CS44191A3 - Derivative of 1-pyridylimidazole and process for preparing and use thereof - Google Patents
Derivative of 1-pyridylimidazole and process for preparing and use thereofInfo
- Publication number
- CS44191A3 CS44191A3 CS91441A CS44191A CS44191A3 CS 44191 A3 CS44191 A3 CS 44191A3 CS 91441 A CS91441 A CS 91441A CS 44191 A CS44191 A CS 44191A CS 44191 A3 CS44191 A3 CS 44191A3
- Authority
- CS
- Czechoslovakia
- Prior art keywords
- pyridylimidazole
- derivative
- preparing
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/64—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms, e.g. histidine
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/66—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D233/84—Sulfur atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
- C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
- C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP17313590 | 1990-06-29 | ||
| JP23543990 | 1990-09-04 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| CS44191A3 true CS44191A3 (en) | 1992-02-19 |
| CZ279634B6 CZ279634B6 (cs) | 1995-05-17 |
Family
ID=26495230
Country Status (14)
| Country | Link |
|---|---|
| US (2) | US5153215A (cs) |
| EP (2) | EP0464979B1 (cs) |
| KR (2) | KR920000745A (cs) |
| AU (2) | AU633183B2 (cs) |
| BR (2) | BR9100662A (cs) |
| CA (2) | CA2036148A1 (cs) |
| CZ (2) | CZ279536B6 (cs) |
| DE (2) | DE69103230T2 (cs) |
| ES (2) | ES2057754T3 (cs) |
| HU (2) | HU206951B (cs) |
| IL (2) | IL97278A0 (cs) |
| MY (2) | MY104627A (cs) |
| SK (1) | SK278039B6 (cs) |
| YU (2) | YU30491A (cs) |
Families Citing this family (34)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| KR910021381A (ko) * | 1990-02-20 | 1991-12-20 | 모리 히데오 | 4-3급 부틸이미다졸 유도체, 및 이의 제조방법 및 용도 |
| CA2036148A1 (en) * | 1990-06-29 | 1991-12-30 | Hiroki Tomioka | A 1-phenylimidazole derivative and its production and use |
| US5252590A (en) * | 1991-06-28 | 1993-10-12 | Sumitomo Chemical Company, Limited | 1-pyridylimidazole derivative |
| EP0599183A1 (en) * | 1992-11-25 | 1994-06-01 | Rhone-Poulenc Agrochimie | Manufacturing of pesticides and intermediates |
| JP3715994B2 (ja) * | 1993-12-21 | 2005-11-16 | 住友化学株式会社 | 害虫防除剤 |
| US6413542B1 (en) | 1996-03-29 | 2002-07-02 | Merial | Direct pour-on antiparasitic skin solution and methods for treating, preventing and controlling myasis |
| US6733767B2 (en) * | 1998-03-19 | 2004-05-11 | Merck & Co., Inc. | Liquid polymeric compositions for controlled release of bioactive substances |
| US6787342B2 (en) | 2000-02-16 | 2004-09-07 | Merial Limited | Paste formulations |
| US20040077703A1 (en) * | 2002-10-02 | 2004-04-22 | Soll Mark D. | Nodulisporic acid derivative spot-on formulations for combating parasites |
| US7262214B2 (en) | 2003-02-26 | 2007-08-28 | Merial Limited | 1-N-arylpyrazole derivatives in prevention of arthropod-borne and mosquito-borne diseases |
| US7531186B2 (en) * | 2003-12-17 | 2009-05-12 | Merial Limited | Topical formulations comprising 1-N-arylpyrazole derivatives and amitraz |
| US20050234119A1 (en) * | 2004-04-16 | 2005-10-20 | Soll Mark D | Antiparasitical agents and methods for treating, preventing and controlling external parasites in animals |
| US8362086B2 (en) | 2005-08-19 | 2013-01-29 | Merial Limited | Long acting injectable formulations |
| AU2007269584B2 (en) * | 2006-07-05 | 2012-05-03 | Boehringer Ingelheim Animal Health USA Inc. | 1-aryl-5-alkyl pyrazole derivative compounds, processes of making and methods of using thereof |
| US8877791B2 (en) * | 2006-08-04 | 2014-11-04 | Beth Israel Deaconess Medical Center, Inc. | Inhibitors of pyruvate kinase and methods of treating disease |
| CN102271672B (zh) | 2008-11-19 | 2015-02-04 | 梅里亚有限公司 | 用于治疗寄生物感染的包含单独的或与甲脒组合的1-芳基吡唑的组合物 |
| US9173728B2 (en) | 2008-11-19 | 2015-11-03 | Merial Inc. | Multi-cavity container having offset indentures for dispensing fluids |
| CN102448951B (zh) * | 2009-04-06 | 2017-05-10 | 安吉奥斯医药品有限公司 | 丙酮酸激酶m2调节剂、治疗组合物和相关使用方法 |
| EP2427441B1 (en) | 2009-05-04 | 2016-12-14 | Agios Pharmaceuticals, Inc. | Pkm2 activators for use in the treatment of cancer |
| AR077292A1 (es) | 2009-06-29 | 2011-08-17 | Agios Pharmaceuticals Inc | Derivados de piperazin - quinolin sulfonamidas y composiciones farmaceuticas |
| CA2766873C (en) | 2009-06-29 | 2018-08-21 | Agios Pharmaceuticals, Inc. | Therapeutic compositions and related methods of use |
| WO2011075592A1 (en) | 2009-12-17 | 2011-06-23 | Merial Limited | Compositions comprising macrocyclic lactone compounds and spirodioxepinoindoles |
| UA108641C2 (uk) | 2010-04-02 | 2015-05-25 | Паразитицидна композиція, яка містить чотири активних агенти, та спосіб її застосування | |
| EP2651898B1 (en) | 2010-12-17 | 2015-12-09 | Agios Pharmaceuticals, Inc. | Novel n-(4-(azetidine-1-carbonyl)phenyl)-(hetero-)arylsulfonamide derivatives as pyruvate kinase m2 (pmk2) modulators |
| US9328077B2 (en) | 2010-12-21 | 2016-05-03 | Agios Pharmaceuticals, Inc | Bicyclic PKM2 activators |
| TWI549947B (zh) | 2010-12-29 | 2016-09-21 | 阿吉歐斯製藥公司 | 治療化合物及組成物 |
| HUE065700T2 (hu) | 2011-05-03 | 2024-06-28 | Agios Pharmaceuticals Inc | Piruvát-kináz aktivátorok terápiában történõ alkalmazásra |
| WO2012151440A1 (en) | 2011-05-03 | 2012-11-08 | Agios Pharmaceuticals, Inc. | Pyruvate kinase activators for use for increasing lifetime of the red blood cells and treating anemia |
| KR102066757B1 (ko) | 2011-11-17 | 2020-01-15 | 뵈링거 잉겔하임 애니멀 헬스 유에스에이 인코포레이티드 | 아릴 피라졸 및 치환된 이미다졸을 함유하는 조성물, 그의 방법 및 용도 |
| JO3626B1 (ar) | 2012-02-23 | 2020-08-27 | Merial Inc | تركيبات موضعية تحتوي على فيبرونيل و بيرميثرين و طرق استخدامها |
| TWI579274B (zh) | 2012-04-20 | 2017-04-21 | 龍馬躍公司 | 製備1-芳基-5-烷基吡唑化合物的改良方法 |
| WO2014139144A1 (en) | 2013-03-15 | 2014-09-18 | Agios Pharmaceuticals, Inc. | Therapeutic compounds and compositions |
| EP3211998B1 (en) | 2014-10-31 | 2021-04-07 | Boehringer Ingelheim Animal Health USA Inc. | Parasiticidal composition comprising fipronil |
| PL3307271T3 (pl) | 2015-06-11 | 2024-02-05 | Agios Pharmaceuticals, Inc. | Sposoby stosowania aktywatorów kinazy pirogronianowej |
Family Cites Families (14)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3940484A (en) * | 1971-12-07 | 1976-02-24 | The Boots Company Limited | Insecticidal compositions and methods of combatting insects using substituted imidazoles |
| US4048188A (en) * | 1971-12-07 | 1977-09-13 | The Boots Company Limited | 1-Carbonamido imidazoles |
| GB1408877A (en) * | 1971-12-07 | 1975-10-08 | Boots Co Ltd | Substituted imidazoles and their use as pesticides |
| US3996366A (en) * | 1973-11-19 | 1976-12-07 | The Boots Company Limited | Thio derivatives of imidazol-1-yl carboxamides |
| US4301169A (en) * | 1978-11-14 | 1981-11-17 | Eisai Co., Ltd. | Novel imidazole compound and anti-depressing agent containing the same |
| US4600430A (en) * | 1985-02-22 | 1986-07-15 | Eli Lilly And Company | Pyridinylimidazolidinone compounds |
| US4634711A (en) * | 1985-08-02 | 1987-01-06 | Smithkline Beckman Corporation | Pyridylalkyl imidazole-2-thiols |
| DE3614364A1 (de) * | 1986-04-28 | 1987-10-29 | Hoechst Ag | 1-phenyl-imidazolverbindungen, verfahren zu ihrer herstellung und ihre verwendung als wachstumsregulatoren |
| CA1334092C (en) * | 1986-07-11 | 1995-01-24 | David John Carini | Angiotensin ii receptor blocking imidazoles |
| FI91754C (fi) * | 1986-12-02 | 1994-08-10 | Tanabe Seiyaku Co | Analogiamenetelmä lääkeaineena käyttökelpoisen imidatsolijohdannaisen valmistamiseksi |
| DE3811574A1 (de) * | 1988-03-31 | 1989-10-19 | Schering Ag | N-substituierte imidazole, verfahren zu ihrer herstellung sowie ihre verwendung in arzneimitteln |
| CA2015366C (en) * | 1989-05-05 | 2001-09-11 | Rhone-Poulenc Agrochimie | Pesticidal 1-arylimidazoles |
| KR910021381A (ko) * | 1990-02-20 | 1991-12-20 | 모리 히데오 | 4-3급 부틸이미다졸 유도체, 및 이의 제조방법 및 용도 |
| CA2036148A1 (en) * | 1990-06-29 | 1991-12-30 | Hiroki Tomioka | A 1-phenylimidazole derivative and its production and use |
-
1991
- 1991-02-12 CA CA002036148A patent/CA2036148A1/en not_active Abandoned
- 1991-02-12 CA CA002036147A patent/CA2036147A1/en not_active Abandoned
- 1991-02-18 KR KR1019910002563A patent/KR920000745A/ko not_active Withdrawn
- 1991-02-18 MY MYPI91000254A patent/MY104627A/en unknown
- 1991-02-18 KR KR1019910002564A patent/KR920000729A/ko not_active Withdrawn
- 1991-02-18 MY MYPI91000253A patent/MY104626A/en unknown
- 1991-02-19 BR BR919100662A patent/BR9100662A/pt unknown
- 1991-02-19 DE DE69103230T patent/DE69103230T2/de not_active Expired - Fee Related
- 1991-02-19 EP EP91301290A patent/EP0464979B1/en not_active Expired - Lifetime
- 1991-02-19 EP EP91301291A patent/EP0464980B1/en not_active Expired - Lifetime
- 1991-02-19 IL IL97278A patent/IL97278A0/xx unknown
- 1991-02-19 DE DE69103231T patent/DE69103231T2/de not_active Expired - Fee Related
- 1991-02-19 HU HU91549A patent/HU206951B/hu not_active IP Right Cessation
- 1991-02-19 IL IL9727991A patent/IL97279A/en not_active IP Right Cessation
- 1991-02-19 ES ES91301290T patent/ES2057754T3/es not_active Expired - Lifetime
- 1991-02-19 ES ES91301291T patent/ES2057755T3/es not_active Expired - Lifetime
- 1991-02-19 HU HU91548A patent/HUT58058A/hu unknown
- 1991-02-19 BR BR919100663A patent/BR9100663A/pt unknown
- 1991-02-20 US US07/658,326 patent/US5153215A/en not_active Expired - Fee Related
- 1991-02-20 SK SK440-91A patent/SK278039B6/sk unknown
- 1991-02-20 YU YU30491A patent/YU30491A/sh unknown
- 1991-02-20 CZ CS91440A patent/CZ279536B6/cs unknown
- 1991-02-20 AU AU71186/91A patent/AU633183B2/en not_active Ceased
- 1991-02-20 YU YU30391A patent/YU30391A/sh unknown
- 1991-02-20 US US07/658,324 patent/US5122530A/en not_active Expired - Fee Related
- 1991-02-20 CZ CS91441A patent/CZ279634B6/cs unknown
- 1991-02-20 AU AU71188/91A patent/AU633184B2/en not_active Ceased
Also Published As
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| CS44191A3 (en) | Derivative of 1-pyridylimidazole and process for preparing and use thereof | |
| HU911789D0 (en) | Process for producing derivatives of triazolo-triazine and pyrazolo-triazine | |
| HU911443D0 (en) | Process for the production of medical preparations containing pravastaine and fibrinous-acid derivatives | |
| CS330891A3 (en) | Mirroring article and process for preparing thereof | |
| HU911502D0 (en) | Process for separing enanthiomers of cimaterole and for preparing pharmaceutical preparatives and performance raising ones containing cimaterole | |
| HU9400478D0 (en) | Process for the preparation of beta-phenylisoserine derivatives and use thereof | |
| GB2240104B (en) | New arylvinylamide derivatives and process for their preparation | |
| YU236989A (en) | Derivatives of 2-iminobenzothiazoline and process for obtaining thereof | |
| HU9802965D0 (en) | Iminothiazolidine intermediers and process for their preparation | |
| EP0483597A3 (en) | Process of preparation of carebastin | |
| GB9120628D0 (en) | Pyrrolobenzoxazine derivatives and process for preparation thereof | |
| EP0457730A3 (en) | Process for preparation of thioderivatives of alkylhydroxyanilinotriazine | |
| ZA933899B (en) | Thienothiazine derivatives process for their preparation and their use | |
| CS199791A3 (en) | Aminodiole derivatives and process for preparing thereof | |
| ZA911927B (en) | Labdanes and process for their preparation | |
| HUT67274A (en) | Process for producing of tetrahydroindenoindoles and farmaceutical composition comprising them | |
| CS270091A3 (en) | Cement of spherical-silicate type and process for preparing thereof | |
| YU51790A (en) | Triazinic derivative and process for obtaining | |
| HU911086D0 (en) | Process for the production and use of 2-dezoxy-d-treo-pentofluoranozides and intermediers thereof | |
| EP0450180A3 (en) | Process for the preparation of aminoethanol derivatives | |
| CS339791A3 (en) | Aerosol preparation and process for preparing thereof | |
| HU913159D0 (en) | Process for the production of 3-piperazino-sydnonymine derivatives and medical preparations containing them | |
| HU900888D0 (en) | Process for preparation of 1-arylsulfonyl-pyrrolidin-2-thion and 1-arylsulfonyl-piperidin-2-thion derivatives | |
| CS270391A3 (en) | Novel 5-benzyl-substituted benzimidazoline-2-thione derivatives and process for preparing thereof | |
| YU83090A (en) | Process for preparing derivatives of glycerophospholine and glycerophosphoethanolamine |