DK1354875T3 - Ny syntesefremgangsmåde for (2S, 3aS, 7aS)-perhydroindol-2-carboxylsyre og estere heraf samt anvendelse ved syntese af perindopril - Google Patents
Ny syntesefremgangsmåde for (2S, 3aS, 7aS)-perhydroindol-2-carboxylsyre og estere heraf samt anvendelse ved syntese af perindoprilInfo
- Publication number
- DK1354875T3 DK1354875T3 DK03291157T DK03291157T DK1354875T3 DK 1354875 T3 DK1354875 T3 DK 1354875T3 DK 03291157 T DK03291157 T DK 03291157T DK 03291157 T DK03291157 T DK 03291157T DK 1354875 T3 DK1354875 T3 DK 1354875T3
- Authority
- DK
- Denmark
- Prior art keywords
- synthesis
- perhydroindole
- perindopril
- esters
- carboxylic acid
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/04—Indoles; Hydrogenated indoles
- C07D209/30—Indoles; Hydrogenated indoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to carbon atoms of the hetero ring
- C07D209/42—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Indole Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP03291157A EP1354875B1 (fr) | 2003-05-19 | 2003-05-19 | Nouveau procédé de synthèse de l'acide (2S, 3aS, 7aS)-perhydroindole-2-carboxilique et de ses esters, et application à la synthèse du perindopril |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| DK1354875T3 true DK1354875T3 (da) | 2005-03-14 |
Family
ID=28459641
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK03291157T DK1354875T3 (da) | 2003-05-19 | 2003-05-19 | Ny syntesefremgangsmåde for (2S, 3aS, 7aS)-perhydroindol-2-carboxylsyre og estere heraf samt anvendelse ved syntese af perindopril |
Country Status (10)
| Country | Link |
|---|---|
| EP (1) | EP1354875B1 (da) |
| AR (1) | AR044392A1 (da) |
| AT (1) | ATE283258T1 (da) |
| DE (1) | DE60300168T2 (da) |
| DK (1) | DK1354875T3 (da) |
| ES (1) | ES2233914T3 (da) |
| MY (1) | MY136639A (da) |
| PT (1) | PT1354875E (da) |
| SI (1) | SI1354875T1 (da) |
| WO (1) | WO2004103969A1 (da) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN100391945C (zh) * | 2005-05-31 | 2008-06-04 | 浙江大学 | 一种s-(-)-吲哚啉-2-羧酸的合成方法 |
| DK2875000T3 (da) | 2012-07-17 | 2016-10-24 | Hoffmann La Roche | Arylethynylderivater |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| NZ202903A (en) * | 1981-12-29 | 1988-01-08 | Hoechst Ag | 1-- pe pyrrol-2-yl-carboxylic acid derivatives and pharmaceutical compositions |
| FR2620703B1 (fr) * | 1987-09-17 | 1991-10-04 | Adir | Procede de synthese industrielle de l'acide perhydroindole carboxylique - 2(2s, 3as, 7as). application a la synthese de carboxyalkyl dipeptides |
-
2003
- 2003-05-19 SI SI200330011T patent/SI1354875T1/xx unknown
- 2003-05-19 PT PT03291157T patent/PT1354875E/pt unknown
- 2003-05-19 EP EP03291157A patent/EP1354875B1/fr not_active Expired - Lifetime
- 2003-05-19 AT AT03291157T patent/ATE283258T1/de active
- 2003-05-19 DE DE60300168T patent/DE60300168T2/de not_active Expired - Lifetime
- 2003-05-19 DK DK03291157T patent/DK1354875T3/da active
- 2003-05-19 ES ES03291157T patent/ES2233914T3/es not_active Expired - Lifetime
-
2004
- 2004-05-19 AR ARP040101725A patent/AR044392A1/es not_active Application Discontinuation
- 2004-05-19 MY MYPI20041884A patent/MY136639A/en unknown
- 2004-05-19 WO PCT/FR2004/001225 patent/WO2004103969A1/fr unknown
Also Published As
| Publication number | Publication date |
|---|---|
| AR044392A1 (es) | 2005-09-14 |
| PT1354875E (pt) | 2005-03-31 |
| WO2004103969A1 (fr) | 2004-12-02 |
| DE60300168D1 (de) | 2004-12-30 |
| EP1354875B1 (fr) | 2004-11-24 |
| DE60300168T2 (de) | 2005-12-01 |
| ATE283258T1 (de) | 2004-12-15 |
| SI1354875T1 (en) | 2005-02-28 |
| MY136639A (en) | 2008-11-28 |
| EP1354875A1 (fr) | 2003-10-22 |
| ES2233914T3 (es) | 2005-06-16 |
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