CN116783198A - 螺环jak抑制剂、含其的药物组合物及其应用 - Google Patents
螺环jak抑制剂、含其的药物组合物及其应用 Download PDFInfo
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- CN116783198A CN116783198A CN202180080571.9A CN202180080571A CN116783198A CN 116783198 A CN116783198 A CN 116783198A CN 202180080571 A CN202180080571 A CN 202180080571A CN 116783198 A CN116783198 A CN 116783198A
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P21/00—Drugs for disorders of the muscular or neuromuscular system
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
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- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
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- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pulmonology (AREA)
- Dermatology (AREA)
- Neurology (AREA)
- Orthopedic Medicine & Surgery (AREA)
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Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CN202011399496 | 2020-12-02 | ||
| CN2020113994966 | 2020-12-02 | ||
| PCT/CN2021/134880 WO2022117012A1 (fr) | 2020-12-02 | 2021-12-01 | Inhibiteur de jak spirocyclique, composition pharmaceutique le contenant, et son application |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CN116783198A true CN116783198A (zh) | 2023-09-19 |
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| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CN202180080571.9A Pending CN116783198A (zh) | 2020-12-02 | 2021-12-01 | 螺环jak抑制剂、含其的药物组合物及其应用 |
Country Status (2)
| Country | Link |
|---|---|
| CN (1) | CN116783198A (fr) |
| WO (1) | WO2022117012A1 (fr) |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN105732636B (zh) * | 2014-12-30 | 2020-04-21 | 广东东阳光药业有限公司 | 杂芳化合物及其在药物中的应用 |
| EP3576743B1 (fr) * | 2017-02-03 | 2023-01-18 | LEO Pharma A/S | Dérivés des acides 5-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)- 5-azaspiro[2 5]octane-8-carboxyliques comme inhibiteurs de la kinase jak |
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2021
- 2021-12-01 WO PCT/CN2021/134880 patent/WO2022117012A1/fr active Application Filing
- 2021-12-01 CN CN202180080571.9A patent/CN116783198A/zh active Pending
Also Published As
| Publication number | Publication date |
|---|---|
| WO2022117012A1 (fr) | 2022-06-09 |
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