DE102008038220A1 - Oxadiazolderivate - Google Patents
Oxadiazolderivate Download PDFInfo
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- DE102008038220A1 DE102008038220A1 DE102008038220A DE102008038220A DE102008038220A1 DE 102008038220 A1 DE102008038220 A1 DE 102008038220A1 DE 102008038220 A DE102008038220 A DE 102008038220A DE 102008038220 A DE102008038220 A DE 102008038220A DE 102008038220 A1 DE102008038220 A1 DE 102008038220A1
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- stereoisomers
- pharmaceutically acceptable
- atoms
- acceptable salts
- compounds
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Classifications
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/06—Antihyperlipidemics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A61P35/04—Antineoplastic agents specific for metastasis
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
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- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Diabetes (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Ophthalmology & Optometry (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Cardiology (AREA)
- Biomedical Technology (AREA)
- Heart & Thoracic Surgery (AREA)
- Urology & Nephrology (AREA)
- Oncology (AREA)
- Rheumatology (AREA)
- Hospice & Palliative Care (AREA)
- Psychiatry (AREA)
- Child & Adolescent Psychology (AREA)
- Endocrinology (AREA)
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- Pain & Pain Management (AREA)
- Vascular Medicine (AREA)
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Priority Applications (9)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE102008038220A DE102008038220A1 (de) | 2008-08-18 | 2008-08-18 | Oxadiazolderivate |
| US13/059,079 US8377975B2 (en) | 2008-08-18 | 2009-07-09 | Oxadiazole derivatives for the treatment of diabetes |
| ES09777077.0T ES2444129T3 (es) | 2008-08-18 | 2009-07-09 | Derivados de oxadiazol para el tratamiento de diabetes |
| EP09777077.0A EP2313380B1 (de) | 2008-08-18 | 2009-07-09 | Oxadiazolderivate für die behandlung von diabetes |
| PCT/EP2009/004992 WO2010020305A1 (de) | 2008-08-18 | 2009-07-09 | Oxadiazolderivate für die behandlung von diabetes |
| AU2009284453A AU2009284453B2 (en) | 2008-08-18 | 2009-07-09 | Oxadiazole derivatives for treating diabetes |
| JP2011523312A JP5571665B2 (ja) | 2008-08-18 | 2009-07-09 | 糖尿病を処置するためのオキサジアゾール誘導体 |
| CA2734397A CA2734397C (en) | 2008-08-18 | 2009-07-09 | Oxadiazole derivatives for the treatment of diabetes |
| IL211267A IL211267A (en) | 2008-08-18 | 2011-02-17 | Oxadiazole derivatives and drugs and their use in the treatment of diabetes |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE102008038220A DE102008038220A1 (de) | 2008-08-18 | 2008-08-18 | Oxadiazolderivate |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| DE102008038220A1 true DE102008038220A1 (de) | 2010-02-25 |
Family
ID=41010866
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DE102008038220A Withdrawn DE102008038220A1 (de) | 2008-08-18 | 2008-08-18 | Oxadiazolderivate |
Country Status (9)
| Country | Link |
|---|---|
| US (1) | US8377975B2 (https=) |
| EP (1) | EP2313380B1 (https=) |
| JP (1) | JP5571665B2 (https=) |
| AU (1) | AU2009284453B2 (https=) |
| CA (1) | CA2734397C (https=) |
| DE (1) | DE102008038220A1 (https=) |
| ES (1) | ES2444129T3 (https=) |
| IL (1) | IL211267A (https=) |
| WO (1) | WO2010020305A1 (https=) |
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN111511723A (zh) * | 2017-08-21 | 2020-08-07 | 米可如比奥提克斯有限公司 | 用作抗菌剂的代谢稳定的n-酰基氨基噁二唑 |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP2771069A4 (en) * | 2011-10-27 | 2015-08-26 | Mayo Foundation | INHIBITION OF G-PROTEIN-COUPLED RECEPTOR-6-KINASE POLYPEPTIDE |
| DE102013226711A1 (de) * | 2013-12-19 | 2015-06-25 | Beiersdorf Ag | Verwendung von Alkylamidothiazolen in kosmetischen oder dermatologischen Zubereitungen zur Prophylaxe vor und Behandlung von sensibler Haut |
| EP3134399A4 (en) | 2014-04-21 | 2017-12-27 | Mayo Foundation for Medical Education and Research | Small molecule inhibitors of g protein coupled receptor 6 kinases polypeptides |
| US11447482B1 (en) | 2019-02-14 | 2022-09-20 | KUDA Therapeutics, Inc. | Imidazopyridine and oxazolopyridine derivatives and analogs thereof, methods of preparation thereof, methods of HIF-2A pathway inhibition, and induction of ferroptosis |
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-
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- 2008-08-18 DE DE102008038220A patent/DE102008038220A1/de not_active Withdrawn
-
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- 2009-07-09 EP EP09777077.0A patent/EP2313380B1/de not_active Not-in-force
- 2009-07-09 AU AU2009284453A patent/AU2009284453B2/en not_active Ceased
- 2009-07-09 ES ES09777077.0T patent/ES2444129T3/es active Active
- 2009-07-09 JP JP2011523312A patent/JP5571665B2/ja not_active Expired - Fee Related
- 2009-07-09 US US13/059,079 patent/US8377975B2/en not_active Expired - Fee Related
- 2009-07-09 CA CA2734397A patent/CA2734397C/en not_active Expired - Fee Related
- 2009-07-09 WO PCT/EP2009/004992 patent/WO2010020305A1/de not_active Ceased
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Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN111511723A (zh) * | 2017-08-21 | 2020-08-07 | 米可如比奥提克斯有限公司 | 用作抗菌剂的代谢稳定的n-酰基氨基噁二唑 |
Also Published As
| Publication number | Publication date |
|---|---|
| US20110139654A1 (en) | 2011-06-16 |
| CA2734397A1 (en) | 2010-02-25 |
| IL211267A0 (en) | 2011-04-28 |
| EP2313380B1 (de) | 2013-12-11 |
| US8377975B2 (en) | 2013-02-19 |
| WO2010020305A1 (de) | 2010-02-25 |
| ES2444129T3 (es) | 2014-02-24 |
| AU2009284453A1 (en) | 2010-02-25 |
| JP2012500232A (ja) | 2012-01-05 |
| CA2734397C (en) | 2016-09-20 |
| AU2009284453B2 (en) | 2014-02-20 |
| EP2313380A1 (de) | 2011-04-27 |
| JP5571665B2 (ja) | 2014-08-13 |
| IL211267A (en) | 2015-07-30 |
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