazole derivative |
DE3248281A1 (en) * | 1982-12-28 | 1984-06-28 | Hoechst Ag, 6230 Frankfurt | CRYSTALIZED CEPHEMIC ACID ADDITION SALTS AND METHOD FOR THE PRODUCTION THEREOF |
JPS59155391A (en) * | 1983-02-22 | 1984-09-04 | Tanabe Seiyaku Co Ltd | Novel cephalosporin derivative and its preparation |
JPS6066987A (en) * | 1983-09-20 | 1985-04-17 | Takeda Chem Ind Ltd | Antibiotic substance tan-547, production thereof and microorganism |
US4600773A (en) * | 1983-12-01 | 1986-07-15 | Eli Lilly And Company | Crystalline cephalexin hydrochloride monohydrate |
EP0150507B1 (en) * | 1983-12-29 | 1992-08-05 | Mochida Pharmaceutical Co., Ltd. | Cephalosporin derivatives, processes for producing the same and compositions containing them |
JPS61126089A (en) * | 1984-11-26 | 1986-06-13 | Mochida Pharmaceut Co Ltd | Cephalosporin derivative, production thereof, and antibacterial agent containing same |
JPS60142987A (en) * | 1983-12-29 | 1985-07-29 | Mochida Pharmaceut Co Ltd | Cephalosporin derivative |
NZ215527A (en) * | 1985-04-01 | 1989-06-28 | Mochida Pharm Co Ltd | Cephalosporin derivatives and pharmaceutical compositions |
US4880798A (en) * | 1986-11-25 | 1989-11-14 | Mochida Pharmaceutical Co., Ltd. | Cephalosporin derivatives |
-
1986
- 1986-11-25 JP JP61280019A patent/JPS63132893A/en active Pending
-
1987
- 1987-11-16 US US07/120,932 patent/US4866055A/en not_active Expired - Fee Related
- 1987-11-20 WO PCT/JP1987/000902 patent/WO1988003924A1/en active Application Filing
- 1987-11-24 IL IL84580A patent/IL84580A0/en unknown
- 1987-11-24 NZ NZ222670A patent/NZ222670A/en unknown
- 1987-11-24 AU AU81631/87A patent/AU598607B2/en not_active Ceased
- 1987-11-25 ZW ZW217/87A patent/ZW21787A1/en unknown
- 1987-11-25 PH PH36125A patent/PH24993A/en unknown
- 1987-11-25 ZA ZA878835A patent/ZA878835B/en unknown
- 1987-11-25 EP EP87117396A patent/EP0272487A1/en not_active Withdrawn
-
1988
- 1988-07-25 KR KR1019880700878A patent/KR890700128A/en not_active Application Discontinuation
- 1988-07-25 FI FI883496A patent/FI883496A/en not_active IP Right Cessation
- 1988-07-25 DK DK416888A patent/DK416888D0/en not_active Application Discontinuation
-
1990
- 1990-09-24 AU AU63167/90A patent/AU6316790A/en not_active Abandoned
Also Published As
Publication number | Publication date |
---|---|
PH24993A (en) | 1990-12-26 |
AU8163187A (en) | 1988-05-26 |
EP0272487A1 (en) | 1988-06-29 |
FI883496A0 (en) | 1988-07-25 |
ZA878835B (en) | 1988-05-25 |
AU598607B2 (en) | 1990-06-28 |
ZW21787A1 (en) | 1988-09-07 |
NZ222670A (en) | 1990-08-28 |
US4866055A (en) | 1989-09-12 |
IL84580A0 (en) | 1988-04-29 |
KR890700128A (en) | 1989-03-02 |
DK416888A (en) | 1988-07-25 |
JPS63132893A (en) | 1988-06-04 |
WO1988003924A1 (en) | 1988-06-02 |
FI883496A (en) | 1988-07-25 |
AU6316790A (en) | 1991-03-28 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
AHB | Application shelved due to non-payment |