DK146541C - METHOD OF ANALOGUE FOR THE PREPARATION OF 4'-EPI-DAUNOMYCINE OR ITS INDIVIDUAL ALFA OR BETA ANOMERS THEREOF - Google Patents

METHOD OF ANALOGUE FOR THE PREPARATION OF 4'-EPI-DAUNOMYCINE OR ITS INDIVIDUAL ALFA OR BETA ANOMERS THEREOF

Info

Publication number
DK146541C
DK146541C DK109275A DK109275A DK146541C DK 146541 C DK146541 C DK 146541C DK 109275 A DK109275 A DK 109275A DK 109275 A DK109275 A DK 109275A DK 146541 C DK146541 C DK 146541C
Authority
DK
Denmark
Prior art keywords
daunomycine
alfa
epi
analogue
individual
Prior art date
Application number
DK109275A
Other languages
Danish (da)
Other versions
DK146541B (en
DK109275A (en
Inventor
Federico Arcamone
Aurelio Di Marco
Sergio Penco
Original Assignee
Farmaceutici Italia
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Farmaceutici Italia filed Critical Farmaceutici Italia
Publication of DK109275A publication Critical patent/DK109275A/da
Publication of DK146541B publication Critical patent/DK146541B/en
Application granted granted Critical
Publication of DK146541C publication Critical patent/DK146541C/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/20Carbocyclic rings
    • C07H15/24Condensed ring systems having three or more rings
    • C07H15/252Naphthacene radicals, e.g. daunomycins, adriamycins
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
DK109275A 1974-03-20 1975-03-18 METHOD OF ANALOGUE FOR THE PREPARATION OF 4'-EPI-DAUNOMYCINE OR ITS INDIVIDUAL ALFA OR BETA ANOMERS THEREOF DK146541C (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB1225474 1974-03-20
GB1225474A GB1457559A (en) 1974-03-20 1974-03-20 Daunomycins

Publications (3)

Publication Number Publication Date
DK109275A DK109275A (en) 1975-09-21
DK146541B DK146541B (en) 1983-10-31
DK146541C true DK146541C (en) 1984-04-09

Family

ID=10001195

Family Applications (1)

Application Number Title Priority Date Filing Date
DK109275A DK146541C (en) 1974-03-20 1975-03-18 METHOD OF ANALOGUE FOR THE PREPARATION OF 4'-EPI-DAUNOMYCINE OR ITS INDIVIDUAL ALFA OR BETA ANOMERS THEREOF

Country Status (13)

Country Link
JP (1) JPS5833880B2 (en)
AT (1) AT338419B (en)
BE (1) BE826848A (en)
CA (1) CA1046508A (en)
CH (1) CH615198A5 (en)
DE (1) DE2510926C3 (en)
DK (1) DK146541C (en)
FR (1) FR2264554B1 (en)
GB (1) GB1457559A (en)
NL (1) NL176636C (en)
SE (1) SE434843B (en)
SU (1) SU589926A3 (en)
ZA (1) ZA751687B (en)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5124317A (en) * 1985-08-02 1992-06-23 Farmitalia Carlo Erba S.P.A. Injectable ready-to-use solutions containing an antitumor anthracycline glycoside
US5977082A (en) * 1985-08-02 1999-11-02 Pharmacia & Upjohn Company Injectable ready-to-use solutions containing an antitumor anthracycline glycoside
FR2678274A1 (en) * 1991-06-25 1992-12-31 Medgenix Group Sa N-Leucylepirubicin, application as antitumour medicinal product and process for preparing it

Also Published As

Publication number Publication date
JPS50126657A (en) 1975-10-04
CH615198A5 (en) 1980-01-15
DE2510926A1 (en) 1975-09-25
NL176636C (en) 1985-05-17
GB1457559A (en) 1976-12-08
DK146541B (en) 1983-10-31
SE7503084L (en) 1975-09-21
ATA202875A (en) 1976-12-15
AT338419B (en) 1977-08-25
NL176636B (en) 1984-12-17
CA1046508A (en) 1979-01-16
ZA751687B (en) 1976-02-25
FR2264554A1 (en) 1975-10-17
NL7503079A (en) 1975-09-23
SE7503084A (en) 1975-09-22
DE2510926C3 (en) 1980-03-13
BE826848A (en) 1975-09-19
FR2264554B1 (en) 1978-07-28
AU7919775A (en) 1976-09-23
DE2510926B2 (en) 1979-07-19
SE434843B (en) 1984-08-20
SU589926A3 (en) 1978-01-25
JPS5833880B2 (en) 1983-07-22
DK109275A (en) 1975-09-21

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