CR10324A - Moleculas no peptidicas para detectar y tratar tumores - Google Patents

Moleculas no peptidicas para detectar y tratar tumores

Info

Publication number
CR10324A
CR10324A CR10324A CR10324A CR10324A CR 10324 A CR10324 A CR 10324A CR 10324 A CR10324 A CR 10324A CR 10324 A CR10324 A CR 10324A CR 10324 A CR10324 A CR 10324A
Authority
CR
Costa Rica
Prior art keywords
detect
treat tumors
peptidic molecules
acidity
tumors
Prior art date
Application number
CR10324A
Other languages
English (en)
Inventor
E Summerton James
Original Assignee
E Summerton James
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US11/395,487 external-priority patent/US20070231256A1/en
Priority claimed from US11/449,495 external-priority patent/US8084610B2/en
Priority claimed from US11/449,508 external-priority patent/US20080124274A1/en
Application filed by E Summerton James filed Critical E Summerton James
Publication of CR10324A publication Critical patent/CR10324A/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/185Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19Carboxylic acids, e.g. valproic acid
    • A61K31/195Carboxylic acids, e.g. valproic acid having an amino group
    • A61K31/197Carboxylic acids, e.g. valproic acid having an amino group the amino and the carboxyl groups being attached to the same acyclic carbon chain, e.g. gamma-aminobutyric acid [GABA], beta-alanine, epsilon-aminocaproic acid or pantothenic acid
    • A61K31/198Alpha-amino acids, e.g. alanine or edetic acid [EDTA]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/185Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19Carboxylic acids, e.g. valproic acid
    • A61K31/20Carboxylic acids, e.g. valproic acid having a carboxyl group bound to a chain of seven or more carbon atoms, e.g. stearic, palmitic, arachidic acids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Abstract

Una de las caracteristicas mas universales de los tumores malignos es su acidez. Las oncotools son pequenas moleculas sinteticas no peptidicas disenadas para aprovechar esta acidez para la deteccion temprana y la destruccion de tumores. Cada oncotool tiene una estructura que es anionica e hidrofila a pH 7,4 y de este modo repele las superficies cargadas negativamente de las celulas en los tejidos normales.
CR10324A 2006-03-30 2008-09-29 Moleculas no peptidicas para detectar y tratar tumores CR10324A (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US11/395,487 US20070231256A1 (en) 2006-03-30 2006-03-30 Compositions and methods for detecting and treating tumors containing acidic areas
US11/449,495 US8084610B2 (en) 2006-06-07 2006-06-07 Compositions and methods for detecting and treating tumors containing acidic areas
US11/449,508 US20080124274A1 (en) 2006-06-07 2006-06-07 Compositions and methods for detecting and treating tumors containing acidic areas

Publications (1)

Publication Number Publication Date
CR10324A true CR10324A (es) 2008-11-26

Family

ID=39870100

Family Applications (1)

Application Number Title Priority Date Filing Date
CR10324A CR10324A (es) 2006-03-30 2008-09-29 Moleculas no peptidicas para detectar y tratar tumores

Country Status (1)

Country Link
CR (1) CR10324A (es)

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