CN1771031A - 用sarms治疗与女性雄激素缺乏(ad if)相关的疾病 - Google Patents
用sarms治疗与女性雄激素缺乏(ad if)相关的疾病 Download PDFInfo
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- CN1771031A CN1771031A CNA2004800077667A CN200480007766A CN1771031A CN 1771031 A CN1771031 A CN 1771031A CN A2004800077667 A CNA2004800077667 A CN A2004800077667A CN 200480007766 A CN200480007766 A CN 200480007766A CN 1771031 A CN1771031 A CN 1771031A
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Cited By (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN103251579A (zh) * | 2006-08-24 | 2013-08-21 | 田纳西大学研究基金会 | 取代的n-酰基苯胺及其使用方法 |
| CN104754939A (zh) * | 2012-07-13 | 2015-07-01 | Gtx公司 | 用选择性雄激素受体调节剂(sarm)治疗雄激素受体(ar)阳性乳癌的方法 |
| WO2025102293A1 (zh) * | 2023-11-16 | 2025-05-22 | 北京脑科学与类脑研究所 | 神经活性雄激素受体调节剂及其用途 |
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| US7759520B2 (en) | 1996-11-27 | 2010-07-20 | University Of Tennessee Research Foundation | Synthesis of selective androgen receptor modulators |
| US20040260108A1 (en) * | 2001-06-25 | 2004-12-23 | Dalton James T. | Metabolites of selective androgen receptor modulators and methods of use thereof |
| US8445534B2 (en) | 2000-08-24 | 2013-05-21 | University Of Tennessee Research Foundation | Treating androgen decline in aging male (ADAM)-associated conditions with SARMs |
| US20060276539A1 (en) * | 2002-10-16 | 2006-12-07 | Dalton James T | Treating Androgen Decline in Aging Male (ADAM)- associated conditions with SARMS |
| WO2004035739A2 (en) * | 2002-10-16 | 2004-04-29 | Gtx, Inc. | Treating androgen decline in aging male (adam)-associated conditions with sarms |
| US8309603B2 (en) | 2004-06-07 | 2012-11-13 | University Of Tennessee Research Foundation | SARMs and method of use thereof |
| FI20030958A0 (fi) * | 2003-06-27 | 2003-06-27 | Orion Corp | Uusia yhdisteitä |
| MXPA06002462A (es) * | 2003-10-14 | 2006-06-20 | Gtx Inc | Tratamiento de desordenes relacionados con huesos con moduladores del receptor de angrogeno selectivo. |
| US9884038B2 (en) | 2004-06-07 | 2018-02-06 | University Of Tennessee Research Foundation | Selective androgen receptor modulator and methods of use thereof |
| US20090215731A1 (en) | 2005-10-19 | 2009-08-27 | Chavah Pty Ltd. | Reduction of Side Effects From Aromatase Inhibitors Used for Treating Breast Cancer |
| KR100785038B1 (ko) * | 2006-04-17 | 2007-12-12 | 삼성전자주식회사 | 비정질 ＺｎＯ계 ＴＦＴ |
| CA2658394C (en) * | 2006-07-12 | 2016-08-16 | University Of Tennessee Research Foundation | Substituted acylanilides and methods of use thereof |
| US9730908B2 (en) | 2006-08-24 | 2017-08-15 | University Of Tennessee Research Foundation | SARMs and method of use thereof |
| US9844528B2 (en) | 2006-08-24 | 2017-12-19 | University Of Tennessee Research Foundation | SARMs and method of use thereof |
| US10010521B2 (en) | 2006-08-24 | 2018-07-03 | University Of Tennessee Research Foundation | SARMs and method of use thereof |
| US7968603B2 (en) | 2007-09-11 | 2011-06-28 | University Of Tennessee Research Foundation | Solid forms of selective androgen receptor modulators |
| US8791158B2 (en) | 2010-01-11 | 2014-07-29 | Gtx, Inc. | Methods of treating meibomian gland dysfunction |
| FR2982261B1 (fr) | 2011-11-04 | 2014-06-13 | Galderma Res & Dev | Nouveaux amides, et leur utilisation pharmaceutique ou cosmetique |
| US10314807B2 (en) | 2012-07-13 | 2019-06-11 | Gtx, Inc. | Method of treating HER2-positive breast cancers with selective androgen receptor modulators (SARMS) |
| US9744149B2 (en) | 2012-07-13 | 2017-08-29 | Gtx, Inc. | Method of treating androgen receptor (AR)-positive breast cancers with selective androgen receptor modulator (SARMs) |
| US10258596B2 (en) | 2012-07-13 | 2019-04-16 | Gtx, Inc. | Method of treating HER2-positive breast cancers with selective androgen receptor modulators (SARMS) |
| US9969683B2 (en) | 2012-07-13 | 2018-05-15 | Gtx, Inc. | Method of treating estrogen receptor (ER)-positive breast cancers with selective androgen receptor modulator (SARMS) |
| US10987334B2 (en) | 2012-07-13 | 2021-04-27 | University Of Tennessee Research Foundation | Method of treating ER mutant expressing breast cancers with selective androgen receptor modulators (SARMs) |
| US9622992B2 (en) | 2012-07-13 | 2017-04-18 | Gtx, Inc. | Method of treating androgen receptor (AR)-positive breast cancers with selective androgen receptor modulator (SARMs) |
| CN107405353B (zh) | 2014-10-22 | 2021-07-30 | 哈瓦赫治疗有限公司 | 降低乳房摄影乳腺密度和/或乳腺癌风险的方法 |
| SG11201803260PA (en) | 2015-10-22 | 2018-05-30 | Havah Therapeutics Pty Ltd | Methods of reducing mammographic breast density and/or breast cancer risk |
| CN106405064B (zh) * | 2016-08-30 | 2018-10-26 | 嘉兴行健生物科技有限公司 | 一种40岁以上女性骨转换率的评估方法 |
| JP2022535827A (ja) | 2019-06-03 | 2022-08-10 | ハバ セラピューティクス ピーティワイ エルティディ | アンドロゲン剤およびアロマターゼ阻害剤の送達のための医薬製剤およびシステム、ならびに使用のための方法 |
| US11701332B2 (en) * | 2020-11-18 | 2023-07-18 | Bryce Nicholas Day | Methods and compositions for treating female sexual interest and arousal disorder |
| WO2023101710A1 (en) * | 2021-12-02 | 2023-06-08 | Veru Inc. | Methods of treating breast cancers with selective androgen receptor modulators and additional therapeutic agents |
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| GB8617653D0 (en) * | 1986-07-18 | 1986-08-28 | Ici Plc | Amide derivatives |
| CA2132706C (en) * | 1992-04-10 | 1998-08-04 | John Eugene Macor | Acylaminoindole derivatives as 5-ht1 agonists |
| US7026500B2 (en) * | 2000-08-24 | 2006-04-11 | University Of Tennessee Research Foundation | Halogenated selective androgen receptor modulators and methods of use thereof |
| AU2001285230C1 (en) * | 2000-08-24 | 2008-03-13 | University Of Tennessee Research Foundation | Selective androgen receptor modulators and methods of use thereof |
| EA200401121A1 (ru) * | 2002-02-28 | 2005-10-27 | Юниверсити Оф Теннесси Рисерч Фаундейшн | Необратимые селективные модуляторы андрогенового рецептора и способы их применения |
| BR0308176A (pt) * | 2002-02-28 | 2005-01-04 | Univ Tennessee Res Foundation | Moduladores seletivos receptores de androgênio multi-substituìdos e seus métodos de uso |
| CN100537520C (zh) * | 2002-06-17 | 2009-09-09 | 田纳西大学研究基金会 | N-桥连选择性雄激素受体调节剂及其使用方法 |
| AU2003287077B2 (en) * | 2002-10-15 | 2007-09-20 | University Of Tennessee Research Foundation | Methylene-bridged selective androgen receptor modulators and methods of use thereof |
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2004
- 2004-01-20 CA CA002514024A patent/CA2514024A1/en not_active Abandoned
- 2004-01-20 WO PCT/US2004/001359 patent/WO2004064747A2/en not_active Ceased
- 2004-01-20 AU AU2004206909A patent/AU2004206909A1/en not_active Abandoned
- 2004-01-20 JP JP2006501034A patent/JP2006516286A/ja active Pending
- 2004-01-20 CN CNA2004800077667A patent/CN1771031A/zh active Pending
- 2004-01-20 US US10/759,538 patent/US20050032750A1/en not_active Abandoned
- 2004-01-20 EP EP04703606A patent/EP1594490A4/en not_active Withdrawn
- 2004-01-27 TW TW093101758A patent/TW200503729A/zh unknown
Cited By (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN103251579A (zh) * | 2006-08-24 | 2013-08-21 | 田纳西大学研究基金会 | 取代的n-酰基苯胺及其使用方法 |
| CN103251579B (zh) * | 2006-08-24 | 2016-12-28 | 田纳西大学研究基金会 | 取代的n-酰基苯胺及其使用方法 |
| CN104754939A (zh) * | 2012-07-13 | 2015-07-01 | Gtx公司 | 用选择性雄激素受体调节剂(sarm)治疗雄激素受体(ar)阳性乳癌的方法 |
| CN108143728A (zh) * | 2012-07-13 | 2018-06-12 | Gtx公司 | 选择性雄激素受体调节剂在治疗乳癌中的用途 |
| CN110840870A (zh) * | 2012-07-13 | 2020-02-28 | Gtx公司 | 选择性雄激素受体调节剂在治疗转移性和难治性乳癌中的应用 |
| WO2025102293A1 (zh) * | 2023-11-16 | 2025-05-22 | 北京脑科学与类脑研究所 | 神经活性雄激素受体调节剂及其用途 |
Also Published As
| Publication number | Publication date |
|---|---|
| WO2004064747A3 (en) | 2005-01-27 |
| JP2006516286A (ja) | 2006-06-29 |
| AU2004206909A2 (en) | 2004-08-05 |
| WO2004064747A2 (en) | 2004-08-05 |
| CA2514024A1 (en) | 2004-08-05 |
| AU2004206909A1 (en) | 2004-08-05 |
| EP1594490A2 (en) | 2005-11-16 |
| TW200503729A (en) | 2005-02-01 |
| EP1594490A4 (en) | 2006-03-22 |
| US20050032750A1 (en) | 2005-02-10 |
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