DK133673B - Fremgangsmåde til fremstilling af 3,4-dihydro-2(1H)-quinazolinonderivater. - Google Patents
Fremgangsmåde til fremstilling af 3,4-dihydro-2(1H)-quinazolinonderivater.Info
- Publication number
- DK133673B DK133673B DK635671AA DK635671A DK133673B DK 133673 B DK133673 B DK 133673B DK 635671A A DK635671A A DK 635671AA DK 635671 A DK635671 A DK 635671A DK 133673 B DK133673 B DK 133673B
- Authority
- DK
- Denmark
- Prior art keywords
- dihydro
- preparation
- quinazolinone derivatives
- quinazolinone
- derivatives
- Prior art date
Links
- CTOUNZIAEBIWAW-UHFFFAOYSA-N 3,4-dihydro-1h-quinazolin-2-one Chemical class C1=CC=C2NC(=O)NCC2=C1 CTOUNZIAEBIWAW-UHFFFAOYSA-N 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
- C07D239/72—Quinazolines; Hydrogenated quinazolines
- C07D239/95—Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in positions 2 and 4
- C07D239/96—Two oxygen atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP45129980A JPS4822715B1 (forum.php) | 1970-12-28 | 1970-12-28 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| DK133673B true DK133673B (da) | 1976-06-28 |
| DK133673C DK133673C (forum.php) | 1977-01-03 |
Family
ID=15023173
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK635671AA DK133673B (da) | 1970-12-28 | 1971-12-27 | Fremgangsmåde til fremstilling af 3,4-dihydro-2(1H)-quinazolinonderivater. |
Country Status (13)
| Country | Link |
|---|---|
| US (1) | US3865827A (forum.php) |
| JP (1) | JPS4822715B1 (forum.php) |
| AT (1) | AT314545B (forum.php) |
| BE (1) | BE777298A (forum.php) |
| CA (1) | CA960672A (forum.php) |
| CH (1) | CH579553A5 (forum.php) |
| DE (1) | DE2165056C3 (forum.php) |
| DK (1) | DK133673B (forum.php) |
| FR (1) | FR2120847A5 (forum.php) |
| GB (1) | GB1343668A (forum.php) |
| HU (1) | HU162888B (forum.php) |
| NL (1) | NL7117876A (forum.php) |
| SE (1) | SE391181B (forum.php) |
Families Citing this family (13)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS5815979A (ja) * | 1981-07-11 | 1983-01-29 | Kyowa Hakko Kogyo Co Ltd | 新規なピペリジン誘導体およびその製造法 |
| US6184377B1 (en) | 1997-12-15 | 2001-02-06 | Sepracor Inc. | Compositions containing N-amino- and N-hydroxy-quinazolinones and methods for preparing libraries thereof |
| US6521630B1 (en) * | 1999-08-31 | 2003-02-18 | Pfizer Inc. | Tetrahydroquinazoline-2,4-diones and therapeutic uses thereof |
| CU24130B1 (es) | 2009-12-22 | 2015-09-29 | Novartis Ag | Isoquinolinonas y quinazolinonas sustituidas |
| US8440693B2 (en) * | 2009-12-22 | 2013-05-14 | Novartis Ag | Substituted isoquinolinones and quinazolinones |
| WO2013175417A1 (en) | 2012-05-24 | 2013-11-28 | Novartis Ag | Pyrrolopyrrolidinone compounds |
| US9556180B2 (en) | 2013-01-22 | 2017-01-31 | Novartis Ag | Pyrazolo[3,4-d]pyrimidinone compounds as inhibitors of the P53/MDM2 interaction |
| US9403827B2 (en) | 2013-01-22 | 2016-08-02 | Novartis Ag | Substituted purinone compounds |
| KR20160012194A (ko) | 2013-05-27 | 2016-02-02 | 노파르티스 아게 | 이미다조피롤리디논 유도체 및 질환의 치료에서의 그의 용도 |
| JP6403761B2 (ja) | 2013-05-28 | 2018-10-10 | ノバルティス アーゲー | ピラゾロ−ピロリジン−4−オン誘導体および疾患の処置におけるその使用 |
| AU2014272695B2 (en) | 2013-05-28 | 2016-10-20 | Novartis Ag | Pyrazolo-pyrrolidin-4-one derivatives as BET inhibitors and their use in the treatment of disease |
| KR20160086930A (ko) | 2013-11-21 | 2016-07-20 | 노파르티스 아게 | 피롤로피롤론 유도체 및 bet 억제제로서의 그의 용도 |
| EP4608817A1 (en) * | 2022-10-24 | 2025-09-03 | The Regents Of The University Of California | Compounds and methods for treating cancer |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3573308A (en) * | 1969-04-03 | 1971-03-30 | Hoffmann La Roche | 3-lower alkoxy methyl-3,4-dihydro-4-hydroxy-4-aryl quinazolin-2(1h) ones and related compounds |
-
1970
- 1970-12-28 JP JP45129980A patent/JPS4822715B1/ja active Pending
-
1971
- 1971-12-13 US US207541A patent/US3865827A/en not_active Expired - Lifetime
- 1971-12-17 GB GB5873571A patent/GB1343668A/en not_active Expired
- 1971-12-23 FR FR7146365A patent/FR2120847A5/fr not_active Expired
- 1971-12-23 CA CA131,028A patent/CA960672A/en not_active Expired
- 1971-12-27 HU HUSU706A patent/HU162888B/hu unknown
- 1971-12-27 AT AT1113371A patent/AT314545B/de not_active IP Right Cessation
- 1971-12-27 NL NL7117876A patent/NL7117876A/xx unknown
- 1971-12-27 DK DK635671AA patent/DK133673B/da unknown
- 1971-12-27 SE SE7116690A patent/SE391181B/xx unknown
- 1971-12-27 BE BE777298A patent/BE777298A/xx unknown
- 1971-12-28 CH CH1906971A patent/CH579553A5/xx not_active IP Right Cessation
- 1971-12-28 DE DE2165056A patent/DE2165056C3/de not_active Expired
Also Published As
| Publication number | Publication date |
|---|---|
| HU162888B (forum.php) | 1973-04-28 |
| DE2165056B2 (de) | 1974-05-30 |
| DE2165056C3 (de) | 1975-01-23 |
| JPS4822715B1 (forum.php) | 1973-07-07 |
| FR2120847A5 (forum.php) | 1972-08-18 |
| GB1343668A (en) | 1974-01-16 |
| SE391181B (sv) | 1977-02-07 |
| DK133673C (forum.php) | 1977-01-03 |
| CA960672A (en) | 1975-01-07 |
| CH579553A5 (forum.php) | 1976-09-15 |
| DE2165056A1 (de) | 1972-07-06 |
| US3865827A (en) | 1975-02-11 |
| NL7117876A (forum.php) | 1972-06-30 |
| BE777298A (fr) | 1972-04-17 |
| AT314545B (de) | 1974-04-10 |
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