CO2023017669A2 - Terapia combinada anti-vhc ventajosa - Google Patents
Terapia combinada anti-vhc ventajosaInfo
- Publication number
- CO2023017669A2 CO2023017669A2 CONC2023/0017669A CO2023017669A CO2023017669A2 CO 2023017669 A2 CO2023017669 A2 CO 2023017669A2 CO 2023017669 A CO2023017669 A CO 2023017669A CO 2023017669 A2 CO2023017669 A2 CO 2023017669A2
- Authority
- CO
- Colombia
- Prior art keywords
- compound
- combination therapy
- advantageous anti
- hcv combination
- pharmaceutically acceptable
- Prior art date
Links
- 238000002648 combination therapy Methods 0.000 title 1
- 208000005176 Hepatitis C Diseases 0.000 abstract 2
- 229940125904 compound 1 Drugs 0.000 abstract 2
- 229940125782 compound 2 Drugs 0.000 abstract 2
- 150000001875 compounds Chemical class 0.000 abstract 2
- 150000003839 salts Chemical class 0.000 abstract 2
- 238000004519 manufacturing process Methods 0.000 abstract 1
- 238000000034 method Methods 0.000 abstract 1
- 230000002195 synergetic effect Effects 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/70—Carbohydrates; Sugars; Derivatives thereof
- A61K31/7042—Compounds having saccharide radicals and heterocyclic rings
- A61K31/7052—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides
- A61K31/706—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom
- A61K31/7064—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom containing condensed or non-condensed pyrimidines
- A61K31/7076—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom containing condensed or non-condensed pyrimidines containing purines, e.g. adenosine, adenylic acid
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/4164—1,3-Diazoles
- A61K31/4184—1,3-Diazoles condensed with carbocyclic rings, e.g. benzimidazoles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
- A61K31/52—Purines, e.g. adenine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
- A61K31/536—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines ortho- or peri-condensed with carbocyclic ring systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
- A61K31/5365—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines ortho- or peri-condensed with heterocyclic ring systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
- A61P31/16—Antivirals for RNA viruses for influenza or rhinoviruses
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K2300/00—Mixtures or combinations of active ingredients, wherein at least one active ingredient is fully defined in groups A61K31/00 - A61K41/00
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical & Material Sciences (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Epidemiology (AREA)
- Virology (AREA)
- Molecular Biology (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Communicable Diseases (AREA)
- Oncology (AREA)
- Pulmonology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Medicinal Preparation (AREA)
Abstract
Una combinación farmacéutica sinérgica del Compuesto 1 o una sal farmacéuticamente aceptable del mismo (por ejemplo, el Compuesto 1-A) y el Compuesto 2 o una sal farmacéuticamente aceptable del mismo, así como sus usos para tratar la hepatitis C o una afección relacionada con la hepatitis C, así como los métodos para la fabricación de la combinación farmacéutica: : Compuesto 1 Compuesto 1-A Compuesto 2
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US202163212047P | 2021-06-17 | 2021-06-17 | |
PCT/US2022/034083 WO2022266497A1 (en) | 2021-06-17 | 2022-06-17 | Advantageous anti-hcv combination therapy |
Publications (1)
Publication Number | Publication Date |
---|---|
CO2023017669A2 true CO2023017669A2 (es) | 2023-12-29 |
Family
ID=84487918
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CONC2023/0017669A CO2023017669A2 (es) | 2021-06-17 | 2023-12-18 | Terapia combinada anti-vhc ventajosa |
Country Status (11)
Country | Link |
---|---|
US (1) | US20240148770A1 (es) |
EP (1) | EP4355319A1 (es) |
JP (1) | JP2024525164A (es) |
KR (1) | KR20240022574A (es) |
CN (1) | CN117500494A (es) |
AU (1) | AU2022291927A1 (es) |
BR (1) | BR112023026356A2 (es) |
CA (1) | CA3174073A1 (es) |
CO (1) | CO2023017669A2 (es) |
IL (1) | IL308921A (es) |
MX (1) | MX2023014898A (es) |
-
2022
- 2022-06-17 JP JP2023577547A patent/JP2024525164A/ja active Pending
- 2022-06-17 CN CN202280042755.0A patent/CN117500494A/zh active Pending
- 2022-06-17 AU AU2022291927A patent/AU2022291927A1/en active Pending
- 2022-06-17 BR BR112023026356A patent/BR112023026356A2/pt unknown
- 2022-06-17 IL IL308921A patent/IL308921A/en unknown
- 2022-06-17 MX MX2023014898A patent/MX2023014898A/es unknown
- 2022-06-17 EP EP22825933.9A patent/EP4355319A1/en active Pending
- 2022-06-17 KR KR1020247001335A patent/KR20240022574A/ko unknown
- 2022-06-17 CA CA3174073A patent/CA3174073A1/en active Pending
-
2023
- 2023-12-14 US US18/540,608 patent/US20240148770A1/en active Pending
- 2023-12-18 CO CONC2023/0017669A patent/CO2023017669A2/es unknown
Also Published As
Publication number | Publication date |
---|---|
CN117500494A (zh) | 2024-02-02 |
KR20240022574A (ko) | 2024-02-20 |
BR112023026356A2 (pt) | 2024-03-05 |
MX2023014898A (es) | 2024-04-29 |
EP4355319A1 (en) | 2024-04-24 |
JP2024525164A (ja) | 2024-07-10 |
US20240148770A1 (en) | 2024-05-09 |
AU2022291927A1 (en) | 2024-01-04 |
CA3174073A1 (en) | 2022-12-17 |
IL308921A (en) | 2024-01-01 |
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