CY1113448T1 - Κυκλικες λακταμες για τη θεραπεια γλαυκωματος ή αυξημενης ενδο-οφθαλμικης πιεσης - Google Patents

Κυκλικες λακταμες για τη θεραπεια γλαυκωματος ή αυξημενης ενδο-οφθαλμικης πιεσης

Info

Publication number
CY1113448T1
CY1113448T1 CY20121101199T CY121101199T CY1113448T1 CY 1113448 T1 CY1113448 T1 CY 1113448T1 CY 20121101199 T CY20121101199 T CY 20121101199T CY 121101199 T CY121101199 T CY 121101199T CY 1113448 T1 CY1113448 T1 CY 1113448T1
Authority
CY
Cyprus
Prior art keywords
glaucoma
pressure therapy
cyclic lactams
ophthalmic pressure
increased endo
Prior art date
Application number
CY20121101199T
Other languages
English (en)
Inventor
David W Old
Original Assignee
Allergan, Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Allergan, Inc. filed Critical Allergan, Inc.
Publication of CY1113448T1 publication Critical patent/CY1113448T1/el

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D409/00Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/12Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/02Ophthalmic agents
    • A61P27/06Antiglaucoma agents or miotics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Ophthalmology & Optometry (AREA)
  • Engineering & Computer Science (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

Στο παρόν αποκαλύπτεται και περιγράφεται μια ένωση έχουσα τις θεραπευτικές μεθόδους, φάρμακα και σχετικές συνθέσεις του τύπου (Ι).
CY20121101199T 2007-05-23 2012-12-10 Κυκλικες λακταμες για τη θεραπεια γλαυκωματος ή αυξημενης ενδο-οφθαλμικης πιεσης CY1113448T1 (el)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US93977307P 2007-05-23 2007-05-23
EP08755837A EP2155733B1 (en) 2007-05-23 2008-05-19 Cyclic lactams for the treatment of glaucoma or elevated intraocular pressure

Publications (1)

Publication Number Publication Date
CY1113448T1 true CY1113448T1 (el) 2016-06-22

Family

ID=39522202

Family Applications (1)

Application Number Title Priority Date Filing Date
CY20121101199T CY1113448T1 (el) 2007-05-23 2012-12-10 Κυκλικες λακταμες για τη θεραπεια γλαυκωματος ή αυξημενης ενδο-οφθαλμικης πιεσης

Country Status (13)

Country Link
US (2) US8198315B2 (el)
EP (1) EP2155733B1 (el)
JP (1) JP5524047B2 (el)
AU (1) AU2008254717B2 (el)
BR (1) BRPI0812385A2 (el)
CA (1) CA2688897A1 (el)
CY (1) CY1113448T1 (el)
DK (1) DK2155733T3 (el)
ES (1) ES2395875T3 (el)
PL (1) PL2155733T3 (el)
PT (1) PT2155733E (el)
SI (1) SI2155733T1 (el)
WO (1) WO2008144623A1 (el)

Family Cites Families (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ATE10838T1 (de) * 1980-02-28 1985-01-15 Fujisawa Pharmaceutical Co., Ltd. 4-substituierte 2-oxoazetidin-verbindungen, verfahren zu deren herstellung und ihre verwendung zur antibiotika-herstellung.
GB2101114B (en) 1981-07-10 1985-05-22 Farmos Group Ltd Substituted imidazole derivatives and their preparation and use
US5212176A (en) 1990-06-29 1993-05-18 Abbott Laboratories R(+)-terazosin
TR200201297T2 (tr) * 1999-02-11 2002-06-21 Pfizer Products Inc. Antikanser maddeleri olarak faydalı heteroaril-ikame edilmiş kinolin-2-on türevleri.
CZ20031257A3 (cs) * 2000-11-27 2004-04-14 Pfizer Products Inc. Selektivní agonisty receptoru EP4 při léčení osteoporosy
AU2002358772B2 (en) * 2001-12-20 2008-11-20 Merck Serono Sa Pyrrolidine derivatives as prostaglandin modulators
US7141597B2 (en) * 2003-09-12 2006-11-28 Allergan, Inc. Nonsedating α-2 agonists
NL1026830C2 (nl) * 2004-08-12 2006-02-14 Frederik Dirk Petrus Wolf Vishaak.
JP5128954B2 (ja) * 2004-12-06 2013-01-23 メルク セローノ ソシエテ アノニム Dp1受容体アゴニストとして使用されるピロリジン−2−オン誘導体
US7091231B2 (en) * 2004-12-10 2006-08-15 Allergan, Inc. 12-Aryl prostaglandin analogs
RU2412933C2 (ru) 2005-03-10 2011-02-27 Аллерган, Инк. Замещенные гамма-лактамы в качестве терапевтических агентов
US7772392B2 (en) * 2005-05-06 2010-08-10 Allergan, Inc. Therapeutic substituted β-lactams
BRPI0714885B8 (pt) * 2006-07-11 2021-05-25 Allergan Inc compostos terapêuticos e seu uso
DK2160386T3 (da) * 2007-05-23 2012-08-27 Allergan Inc Terapeutiske ((phenyl)imidazolyl)methylquinolinylforbindelser
CN101868455B (zh) * 2007-10-23 2013-11-13 阿勒根公司 治疗性的取代的内酰胺
US7902247B2 (en) * 2008-01-09 2011-03-08 Allergan, Inc. Substituted-aryl-2-phenylethyl-1H-imidazole compounds as subtype selective modulators of alpha 2B and/or alpha 2C adrenergic receptors
US8063033B2 (en) * 2008-01-18 2011-11-22 Allergan, Inc. Therapeutic beta-lactams

Also Published As

Publication number Publication date
BRPI0812385A2 (pt) 2019-09-24
DK2155733T3 (da) 2012-10-29
CA2688897A1 (en) 2008-11-23
AU2008254717B2 (en) 2014-06-05
US8383646B2 (en) 2013-02-26
US20100190823A1 (en) 2010-07-29
US20100160407A1 (en) 2010-06-24
ES2395875T3 (es) 2013-02-15
EP2155733A1 (en) 2010-02-24
SI2155733T1 (sl) 2012-12-31
AU2008254717A1 (en) 2008-11-27
JP5524047B2 (ja) 2014-06-18
EP2155733B1 (en) 2012-09-26
PL2155733T3 (pl) 2013-02-28
JP2010528030A (ja) 2010-08-19
US8198315B2 (en) 2012-06-12
PT2155733E (pt) 2013-01-07
WO2008144623A1 (en) 2008-11-27

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