DK149625C - Analogifremgangsmaade til fremstilling af n-substituerede (8-halogen- eller -trifluormethyl-4-quinolylamino)-benzamider eller et farmaceutiskacceptabelt syreadditionssalt deraf - Google Patents
Analogifremgangsmaade til fremstilling af n-substituerede (8-halogen- eller -trifluormethyl-4-quinolylamino)-benzamider eller et farmaceutiskacceptabelt syreadditionssalt derafInfo
- Publication number
- DK149625C DK149625C DK403878A DK403878A DK149625C DK 149625 C DK149625 C DK 149625C DK 403878 A DK403878 A DK 403878A DK 403878 A DK403878 A DK 403878A DK 149625 C DK149625 C DK 149625C
- Authority
- DK
- Denmark
- Prior art keywords
- quinolylamino
- trifluormethyl
- benzamides
- analogue
- halogen
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
- C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
- C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D215/38—Nitrogen atoms
- C07D215/42—Nitrogen atoms attached in position 4
- C07D215/44—Nitrogen atoms attached in position 4 with aryl radicals attached to said nitrogen atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Pain & Pain Management (AREA)
- Animal Behavior & Ethology (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Rheumatology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Quinoline Compounds (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GB38264/77A GB1573186A (en) | 1977-09-14 | 1977-09-14 | 4-aminoquinoline derivatives |
GB3826477 | 1978-05-24 |
Publications (3)
Publication Number | Publication Date |
---|---|
DK403878A DK403878A (da) | 1979-03-15 |
DK149625B DK149625B (da) | 1986-08-18 |
DK149625C true DK149625C (da) | 1987-01-26 |
Family
ID=10402337
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
DK403878A DK149625C (da) | 1977-09-14 | 1978-09-13 | Analogifremgangsmaade til fremstilling af n-substituerede (8-halogen- eller -trifluormethyl-4-quinolylamino)-benzamider eller et farmaceutiskacceptabelt syreadditionssalt deraf |
Country Status (9)
Country | Link |
---|---|
US (1) | US4357333A (de) |
EP (1) | EP0001175B1 (de) |
JP (1) | JPS5492974A (de) |
AU (1) | AU516318B2 (de) |
CA (1) | CA1096870A (de) |
DK (1) | DK149625C (de) |
GB (1) | GB1573186A (de) |
IE (1) | IE47249B1 (de) |
ZA (1) | ZA784709B (de) |
Families Citing this family (10)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
YU192782A (en) * | 1981-09-30 | 1985-04-30 | Recordati Chem Pharm | Process for obtaining anthranilic acid esters |
PH22302A (en) * | 1985-02-11 | 1988-07-22 | Fujisawa Pharmaceutical Co | Piperidine compounds |
US5212182A (en) * | 1990-10-03 | 1993-05-18 | American Home Products Corpooration | Substituted quinolinyl- and naphthalenylbenzamides or benzylamines and related compounds useful as analgesics |
US5438064A (en) * | 1991-12-23 | 1995-08-01 | American Home Products Corporation | Derivatives of 4-anilinoquinoline-3-carboxamide as analgesic agents |
US5656642A (en) * | 1993-04-07 | 1997-08-12 | Otsuka Pharmaceutical Co., Ltd. | Peripheral vasodilating agent containing piperidine derivative as active ingredient |
US6028111A (en) * | 1996-03-08 | 2000-02-22 | Oxigene, Inc. | Compositions and use of benzamides and nicotinamides as anti-inflammatory agents |
SE0102858D0 (sv) * | 2001-08-27 | 2001-08-27 | Astrazeneca Ab | N-type calcium channel antagonists for the treatment of pain |
SE0102857D0 (sv) * | 2001-08-27 | 2001-08-27 | Astrazeneca Ab | N-type calcium channel antagonists for the treatment of pain |
US7307088B2 (en) | 2002-07-09 | 2007-12-11 | Amgen Inc. | Substituted anthranilic amide derivatives and methods of use |
MY142362A (en) | 2004-01-29 | 2010-11-30 | Otsuka Pharma Co Ltd | Pharmaceutical composition for promoting angiogenesis |
Family Cites Families (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3174972A (en) * | 1961-07-10 | 1965-03-23 | Table ii | |
GB1416872A (en) * | 1972-03-10 | 1975-12-10 | Wyeth John & Brother Ltd | 4-aminoquinoline derivatives |
US3875165A (en) * | 1973-02-22 | 1975-04-01 | Wyeth John & Brother Ltd | (4-Quinolylamino)-(N-piperidyl)benzamides and N-{8 (quinolylamino)-benzoyl{9 piperidines |
US4025629A (en) * | 1974-01-07 | 1977-05-24 | The Upjohn Company | P-(trifluoromethylquinolylamino)benzamides, pharmaceutical dosage forms and method of treatment |
GB1474296A (en) * | 1975-01-23 | 1977-05-18 | Wyeth John & Brother Ltd | 4-aminoquinoline derivatives |
JPS5231353A (en) * | 1975-09-05 | 1977-03-09 | Hitachi Ltd | Ac switch controlling device |
-
1977
- 1977-09-14 GB GB38264/77A patent/GB1573186A/en not_active Expired
-
1978
- 1978-08-18 ZA ZA784709A patent/ZA784709B/xx unknown
- 1978-08-23 AU AU39171/78A patent/AU516318B2/en not_active Expired
- 1978-08-28 IE IE1728/78A patent/IE47249B1/en unknown
- 1978-09-01 EP EP78300353A patent/EP0001175B1/de not_active Expired
- 1978-09-07 CA CA310,803A patent/CA1096870A/en not_active Expired
- 1978-09-13 DK DK403878A patent/DK149625C/da not_active IP Right Cessation
- 1978-09-13 JP JP11287178A patent/JPS5492974A/ja active Pending
-
1980
- 1980-08-11 US US06/177,305 patent/US4357333A/en not_active Expired - Lifetime
Also Published As
Publication number | Publication date |
---|---|
DK403878A (da) | 1979-03-15 |
US4357333A (en) | 1982-11-02 |
GB1573186A (en) | 1980-08-20 |
IE47249B1 (en) | 1984-01-25 |
DK149625B (da) | 1986-08-18 |
EP0001175A1 (de) | 1979-03-21 |
EP0001175B1 (de) | 1981-04-15 |
CA1096870A (en) | 1981-03-03 |
AU516318B2 (en) | 1981-05-28 |
ZA784709B (en) | 1980-03-26 |
JPS5492974A (en) | 1979-07-23 |
IE781728L (en) | 1979-03-14 |
AU3917178A (en) | 1980-02-28 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
PBP | Patent lapsed |