CS199274B2 - Process for the asymetric concersion of 2-deutero-3-fluor-l-alanine into corresponding d-isomer - Google Patents

Process for the asymetric concersion of 2-deutero-3-fluor-l-alanine into corresponding d-isomer Download PDF

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Publication number
CS199274B2
CS199274B2 CS761182A CS118276A CS199274B2 CS 199274 B2 CS199274 B2 CS 199274B2 CS 761182 A CS761182 A CS 761182A CS 118276 A CS118276 A CS 118276A CS 199274 B2 CS199274 B2 CS 199274B2
Authority
CS
Czechoslovakia
Prior art keywords
deutero
alanine
fluoro
isomer
acid
Prior art date
Application number
CS761182A
Other languages
Czech (cs)
English (en)
Inventor
Donald F Reinhold
Original Assignee
Merck & Co Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US05/552,474 external-priority patent/US3950411A/en
Application filed by Merck & Co Inc filed Critical Merck & Co Inc
Publication of CS199274B2 publication Critical patent/CS199274B2/cs

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C247/00Compounds containing azido groups
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C265/00Derivatives of isocyanic acid
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C53/00Saturated compounds having only one carboxyl group bound to an acyclic carbon atom or hydrogen
    • C07C53/15Saturated compounds having only one carboxyl group bound to an acyclic carbon atom or hydrogen containing halogen
    • C07C53/19Acids containing three or more carbon atoms
    • C07C53/21Acids containing three or more carbon atoms containing fluorine
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C59/00Compounds having carboxyl groups bound to acyclic carbon atoms and containing any of the groups OH, O—metal, —CHO, keto, ether, groups, groups, or groups
    • C07C59/185Saturated compounds having only one carboxyl group and containing keto groups
    • C07C59/19Pyruvic acid

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
CS761182A 1975-02-24 1976-02-23 Process for the asymetric concersion of 2-deutero-3-fluor-l-alanine into corresponding d-isomer CS199274B2 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US05/552,474 US3950411A (en) 1972-02-03 1975-02-24 Processes for asymmetric conversion of 3-fluoro-L-alanine and 2-deutero-3-fluoro-L-alanine to their D-isomers

Publications (1)

Publication Number Publication Date
CS199274B2 true CS199274B2 (en) 1980-07-31

Family

ID=24205490

Family Applications (1)

Application Number Title Priority Date Filing Date
CS761182A CS199274B2 (en) 1975-02-24 1976-02-23 Process for the asymetric concersion of 2-deutero-3-fluor-l-alanine into corresponding d-isomer

Country Status (21)

Country Link
JP (1) JPS51110513A (enrdf_load_stackoverflow)
AR (1) AR207277A1 (enrdf_load_stackoverflow)
AU (1) AU500536B2 (enrdf_load_stackoverflow)
CA (1) CA1045157A (enrdf_load_stackoverflow)
CH (1) CH620194A5 (enrdf_load_stackoverflow)
CS (1) CS199274B2 (enrdf_load_stackoverflow)
DE (1) DE2607252A1 (enrdf_load_stackoverflow)
DK (1) DK55976A (enrdf_load_stackoverflow)
ES (1) ES445381A1 (enrdf_load_stackoverflow)
FI (1) FI760302A7 (enrdf_load_stackoverflow)
FR (1) FR2301513A1 (enrdf_load_stackoverflow)
GB (1) GB1488332A (enrdf_load_stackoverflow)
GR (1) GR59306B (enrdf_load_stackoverflow)
HU (1) HU173362B (enrdf_load_stackoverflow)
IE (1) IE43351B1 (enrdf_load_stackoverflow)
NL (1) NL7601511A (enrdf_load_stackoverflow)
NO (1) NO760448L (enrdf_load_stackoverflow)
PT (1) PT64805B (enrdf_load_stackoverflow)
SE (1) SE7601423L (enrdf_load_stackoverflow)
YU (1) YU41876A (enrdf_load_stackoverflow)
ZA (1) ZA761045B (enrdf_load_stackoverflow)

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3880922A (en) * 1972-02-03 1975-04-29 Merck & Co Inc Process for preparing 3-fluoro-D-alanine by asymmetric rearrangement of 2-(azidocarbonyl)-3-fluoro-propionic ester or nitrile

Also Published As

Publication number Publication date
DK55976A (da) 1976-08-25
FR2301513A1 (fr) 1976-09-17
AR207277A1 (es) 1976-09-22
YU41876A (en) 1982-02-28
FI760302A7 (enrdf_load_stackoverflow) 1976-08-25
HU173362B (hu) 1979-04-28
NO760448L (enrdf_load_stackoverflow) 1976-08-25
PT64805A (en) 1976-03-01
AU1117876A (en) 1977-08-25
SE7601423L (sv) 1976-08-25
DE2607252A1 (de) 1976-09-02
ES445381A1 (es) 1977-06-01
GR59306B (en) 1977-12-12
CH620194A5 (en) 1980-11-14
NL7601511A (nl) 1976-08-26
AU500536B2 (en) 1979-05-24
IE43351B1 (en) 1981-02-11
CA1045157A (en) 1978-12-26
IE43351L (en) 1976-08-21
ZA761045B (en) 1977-09-28
GB1488332A (en) 1977-10-12
JPS51110513A (enrdf_load_stackoverflow) 1976-09-30
FR2301513B1 (enrdf_load_stackoverflow) 1979-02-02
PT64805B (en) 1978-02-06

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