DK127727B - Fremgangsmåde til fremstilling af et 1,4-diensteroid af androstan- eller pregnanrækken og med usubstitueret 3-stilling. - Google Patents

Fremgangsmåde til fremstilling af et 1,4-diensteroid af androstan- eller pregnanrækken og med usubstitueret 3-stilling.

Info

Publication number
DK127727B
DK127727B DK218567AA DK218567A DK127727B DK 127727 B DK127727 B DK 127727B DK 218567A A DK218567A A DK 218567AA DK 218567 A DK218567 A DK 218567A DK 127727 B DK127727 B DK 127727B
Authority
DK
Denmark
Prior art keywords
diensteroid
androstane
unsubstituted
preparation
pregnane series
Prior art date
Application number
DK218567AA
Other languages
English (en)
Inventor
T Foell
R Rees
H Smith
Original Assignee
American Home Prod
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by American Home Prod filed Critical American Home Prod
Publication of DK127727B publication Critical patent/DK127727B/da

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/57—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone
    • A61K31/573—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone substituted in position 21, e.g. cortisone, dexamethasone, prednisone or aldosterone
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/565—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
    • A61K31/568—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol substituted in positions 10 and 13 by a chain having at least one carbon atom, e.g. androstanes, e.g. testosterone
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/565—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
    • A61K31/568—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol substituted in positions 10 and 13 by a chain having at least one carbon atom, e.g. androstanes, e.g. testosterone
    • A61K31/5685—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol substituted in positions 10 and 13 by a chain having at least one carbon atom, e.g. androstanes, e.g. testosterone having an oxo group in position 17, e.g. androsterone
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/565—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
    • A61K31/568—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol substituted in positions 10 and 13 by a chain having at least one carbon atom, e.g. androstanes, e.g. testosterone
    • A61K31/569—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol substituted in positions 10 and 13 by a chain having at least one carbon atom, e.g. androstanes, e.g. testosterone substituted in position 17 alpha, e.g. ethisterone
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/57—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J5/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane and substituted in position 21 by only one singly bound oxygen atom, i.e. only one oxygen bound to position 21 by a single bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J7/00—Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of two carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J75/00—Processes for the preparation of steroids in general

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Steroid Compounds (AREA)
DK218567AA 1966-04-25 1967-04-25 Fremgangsmåde til fremstilling af et 1,4-diensteroid af androstan- eller pregnanrækken og med usubstitueret 3-stilling. DK127727B (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US54480066A 1966-04-25 1966-04-25
US62246867A 1967-03-13 1967-03-13

Publications (1)

Publication Number Publication Date
DK127727B true DK127727B (da) 1973-12-24

Family

ID=27067737

Family Applications (2)

Application Number Title Priority Date Filing Date
DK218567AA DK127727B (da) 1966-04-25 1967-04-25 Fremgangsmåde til fremstilling af et 1,4-diensteroid af androstan- eller pregnanrækken og med usubstitueret 3-stilling.
DK268871AA DK128208B (da) 1966-04-25 1971-06-02 Fremgangsmåde til fremstilling af 1,4-diensteroider af androstan- eller pregnanrækken med usubstitueret 3-stilling.

Family Applications After (1)

Application Number Title Priority Date Filing Date
DK268871AA DK128208B (da) 1966-04-25 1971-06-02 Fremgangsmåde til fremstilling af 1,4-diensteroider af androstan- eller pregnanrækken med usubstitueret 3-stilling.

Country Status (12)

Country Link
US (1) US3574196A (da)
JP (1) JPS495335B1 (da)
BE (1) BE697544A (da)
CH (1) CH538459A (da)
DE (1) DE1618058B1 (da)
DK (2) DK127727B (da)
ES (1) ES339707A1 (da)
FR (2) FR1529732A (da)
GB (2) GB1192062A (da)
IL (1) IL27840A (da)
NL (1) NL6705803A (da)
SE (2) SE362073B (da)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5135936U (da) * 1974-09-06 1976-03-17
JPS5135937U (da) * 1974-09-06 1976-03-17

Also Published As

Publication number Publication date
IL27840A (en) 1972-04-27
SE342237B (da) 1972-01-31
NL6705803A (da) 1967-10-26
DK128208B (da) 1974-03-18
FR8354M (da) 1971-02-08
BE697544A (da) 1967-10-02
JPS495335B1 (da) 1974-02-06
FR1529732A (fr) 1968-06-21
CH538459A (de) 1973-06-30
SE362073B (da) 1973-11-26
GB1192062A (en) 1970-05-20
DE1793749B2 (de) 1975-07-24
ES339707A1 (es) 1968-05-16
US3574196A (en) 1971-04-06
DE1793749A1 (de) 1973-05-03
GB1192061A (en) 1970-05-20
DE1618058B1 (de) 1972-07-13

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