DK136829B - Analogifremgangsmåde til fremstilling af 17beta-C1-8-alkoxy-3'H-cyclopropa(16alfa,17alfa)5alfa-androstano(2,3-d)isoxazoler. - Google Patents

Analogifremgangsmåde til fremstilling af 17beta-C1-8-alkoxy-3'H-cyclopropa(16alfa,17alfa)5alfa-androstano(2,3-d)isoxazoler.

Info

Publication number
DK136829B
DK136829B DK121572AA DK121572A DK136829B DK 136829 B DK136829 B DK 136829B DK 121572A A DK121572A A DK 121572AA DK 121572 A DK121572 A DK 121572A DK 136829 B DK136829 B DK 136829B
Authority
DK
Denmark
Prior art keywords
androstano
16alpha
5alpha
17alpha
cyclopropa
Prior art date
Application number
DK121572AA
Other languages
English (en)
Other versions
DK136829C (da
Inventor
Kenneth Earl Fahrenholtz
Richard Wightman Kierstead
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of DK136829B publication Critical patent/DK136829B/da
Application granted granted Critical
Publication of DK136829C publication Critical patent/DK136829C/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J75/00—Processes for the preparation of steroids in general

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Steroid Compounds (AREA)
DK121572AA 1971-03-15 1972-03-15 Analogifremgangsmåde til fremstilling af 17beta-C1-8-alkoxy-3'H-cyclopropa(16alfa,17alfa)5alfa-androstano(2,3-d)isoxazoler. DK136829B (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US12458971A 1971-03-15 1971-03-15

Publications (2)

Publication Number Publication Date
DK136829B true DK136829B (da) 1977-11-28
DK136829C DK136829C (da) 1978-06-12

Family

ID=22415750

Family Applications (1)

Application Number Title Priority Date Filing Date
DK121572AA DK136829B (da) 1971-03-15 1972-03-15 Analogifremgangsmåde til fremstilling af 17beta-C1-8-alkoxy-3'H-cyclopropa(16alfa,17alfa)5alfa-androstano(2,3-d)isoxazoler.

Country Status (13)

Country Link
US (1) US3732209A (da)
AU (1) AU468273B2 (da)
BE (1) BE780644A (da)
CA (1) CA955929A (da)
CH (1) CH579104A5 (da)
DE (1) DE2212548A1 (da)
DK (1) DK136829B (da)
FR (1) FR2130285B1 (da)
GB (1) GB1367384A (da)
IL (1) IL38964A (da)
NL (1) NL7202984A (da)
SE (1) SE380028B (da)
ZA (1) ZA721683B (da)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3980638A (en) * 1974-09-20 1976-09-14 The Upjohn Company Testosterone derivatives
US4891367A (en) * 1987-04-22 1990-01-02 Merrell Dow Pharmaceuticals Inc. 17β-(cyclopropyloxy)androst-5-en-3β-ol and related compounds useful as C17-20 lyase inhibitors
US5486511A (en) * 1993-05-25 1996-01-23 Merrell Dow Pharmaceuticals Inc. 4-amino-17β-(cyclopropyloxy)androst-4-en-3-one, 4-amino-17β-(cyclopropylamino)androst-4-en-3-one and related compounds as C17-20 lyase and 5α-reductase
WO2002048171A1 (en) 2000-12-11 2002-06-20 Akzo Nobel N.V. Methylene steroids as novel androgens

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE1240078B (de) * 1964-12-02 1967-05-11 Schering Ag Verfahren zur Herstellung von 16, 17-Methylen-delta 1,3,5(10)-oestratrien-derivaten
US3646074A (en) * 1969-11-26 1972-02-29 Searle & Co 3 17-dioxygenated 16alpha 17alpha-methano-5alpha-androstanes and unsaturated congeners

Also Published As

Publication number Publication date
IL38964A0 (en) 1972-05-30
CA955929A (en) 1974-10-08
US3732209A (en) 1973-05-08
GB1367384A (en) 1974-09-18
IL38964A (en) 1976-03-31
CH579104A5 (da) 1976-08-31
DK136829C (da) 1978-06-12
DE2212548A1 (de) 1972-09-21
BE780644A (fr) 1972-09-14
SE380028B (da) 1975-10-27
FR2130285B1 (da) 1975-06-20
AU3998072A (en) 1973-09-20
AU468273B2 (en) 1973-09-20
ZA721683B (en) 1972-12-27
FR2130285A1 (da) 1972-11-03
NL7202984A (da) 1972-09-19

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