DE602005009158D1 - Anti-hiv-chinuklidinverbindungen - Google Patents

Anti-hiv-chinuklidinverbindungen

Info

Publication number
DE602005009158D1
DE602005009158D1 DE602005009158T DE602005009158T DE602005009158D1 DE 602005009158 D1 DE602005009158 D1 DE 602005009158D1 DE 602005009158 T DE602005009158 T DE 602005009158T DE 602005009158 T DE602005009158 T DE 602005009158T DE 602005009158 D1 DE602005009158 D1 DE 602005009158D1
Authority
DE
Germany
Prior art keywords
infectivity
mammal
chinuklidinverbindungen
hiv
benzoylquinuclidine
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
DE602005009158T
Other languages
English (en)
Inventor
Laurent Lecanu
Janet Greeson
Vassilios Papadopoulos
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Georgetown University
Samaritan Pharmaceuticals Inc
Original Assignee
Georgetown University
Samaritan Pharmaceuticals Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Georgetown University, Samaritan Pharmaceuticals Inc filed Critical Georgetown University
Publication of DE602005009158D1 publication Critical patent/DE602005009158D1/de
Expired - Fee Related legal-status Critical Current
Anticipated expiration legal-status Critical

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/439Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom the ring forming part of a bridged ring system, e.g. quinuclidine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • A61P31/18Antivirals for RNA viruses for HIV
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Virology (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Immunology (AREA)
  • Engineering & Computer Science (AREA)
  • AIDS & HIV (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicinal Preparation (AREA)
DE602005009158T 2004-04-05 2005-04-01 Anti-hiv-chinuklidinverbindungen Expired - Fee Related DE602005009158D1 (de)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US55955004P 2004-04-05 2004-04-05
US59020904P 2004-07-22 2004-07-22
PCT/US2005/011372 WO2006085890A2 (en) 2004-04-05 2005-04-01 Anti-hiv quinuclidine compounds

Publications (1)

Publication Number Publication Date
DE602005009158D1 true DE602005009158D1 (de) 2008-10-02

Family

ID=36793472

Family Applications (1)

Application Number Title Priority Date Filing Date
DE602005009158T Expired - Fee Related DE602005009158D1 (de) 2004-04-05 2005-04-01 Anti-hiv-chinuklidinverbindungen

Country Status (8)

Country Link
US (1) US20080194619A1 (de)
EP (1) EP1732547B1 (de)
JP (1) JP2007531792A (de)
AT (1) ATE405263T1 (de)
AU (1) AU2005327283A1 (de)
CA (1) CA2563109A1 (de)
DE (1) DE602005009158D1 (de)
WO (1) WO2006085890A2 (de)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2012312301A1 (en) * 2011-09-22 2014-03-20 Vertex Pharmaceuticals Incorporated Compounds useful as inhibitors of choline kinase

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2527211A1 (en) * 2003-06-02 2004-12-16 Samaritan Pharmaceuticals, Inc. Anti-hiv benzamide compounds
TWI363759B (en) * 2004-04-27 2012-05-11 Glaxo Group Ltd Muscarinic acetylcholine receptor antagonists

Also Published As

Publication number Publication date
CA2563109A1 (en) 2006-08-17
EP1732547A2 (de) 2006-12-20
AU2005327283A1 (en) 2006-08-17
ATE405263T1 (de) 2008-09-15
JP2007531792A (ja) 2007-11-08
US20080194619A1 (en) 2008-08-14
EP1732547B1 (de) 2008-08-20
WO2006085890A3 (en) 2006-12-07
WO2006085890A2 (en) 2006-08-17

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Legal Events

Date Code Title Description
8364 No opposition during term of opposition
8339 Ceased/non-payment of the annual fee