DE69831959D1 - Verwendung von (E)-metanicotinederivate als Analgetika - Google Patents

Verwendung von (E)-metanicotinederivate als Analgetika

Info

Publication number
DE69831959D1
DE69831959D1 DE69831959T DE69831959T DE69831959D1 DE 69831959 D1 DE69831959 D1 DE 69831959D1 DE 69831959 T DE69831959 T DE 69831959T DE 69831959 T DE69831959 T DE 69831959T DE 69831959 D1 DE69831959 D1 DE 69831959D1
Authority
DE
Germany
Prior art keywords
metanicotine
patient
analgesics
derivatives
relates
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
DE69831959T
Other languages
English (en)
Other versions
DE69831959T2 (de
Inventor
R Martin
L Damaj
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Virginia Commonwealth University
Original Assignee
Virginia Commonwealth University
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Virginia Commonwealth University filed Critical Virginia Commonwealth University
Application granted granted Critical
Publication of DE69831959D1 publication Critical patent/DE69831959D1/de
Publication of DE69831959T2 publication Critical patent/DE69831959T2/de
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4406Non condensed pyridines; Hydrogenated derivatives thereof only substituted in position 3, e.g. zimeldine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Rheumatology (AREA)
  • Pain & Pain Management (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Pyridine Compounds (AREA)
DE69831959T 1997-08-07 1998-08-07 Verwendung von (E)-metanicotinederivate als Analgetika Expired - Fee Related DE69831959T2 (de)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US908440 1997-08-07
US08/908,440 US5914337A (en) 1997-08-07 1997-08-07 Compounds and pharmaceutical compositions thereof for eliciting analgesic effects
PCT/US1998/016485 WO1999007369A1 (en) 1997-08-07 1998-08-07 Compounds and pharmaceutical compositions thereof for eliciting analgesic effects

Publications (2)

Publication Number Publication Date
DE69831959D1 true DE69831959D1 (de) 2006-03-02
DE69831959T2 DE69831959T2 (de) 2006-07-27

Family

ID=25425808

Family Applications (1)

Application Number Title Priority Date Filing Date
DE69831959T Expired - Fee Related DE69831959T2 (de) 1997-08-07 1998-08-07 Verwendung von (E)-metanicotinederivate als Analgetika

Country Status (8)

Country Link
US (2) US5914337A (de)
EP (1) EP1011672B1 (de)
AT (1) ATE306923T1 (de)
AU (1) AU8900498A (de)
DE (1) DE69831959T2 (de)
DK (1) DK1011672T3 (de)
ES (1) ES2251779T3 (de)
WO (1) WO1999007369A1 (de)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DK1056458T3 (da) * 1998-02-24 2005-08-01 Univ Wake Forest Behandling af kronisk smerte
US6232316B1 (en) 1998-06-16 2001-05-15 Targacept, Inc. Methods for treatment of CNS disorders
JP2003501416A (ja) * 1999-06-07 2003-01-14 ターガセプト,インコーポレイテッド 医薬組成物およびその使用法

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5604231A (en) * 1995-01-06 1997-02-18 Smith; Carr J. Pharmaceutical compositions for prevention and treatment of ulcerative colitis
US5616716A (en) * 1996-01-06 1997-04-01 Dull; Gary M. (3-(5-ethoxypyridin)yl)-alkenyl 1 amine compounds

Also Published As

Publication number Publication date
EP1011672B1 (de) 2005-10-19
US6117891A (en) 2000-09-12
EP1011672A4 (de) 2001-04-04
DE69831959T2 (de) 2006-07-27
ES2251779T3 (es) 2006-05-01
ATE306923T1 (de) 2005-11-15
WO1999007369A1 (en) 1999-02-18
EP1011672A1 (de) 2000-06-28
US5914337A (en) 1999-06-22
DK1011672T3 (da) 2006-02-06
AU8900498A (en) 1999-03-01

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Legal Events

Date Code Title Description
8364 No opposition during term of opposition
8339 Ceased/non-payment of the annual fee