DE4307438A1 - Neue antiviral wirksame Pseudopeptide - Google Patents

Neue antiviral wirksame Pseudopeptide

Info

Publication number
DE4307438A1
DE4307438A1 DE4307438A DE4307438A DE4307438A1 DE 4307438 A1 DE4307438 A1 DE 4307438A1 DE 4307438 A DE4307438 A DE 4307438A DE 4307438 A DE4307438 A DE 4307438A DE 4307438 A1 DE4307438 A1 DE 4307438A1
Authority
DE
Germany
Prior art keywords
carbon atoms
chain
straight
formula
hydrogen
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Withdrawn
Application number
DE4307438A
Other languages
German (de)
English (en)
Inventor
Dieter Dr Haebich
Michael Dr Matzke
Klaus Dr Frobel
Thomas Dr Henkel
Hartwig Dr Mueller
Karl-Heinz Dr Weber
Juergen Dr Reefschlaeger
Gert Dr Streissle
Jutta Dr Hansen
Rainer Dr Neumann
Arnold Dr Paessens
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Bayer AG
Original Assignee
Bayer AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer AG filed Critical Bayer AG
Priority to DE4307438A priority Critical patent/DE4307438A1/de
Priority to AU53147/94A priority patent/AU667995B2/en
Priority to EP94101544A priority patent/EP0611776A3/de
Priority to NZ250863A priority patent/NZ250863A/xx
Priority to IL10862494A priority patent/IL108624A0/xx
Priority to CA002115532A priority patent/CA2115532A1/en
Priority to TW083101199A priority patent/TW261607B/zh
Priority to US08/196,939 priority patent/US5492896A/en
Priority to JP6039254A priority patent/JPH06271600A/ja
Priority to HU9400428A priority patent/HUT67373A/hu
Priority to CN94101549A priority patent/CN1108261A/zh
Publication of DE4307438A1 publication Critical patent/DE4307438A1/de
Withdrawn legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K5/00Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/02Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link
    • C07K5/0217Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link containing the structure -C(=O)-C-N-C(=O)-N-C-C(=O)-
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K5/00Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06Dipeptides
    • C07K5/06086Dipeptides with the first amino acid being basic
    • C07K5/06095Arg-amino acid
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K5/00Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/08Tripeptides
    • C07K5/0815Tripeptides with the first amino acid being basic
    • C07K5/0817Tripeptides with the first amino acid being basic the first amino acid being Arg
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Communicable Diseases (AREA)
  • Virology (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
DE4307438A 1993-02-15 1993-03-10 Neue antiviral wirksame Pseudopeptide Withdrawn DE4307438A1 (de)

Priority Applications (11)

Application Number Priority Date Filing Date Title
DE4307438A DE4307438A1 (de) 1993-02-15 1993-03-10 Neue antiviral wirksame Pseudopeptide
AU53147/94A AU667995B2 (en) 1993-02-15 1994-01-12 New pseudopeptides having an antiviral action
EP94101544A EP0611776A3 (de) 1993-02-15 1994-02-02 Neue antiviral wirksame Pseudopeptide.
NZ250863A NZ250863A (en) 1993-02-15 1994-02-11 Pseudopeptides, preparation and antiviral compositions
IL10862494A IL108624A0 (en) 1993-02-15 1994-02-11 Pseudopeptides, their preparation and pharmaceutical compositions containing them
CA002115532A CA2115532A1 (en) 1993-02-15 1994-02-11 Pseudopeptides having an antiviral action
TW083101199A TW261607B (xx) 1993-02-15 1994-02-14
US08/196,939 US5492896A (en) 1993-02-15 1994-02-15 Pseudopeptides having an antiviral action
JP6039254A JPH06271600A (ja) 1993-02-15 1994-02-15 抗ウイルス作用を有するシユードペプチド
HU9400428A HUT67373A (en) 1993-02-15 1994-02-15 Virucide pseudopeptides
CN94101549A CN1108261A (zh) 1993-02-15 1994-02-15 具有抗病毒作用的新的假肽

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE4304453 1993-02-15
DE4307438A DE4307438A1 (de) 1993-02-15 1993-03-10 Neue antiviral wirksame Pseudopeptide

Publications (1)

Publication Number Publication Date
DE4307438A1 true DE4307438A1 (de) 1994-08-18

Family

ID=6480445

Family Applications (1)

Application Number Title Priority Date Filing Date
DE4307438A Withdrawn DE4307438A1 (de) 1993-02-15 1993-03-10 Neue antiviral wirksame Pseudopeptide

Country Status (3)

Country Link
DE (1) DE4307438A1 (xx)
TW (1) TW261607B (xx)
ZA (1) ZA94986B (xx)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1997030075A1 (de) * 1996-02-16 1997-08-21 Bayer Aktiengesellschaft Antiviral wirksame oxim- und nitronsubstituierte pseudopeptide

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1997030075A1 (de) * 1996-02-16 1997-08-21 Bayer Aktiengesellschaft Antiviral wirksame oxim- und nitronsubstituierte pseudopeptide

Also Published As

Publication number Publication date
ZA94986B (en) 1996-06-26
TW261607B (xx) 1995-11-01

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Legal Events

Date Code Title Description
8130 Withdrawal