DK119010B - Fremgangsmåde til fremstilling af 1,3-dihydro-5-aryl-2H-1,4-benzodiazepin-2-on-4-oxider eller tilsvarende deoxyforbindelser. - Google Patents

Fremgangsmåde til fremstilling af 1,3-dihydro-5-aryl-2H-1,4-benzodiazepin-2-on-4-oxider eller tilsvarende deoxyforbindelser.

Info

Publication number
DK119010B
DK119010B DK583364AA DK583364A DK119010B DK 119010 B DK119010 B DK 119010B DK 583364A A DK583364A A DK 583364AA DK 583364 A DK583364 A DK 583364A DK 119010 B DK119010 B DK 119010B
Authority
DK
Denmark
Prior art keywords
benzodiazepin
dihydro
oxides
aryl
preparation
Prior art date
Application number
DK583364AA
Other languages
English (en)
Inventor
A Stempel
L Sternbach
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of DK119010B publication Critical patent/DK119010B/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72Quinazolines; Hydrogenated quinazolines
    • C07D239/74Quinazolines; Hydrogenated quinazolines with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, attached to ring carbon atoms of the hetero ring
    • C07D239/76N-oxides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
DK583364AA 1963-11-27 1964-11-26 Fremgangsmåde til fremstilling af 1,3-dihydro-5-aryl-2H-1,4-benzodiazepin-2-on-4-oxider eller tilsvarende deoxyforbindelser. DK119010B (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US326372A US3321467A (en) 1963-11-27 1963-11-27 3-halo-1, 4-benzodiazepin-2-ones
US369020A US3297698A (en) 1963-11-27 1964-05-20 Process for the preparation of quinazoline 3-oxides

Publications (1)

Publication Number Publication Date
DK119010B true DK119010B (da) 1970-11-02

Family

ID=26985379

Family Applications (3)

Application Number Title Priority Date Filing Date
DK583364AA DK119010B (da) 1963-11-27 1964-11-26 Fremgangsmåde til fremstilling af 1,3-dihydro-5-aryl-2H-1,4-benzodiazepin-2-on-4-oxider eller tilsvarende deoxyforbindelser.
DK583464AA DK107031C (da) 1963-11-27 1964-11-26 Fremgangsmåde til fremstilling af 2-halogenmethyl-quinazolin-3-oxider.
DK81369AA DK122960B (da) 1963-11-27 1969-02-14 Quinazolinderivater til anvendelse som mellemprodukter ved fremstillingen af 1,4-benzodiazepin-4-oxider.

Family Applications After (2)

Application Number Title Priority Date Filing Date
DK583464AA DK107031C (da) 1963-11-27 1964-11-26 Fremgangsmåde til fremstilling af 2-halogenmethyl-quinazolin-3-oxider.
DK81369AA DK122960B (da) 1963-11-27 1969-02-14 Quinazolinderivater til anvendelse som mellemprodukter ved fremstillingen af 1,4-benzodiazepin-4-oxider.

Country Status (12)

Country Link
US (2) US3321467A (da)
BE (2) BE656226A (da)
BR (2) BR6464383D0 (da)
CH (2) CH443318A (da)
DE (2) DE1795469A1 (da)
DK (3) DK119010B (da)
ES (1) ES306429A1 (da)
FR (2) FR1453248A (da)
GB (4) GB1081945A (da)
IL (6) IL22440A (da)
NL (2) NL6413591A (da)
SE (4) SE316778B (da)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL23270A (en) * 1964-04-10 1969-02-27 Hoffmann La Roche Quinazoline derivatives and process for the manufacture and conversion thereof
NL131198C (da) * 1966-01-19
US4182760A (en) * 1977-06-16 1980-01-08 E. I. Du Pont De Nemours And Company Benzophenone anti-oximes, diazepin-N-oxides, and their use as pharmaceutical agents and as intermediates for pharmaceutical agents
US4244730A (en) * 1979-07-02 1981-01-13 Chevron Research Company Herbicidal N-haloacetyl-2-alkyl-6-acylanilines
US4753943A (en) * 1981-09-29 1988-06-28 Chevron Research Company Algicidal and fungicidal 2-haloalkyl-3-oxo-4-substituted quinazoline

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3179656A (en) * 1965-04-20 Azepine x-oxidss
NL122319C (da) * 1961-06-20

Also Published As

Publication number Publication date
IL22440A (en) 1968-12-26
SE308317B (da) 1969-02-10
BR6464383D0 (pt) 1973-07-26
GB1081948A (en) 1967-09-06
IL29815A0 (en) 1968-06-20
IL22464A (en) 1968-04-25
DE1445913A1 (de) 1969-01-30
FR1415205A (fr) 1965-10-22
BE656251A (da) 1965-05-26
SE322783B (da) 1970-04-20
IL29814A (en) 1968-12-26
GB1081947A (en) 1967-09-06
CH443318A (de) 1967-09-15
ES306429A1 (es) 1965-05-01
NL6413744A (da) 1965-05-28
US3321467A (en) 1967-05-23
DK107031C (da) 1967-04-17
GB1081945A (en) 1967-09-06
IL29815A (en) 1969-06-25
IL29814A0 (en) 1968-06-20
BR6464771D0 (pt) 1973-08-02
DK122960B (da) 1972-05-01
BE656226A (da) 1965-05-25
CH441335A (de) 1967-08-15
FR1453248A (fr) 1966-06-03
GB1081944A (en) 1967-09-06
SE352634B (da) 1973-01-08
NL6413591A (da) 1965-05-28
SE316778B (da) 1969-11-03
DE1795469A1 (de) 1972-01-20
US3297698A (en) 1967-01-10

Similar Documents

Publication Publication Date Title
DK106552C (da) Fremgangsmåde til fremstilling af substituerede 6,7-benzomorphaner.
DK114837B (da) Fremgangsmåde til fremstilling af mitosanforbindelser.
DK121904B (da) Analogifremgangsmåde til fremstilling af spiro-(steroido-6,1'-cyclopropan)-forbindelser.
DK117957B (da) Fremgangsmåde til fremstilling af 13β-alkyl-3-oxogona-4,9,11-triener.
DK127726B (da) Analogifremgangsmåde til fremstilling af 1-halogenbenzoylaminomethyl-2-phenyl-cyclopropan-forbindelser.
DK106185C (da) Fremgangsmåde til fremstilling af 17α-acyloxy-4,6-pregnadien-20-oner.
DK119010B (da) Fremgangsmåde til fremstilling af 1,3-dihydro-5-aryl-2H-1,4-benzodiazepin-2-on-4-oxider eller tilsvarende deoxyforbindelser.
DK116511B (da) Fremgangsmåde til fremstilling af substituerede 1,4-benzodiazepinforbindelser.
DK119107B (da) Fremgangsmåde til fremstilling af 11β-hydroperoxy-3-oxo-13-alkyl-Δ<4,9>-gonadiener.
DK108004C (da) Fremgangsmåde til fremstilling af 2,6-dichlorbenzonitril.
DK121120B (da) Fremgangsmåde til fremstilling af 3-hydroxy-Δ<1,5>-androstadiener eller 3-estere eller 3-ethere deraf.
DK105592C (da) Fremgangsmåde til fremstilling af substituerede 5-fluor-pyrimidiner.
DK105471C (da) Fremgangsmåde til fremstilling af 1,4-benzodiazepin-3H-forbindelser.
DK115537B (da) Fremgangsmåde til fremstilling af 6-methyl-Δ<8,9>-ergolen-8-carboxylsyre eller lysergsyre.
DK127507B (da) Analogifremgangsmåde til fremstilling af 1,4-benzodiazepinforbindelser eller syreadditionssalte deraf.
DK106329C (da) Fremgangsmåde til fremstilling af 3,20-dioxo-19-nor-4,9,11-pregnatrien.
DK117151B (da) Fremgangsmåde til fremstilling af 3,4-dihydroxy-benzyl-alkylketonforbindelser.
DK109260C (da) Fremgangsmåde til fremstilling af 3,5-diklor-2, 6-dimetyl-4-pyridinol.
DK109895C (da) Fremgangsmåde til fremstilling af 1,3-dioxo-2-alkyl-cyclopentaner.
DK114904B (da) Fremgangsmåde til fremstilling af 3,5-diiodthyroniner.
DK108919C (da) Fremgangsmåde til fremstilling af 1,2-diaryl-4-alkyl-3,5-dioxo-pyrazolidiner eller salte deraf.
DK104173C (da) Fremgangsmåde til fremstilling af 1,2-dimetylhexahydropyridaziner eller kvaternære ammoniumforbindelser deraf.
DK105983C (da) Fremgangsmåde til fremstilling af 2-alkoxy-5-aryl-3H-1,4-benzodiazepin-4-oxider.
DK108211C (da) Fremgangsmåde til fremstilling af Δ<4,9>-estradien-3β,17-dioler eller 3-monoestere, 17-monoestere eller 3,17-diestere heraf.
DK105920C (da) Fremgangsmåde til fremstilling af 3-β-hydroxyethylimino-17 α-acyloxy-20-keto-4,6-pregnadien-(eller 1,4,6-pregnatrien)-derivater.