DE60000969D1 - Pyrrolobenzodiazepine carboxamide vasopressin agonisten - Google Patents
Pyrrolobenzodiazepine carboxamide vasopressin agonistenInfo
- Publication number
- DE60000969D1 DE60000969D1 DE60000969T DE60000969T DE60000969D1 DE 60000969 D1 DE60000969 D1 DE 60000969D1 DE 60000969 T DE60000969 T DE 60000969T DE 60000969 T DE60000969 T DE 60000969T DE 60000969 D1 DE60000969 D1 DE 60000969D1
- Authority
- DE
- Germany
- Prior art keywords
- hydrogen
- chain alkyl
- branched chain
- alkoxyalkyl
- cycloalkyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Lifetime
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/04—Antihaemorrhagics; Procoagulants; Haemostatic agents; Antifibrinolytic agents
Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Medicinal Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Public Health (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Diabetes (AREA)
- Hematology (AREA)
- Urology & Nephrology (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US24418099A | 1999-02-04 | 1999-02-04 | |
PCT/US2000/000658 WO2000046228A2 (en) | 1999-02-04 | 2000-01-11 | Pyrrolobenzodiazepine carboxyamide vasopressin agonists |
Publications (1)
Publication Number | Publication Date |
---|---|
DE60000969D1 true DE60000969D1 (de) | 2003-01-23 |
Family
ID=22921685
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
DE60000969T Expired - Lifetime DE60000969D1 (de) | 1999-02-04 | 2000-01-11 | Pyrrolobenzodiazepine carboxamide vasopressin agonisten |
Country Status (8)
Country | Link |
---|---|
EP (1) | EP1149104B1 (de) |
JP (1) | JP2002536378A (de) |
CN (1) | CN1339037A (de) |
AT (1) | ATE229528T1 (de) |
AU (1) | AU2607300A (de) |
CA (1) | CA2358892A1 (de) |
DE (1) | DE60000969D1 (de) |
WO (1) | WO2000046228A2 (de) |
Families Citing this family (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US7138393B2 (en) * | 1998-07-24 | 2006-11-21 | Wyeth | Biologically active vasopressin agonist metabolites |
GB201005623D0 (en) | 2010-04-01 | 2010-05-19 | Vantia Ltd | New polymorph |
CN103420890B (zh) * | 2012-05-15 | 2015-06-24 | 天津药物研究院 | 3-吡咯甲酸衍生物及其制备方法和用途 |
Family Cites Families (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5516774A (en) * | 1993-07-29 | 1996-05-14 | American Cyanamid Company | Tricyclic diazepine vasopressin antagonists and oxytocin antagonists |
-
2000
- 2000-01-11 JP JP2000597298A patent/JP2002536378A/ja active Pending
- 2000-01-11 CN CN00803461A patent/CN1339037A/zh active Pending
- 2000-01-11 AT AT00904291T patent/ATE229528T1/de not_active IP Right Cessation
- 2000-01-11 CA CA002358892A patent/CA2358892A1/en not_active Abandoned
- 2000-01-11 AU AU26073/00A patent/AU2607300A/en not_active Abandoned
- 2000-01-11 WO PCT/US2000/000658 patent/WO2000046228A2/en active IP Right Grant
- 2000-01-11 EP EP00904291A patent/EP1149104B1/de not_active Expired - Lifetime
- 2000-01-11 DE DE60000969T patent/DE60000969D1/de not_active Expired - Lifetime
Also Published As
Publication number | Publication date |
---|---|
WO2000046228A3 (en) | 2000-12-14 |
JP2002536378A (ja) | 2002-10-29 |
EP1149104A2 (de) | 2001-10-31 |
AU2607300A (en) | 2000-08-25 |
EP1149104B1 (de) | 2002-12-11 |
ATE229528T1 (de) | 2002-12-15 |
CA2358892A1 (en) | 2000-08-10 |
WO2000046228A2 (en) | 2000-08-10 |
CN1339037A (zh) | 2002-03-06 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
8332 | No legal effect for de |