DK139973B - Analogifremgangsmåde til fremstilling af s-triazolo-(4,3-a)(1,4)-benzodiazepinderivater eller syreadditionssalte deraf. - Google Patents

Analogifremgangsmåde til fremstilling af s-triazolo-(4,3-a)(1,4)-benzodiazepinderivater eller syreadditionssalte deraf.

Info

Publication number
DK139973B
DK139973B DK101170AA DK101170A DK139973B DK 139973 B DK139973 B DK 139973B DK 101170A A DK101170A A DK 101170AA DK 101170 A DK101170 A DK 101170A DK 139973 B DK139973 B DK 139973B
Authority
DK
Denmark
Prior art keywords
triazolo
preparation
acid addition
addition salts
benzodiazepine derivatives
Prior art date
Application number
DK101170AA
Other languages
Danish (da)
English (en)
Other versions
DK139973C (no
Inventor
Kanji Meguro
Yutaka Kuwada
Original Assignee
Takeda Chemical Industries Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Takeda Chemical Industries Ltd filed Critical Takeda Chemical Industries Ltd
Publication of DK139973B publication Critical patent/DK139973B/da
Application granted granted Critical
Publication of DK139973C publication Critical patent/DK139973C/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D243/00—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
    • C07D243/06—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
    • C07D243/10—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D243/14—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines
    • C07D243/16—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals
    • C07D243/18—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals substituted in position 2 by nitrogen, oxygen or sulfur atoms
    • C07D243/20—Nitrogen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
DK101170AA 1969-03-08 1970-03-02 Analogifremgangsmåde til fremstilling af s-triazolo-(4,3-a)(1,4)-benzodiazepinderivater eller syreadditionssalte deraf. DK139973B (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP44017663A JPS4837280B1 (no) 1969-03-08 1969-03-08

Publications (2)

Publication Number Publication Date
DK139973B true DK139973B (da) 1979-05-28
DK139973C DK139973C (no) 1979-10-29

Family

ID=11950078

Family Applications (1)

Application Number Title Priority Date Filing Date
DK101170AA DK139973B (da) 1969-03-08 1970-03-02 Analogifremgangsmåde til fremstilling af s-triazolo-(4,3-a)(1,4)-benzodiazepinderivater eller syreadditionssalte deraf.

Country Status (15)

Country Link
US (1) US3907820A (no)
JP (1) JPS4837280B1 (no)
AT (2) AT297707B (no)
BE (1) BE746735A (no)
CH (3) CH550812A (no)
DE (1) DE2010884C2 (no)
DK (1) DK139973B (no)
ES (1) ES377099A1 (no)
FR (1) FR2034750B1 (no)
GB (1) GB1248727A (no)
MY (1) MY7500010A (no)
NL (1) NL166023C (no)
NO (1) NO126326B (no)
PH (2) PH10048A (no)
SE (2) SE367201B (no)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3681343A (en) * 1971-05-11 1972-08-01 Upjohn Co 6-phenyl-s-triazolo{8 4,3-a{9 {8 1,4{9 {0 benzodiazepines
US3879406A (en) * 1972-07-13 1975-04-22 Hoffmann La Roche Preparation of triazolobenzodiazepines
JPS5747914B2 (no) * 1974-04-12 1982-10-13
US4588721A (en) * 1983-09-12 1986-05-13 The Upjohn Company Treatment of negative symptoms of schizophrenia
JPS6193487U (no) * 1984-11-22 1986-06-17

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3464978A (en) * 1967-04-21 1969-09-02 Hoffmann La Roche 1-substituted urea alkyl 1,2-dihydro-1,4-benzodiazepines and benzodiazepin - 2-ones
US3498973A (en) * 1967-06-19 1970-03-03 Hoffmann La Roche 2,3-dihydro-5-phenyl-1h-1,4-benzodiazepin-3-ol derivatives
US3523939A (en) * 1967-07-03 1970-08-11 Hoffmann La Roche 5-(2,6-disubstituted phenyl)-1,4-benzodiazepines and methods for their preparation

Also Published As

Publication number Publication date
CH542865A (de) 1973-11-30
BE746735A (fr) 1970-08-17
ES377099A1 (es) 1972-06-01
CH546778A (de) 1974-03-15
GB1248727A (en) 1971-10-06
JPS4837280B1 (no) 1973-11-09
SE367201B (no) 1974-05-20
FR2034750B1 (no) 1974-04-12
AT297718B (de) 1972-04-10
PH11202A (en) 1977-10-28
US3907820A (en) 1975-09-23
DE2010884C2 (de) 1982-12-09
NL166023C (nl) 1981-06-15
DK139973C (no) 1979-10-29
NL166023B (nl) 1981-01-15
CH550812A (de) 1974-06-28
NL7002884A (no) 1970-09-10
NO126326B (no) 1973-01-22
AT297707B (de) 1972-04-10
SE397832B (sv) 1977-11-21
PH10048A (en) 1976-07-27
FR2034750A1 (no) 1970-12-11
DE2010884A1 (de) 1970-12-10
MY7500010A (en) 1975-12-31

Similar Documents

Publication Publication Date Title
DK134984B (da) Analogifremgangsmåde til fremstilling af alfa-alkylaminopropiophenoner eller syreadditionssalte heraf.
DK125794B (da) Analogifremgangsmåde til fremstilling af 2,3-dichlorphenoxyeddikesyrederivater.
DK139869B (da) Analogifremgangsmåde til fremstilling af phenyl-imidazolyl-alkansyrederivater eller salte deraf.
DK129581B (da) Analogifremgangsmåde til fremstilling af substituerede N-allyl-2-arylamino-imidazolin-(2)-forbindelser eller syreadditionssalte deraf.
DK139717B (da) Analogifremgangsmåde til fremstilling af beta-aryl-2-aminoalkoxystyroler eller syreadditionssalte heraf.
DK135278B (da) Analogifremgangsmåde til fremstilling af fenoksyisopropanolaminderivater eller syreadditionssalte deraf.
DK124203B (da) Analogifremgangsmåde til fremstilling af 1,2,3,11b-tetrahydropyrido[3,4,5:m,n]thioxanthener eller syreadditionssalte deraf.
DK136526B (da) Analogifremgangsmåde til fremstilling af substituerede naphthylalkylaminer eller syreadditionssalte deraf.
DK130410B (da) Fremgangsmåde til fremstilling af substituerede N-aminoalkyl-arylaminoimidazolin-(2)-forbindelser eller syreadditionssalte deraf.
DK137382B (da) Analogifremgangsmåde til fremstilling af 2,2-diaryl-4-(4'-aryl-4'-hydroxy-piperidin)butyramider eller syreadditionssalte deraf.
DK131721B (da) Analogifremgangsmåde til fremstilling af adamantanylaminer eller 3,5,7-trimethylhomologe eller syreadditionssalte deraf.
DK129577B (da) Analogifremgangsmåde til fremstilling af phenacetylguanidiner eller syreadditionssalte deraf.
DK127116B (da) Analogifremgangsmåde til fremstilling af imidazolidinonderivater eller syreadditionssalte deraf.
DK125245B (da) Fremgangsmåde til fremstilling af γpiperidinobutyrophenonderivater eller syreadditionssalte deraf.
DK138015B (da) Fremgangsmåde til fremstilling af substituerede N-cycloalkyl-arylamino-imidazoliner-(2) eller syreadditionssalte deraf.
DK121367B (da) Analogifremgangsmåde til fremstilling af 3,3-difenylallylaminderivater eller syreadditionssalte deraf.
DK127424B (da) Analogifremgangsmåde til fremstilling af 4-aryl-1-(4,4-diarylbutyl)-4-hydroxypiperidiner eller syreadditionssalte deraf.
DK139973B (da) Analogifremgangsmåde til fremstilling af s-triazolo-(4,3-a)(1,4)-benzodiazepinderivater eller syreadditionssalte deraf.
DK125472B (da) Analogifremgangsmåde til fremstilling af pyrimidopyridazinderivater eller syreadditionssalte deraf.
DK129454B (da) Analogifremgangsmåde til fremstilling af ergonorcornin eller syreadditionssalte deraf.
DK137044B (da) Analogifremgangsmåde til fremstilling af 4,4-diphenylhexahydroazepinderivater eller syreadditionssalte deraf.
DK131727B (da) Analogifremgangsmåde til fremstilling af oxazinobenzoxaziner eller syreadditionssalte deraf.
DK127117B (da) Analogifremgangsmåde til fremstilling af imidazolidinonderivater eller syreadditionssalte deraf.
DK134023B (da) Analogifremgangsmåde til fremstilling af acyloxypiperazinylforbindelser eller syreadditionssalte deraf.
DK139943B (da) Fremgangsmåde til fremstilling af triazolo(4,3a)(1,4)benzodiazepin-5N-oxydderivater eller syreadditionssalte deraf.