CS127784A2 - Zpusob vyroby 2 amino 1,5 ( 6 ) substituovanych benzimidazolu - Google Patents

Zpusob vyroby 2 amino 1,5 ( 6 ) substituovanych benzimidazolu

Info

Publication number
CS127784A2
CS127784A2 CS841277A CS127784A CS127784A2 CS 127784 A2 CS127784 A2 CS 127784A2 CS 841277 A CS841277 A CS 841277A CS 127784 A CS127784 A CS 127784A CS 127784 A2 CS127784 A2 CS 127784A2
Authority
CS
Czechoslovakia
Prior art keywords
amino
production
substituted
substituted benzimidazole
water
Prior art date
Application number
CS841277A
Other languages
Czech (cs)
English (en)
Inventor
James H Wikel
Original Assignee
Lilly Co Eli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lilly Co Eli filed Critical Lilly Co Eli
Publication of CS127784A2 publication Critical patent/CS127784A2/cs

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D235/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
    • C07D235/02Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
    • C07D235/04Benzimidazoles; Hydrogenated benzimidazoles
    • C07D235/24Benzimidazoles; Hydrogenated benzimidazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
    • C07D235/28Sulfur atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D235/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
    • C07D235/02Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
    • C07D235/04Benzimidazoles; Hydrogenated benzimidazoles
    • C07D235/24Benzimidazoles; Hydrogenated benzimidazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
    • C07D235/30Nitrogen atoms not forming part of a nitro radical
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/04Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Macromolecular Compounds Obtained By Forming Nitrogen-Containing Linkages In General (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Solid-Sorbent Or Filter-Aiding Compositions (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
CS841277A 1982-04-08 1983-04-08 Zpusob vyroby 2 amino 1,5 ( 6 ) substituovanych benzimidazolu CS127784A2 (cs)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US06/366,883 US4434288A (en) 1982-04-08 1982-04-08 Preparation of substituted 1-thiazinyl or 1-thiazolyl-2-aminobenzimidazoles

Publications (1)

Publication Number Publication Date
CS127784A2 true CS127784A2 (cs) 1984-12-14

Family

ID=23444984

Family Applications (2)

Application Number Title Priority Date Filing Date
CS832539A CS253983A2 (en) 1982-04-08 1983-04-08 Zpusob vyroby 2 amino 1,5 ( 6 ) substituovanych benzimidazolu
CS841277A CS127784A2 (cs) 1982-04-08 1983-04-08 Zpusob vyroby 2 amino 1,5 ( 6 ) substituovanych benzimidazolu

Family Applications Before (1)

Application Number Title Priority Date Filing Date
CS832539A CS253983A2 (en) 1982-04-08 1983-04-08 Zpusob vyroby 2 amino 1,5 ( 6 ) substituovanych benzimidazolu

Country Status (21)

Country Link
US (1) US4434288A (ja)
EP (1) EP0091794B1 (ja)
JP (1) JPS58188866A (ja)
KR (1) KR860001582B1 (ja)
AT (1) ATE38986T1 (ja)
CA (1) CA1187874A (ja)
CS (2) CS253983A2 (ja)
DD (1) DD209623A5 (ja)
DE (1) DE3378578D1 (ja)
DK (1) DK152983A (ja)
ES (1) ES8405376A1 (ja)
FI (1) FI831192L (ja)
GB (1) GB2118550B (ja)
GR (1) GR78170B (ja)
HU (1) HU193501B (ja)
IE (1) IE54836B1 (ja)
IL (1) IL68298A (ja)
PL (1) PL241386A1 (ja)
PT (1) PT76500B (ja)
RO (1) RO86853B (ja)
SU (1) SU1189338A3 (ja)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4435418A (en) * 1982-12-13 1984-03-06 Smithkline Beckman Corporation 5-Phenylethenylbenzimidazoles
JPS62221672A (ja) * 1986-03-20 1987-09-29 Nippon Tokushu Noyaku Seizo Kk 新規スルホニルアゾ−ル
US5545653A (en) * 1995-06-07 1996-08-13 Eli Lilly And Company Anti-viral compounds
US5693661A (en) * 1995-06-07 1997-12-02 Eli Lilly And Company Anti-viral compounds
AU3212897A (en) * 1996-06-05 1998-01-05 Eli Lilly And Company Anti-viral compounds
US5891874A (en) * 1996-06-05 1999-04-06 Eli Lilly And Company Anti-viral compound
US5821242A (en) * 1996-06-06 1998-10-13 Eli Lilly And Company Anti-viral compounds
AU741772B2 (en) 1997-02-25 2001-12-06 Government Of The United States Of America, As Represented By The Secretary Of The Department Of Health And Human Services, The Substituted benzimidazoles as non-nucleoside inhibitors of reverse transcriptase
AU7715198A (en) * 1997-06-04 1998-12-21 Eli Lilly And Company Anti-viral compounds
US10292390B2 (en) 2011-11-04 2019-05-21 Wisconsin Alumni Research Foundation Inhibition and dispersion of bacterial biofilms with 2-aminobenzimidazole derivatives
CN108997158B (zh) * 2018-07-16 2020-12-15 青岛科技大学 一种实现二取代酰胺与二苯基甲酮偶联的方法

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4243813A (en) * 1974-07-01 1981-01-06 Eli Lilly And Company Substituted 1-sulfonylbenzimidazoles
US4018790A (en) * 1975-05-08 1977-04-19 Eli Lilly And Company Substituted 1-sulfonylbenzimidazoles
US4174454A (en) * 1975-08-28 1979-11-13 Eli Lilly And Company Alkylidenylmethyl-substituted 1-sulfonylbenzimidazoles
NZ181789A (en) * 1975-08-28 1979-01-11 Lilly Co Eli 5(6)-substituted-1-hydrocarbylulphanyl-2-amino-bezimidazoles
CA1076582A (en) * 1975-10-28 1980-04-29 Charles J. Paget Antiviral thiazolinyl or thiazinyl ketobenzimidazoles
US4008243A (en) * 1975-11-19 1977-02-15 Eli Lilly And Company Antiviral thiazolinyl or thiazinyl benzimidazole esters
US4118573A (en) * 1975-11-24 1978-10-03 Eli Lilly And Company Substituted 1-sulfonylbenzimidazoles

Also Published As

Publication number Publication date
US4434288A (en) 1984-02-28
FI831192A0 (fi) 1983-04-08
DK152983D0 (da) 1983-04-06
PL241386A1 (en) 1983-11-21
DD209623A5 (de) 1984-05-16
DK152983A (da) 1983-10-09
IE54836B1 (en) 1990-02-28
CS253983A2 (en) 1984-12-14
ES521319A0 (es) 1984-06-01
IE830795L (en) 1983-10-08
ES8405376A1 (es) 1984-06-01
RO86853A (ro) 1985-05-20
RO86853B (ro) 1985-05-31
PT76500A (en) 1983-05-01
JPS58188866A (ja) 1983-11-04
FI831192L (fi) 1983-10-09
SU1189338A3 (ru) 1985-10-30
IL68298A (en) 1986-09-30
ATE38986T1 (de) 1988-12-15
EP0091794A1 (en) 1983-10-19
EP0091794B1 (en) 1988-11-30
PT76500B (en) 1986-02-06
CA1187874A (en) 1985-05-28
KR840004411A (ko) 1984-10-15
KR860001582B1 (ko) 1986-10-10
HU193501B (en) 1987-10-28
GB2118550B (en) 1985-08-29
GB2118550A (en) 1983-11-02
GR78170B (ja) 1984-09-26
DE3378578D1 (en) 1989-01-05

Similar Documents

Publication Publication Date Title
PT73982B (en) Process for preparing 3-aryloxy-3-phenylpropylamines
ATE20459T1 (de) Verfahren zur herstellung von kaliumtetrafluoroaluminat.
CS127784A2 (cs) Zpusob vyroby 2 amino 1,5 ( 6 ) substituovanych benzimidazolu
MX160738A (es) Un procedimiento mejorado para recuperar oxido de etileno de soluciones acuosas
ES523494A0 (es) Procedimiento para la obtencion de poliaminas con grupos amino primarios.
ES537401A0 (es) Un procedimiento para producir derivados de penem
ATE31309T1 (de) Verfahren zur herstellung von 4-hydroxy-2-methyln-2-pyridyl-2h-1,2-benzothiazin-3-carboxamid 1,1- dioxid.
DK467681A (da) Phosphonohydroxyacetonitril og dens salte fremgangsmaade til dens fremstilling og dens anvendelse som mellemprodukt til frestilling af phosphonohydroxyeddikesyre
BR8402512A (pt) Processo para a producao de um clorato de metal alcalino
DK218686D0 (da) Fremgangsmaade til fremstilling af 6-amino-3-hydrazinopyridazinderivater
DE3762967D1 (de) Verfahren zur herstellung einer waesserigen loesung vom natriumsalz des methionins.
IT8123193A0 (it) Processo per la produzione di esacis(metossimetil)melammina.
ATE1991T1 (de) Verfahren zur herstellung von alkalidifluormethansulfonaten.
DE2967648D1 (en) Utilisation of 2-(n-(2,6-dichloro-phenyl)-n-allyl-amino)-imidazoline-(2) for the production of bradycardiac drugs
DK588289D0 (da) Ny heterocyklisk kemi
PT91562A (pt) Process for preparing hemiphosphate hemihydrate of 2-(1-pentyl--3-guanidino-4-imidazolyl) thiazole
IT8026171A0 (it) Procedimento per la realizzazione di pelli, nonche' pelle cosi'ottenuta.
IT8125953A0 (it) Processo per la produzione di cianoacetilidrazoni di 2-formilchinossalin-1, 4-diossidi.
IT8320984A0 (it) Procedimento per la realizzazione di un elemento scatolare attrezzato, nonche' elemento scatolare cosi' ottenuto.
IT8022003A0 (it) Processo per la produzione di 2-(2,2,28-trifluoroetil)-ammino-benzofenoni 5-sostituiti.
IT8026557A0 (it) Processo per la produzione di metanolo.
IT8024646A0 (it) Procedimento per la realizzazione di nastri a sviluppo chiuso, particolarmente per operazioni di calandratura industriale, nonche'nastro ottenuto.
IT1122203B (it) Processo per la produzione di composti organici alifatici,difunzionali
GB673798A (en) Process for the manufacture of a novel isothiocyanate