CN115811971A - 用于口服施用的新型延迟释放组合物 - Google Patents
用于口服施用的新型延迟释放组合物 Download PDFInfo
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- CN115811971A CN115811971A CN202180042664.2A CN202180042664A CN115811971A CN 115811971 A CN115811971 A CN 115811971A CN 202180042664 A CN202180042664 A CN 202180042664A CN 115811971 A CN115811971 A CN 115811971A
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- OENHQHLEOONYIE-JLTXGRSLSA-N β-Carotene Chemical compound CC=1CCCC(C)(C)C=1\C=C\C(\C)=C\C=C\C(\C)=C\C=C\C=C(/C)\C=C\C=C(/C)\C=C\C1=C(C)CCCC1(C)C OENHQHLEOONYIE-JLTXGRSLSA-N 0.000 description 1
Classifications
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/4841—Filling excipients; Inactive ingredients
- A61K9/4866—Organic macromolecular compounds
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/4891—Coated capsules; Multilayered drug free capsule shells
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/4164—1,3-Diazoles
- A61K31/4178—1,3-Diazoles not condensed 1,3-diazoles and containing further heterocyclic rings, e.g. pilocarpine, nitrofurantoin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/30—Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
- A61K47/36—Polysaccharides; Derivatives thereof, e.g. gums, starch, alginate, dextrin, hyaluronic acid, chitosan, inulin, agar or pectin
- A61K47/38—Cellulose; Derivatives thereof
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
- A61K9/0056—Mouth soluble or dispersible forms; Suckable, eatable, chewable coherent forms; Forms rapidly disintegrating in the mouth; Lozenges; Lollipops; Bite capsules; Baked products; Baits or other oral forms for animals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/4808—Preparations in capsules, e.g. of gelatin, of chocolate characterised by the form of the capsule or the structure of the filling; Capsules containing small tablets; Capsules with outer layer for immediate drug release
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/4816—Wall or shell material
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/4816—Wall or shell material
- A61K9/4825—Proteins, e.g. gelatin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
- A61P31/16—Antivirals for RNA viruses for influenza or rhinoviruses
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical & Material Sciences (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Medicinal Chemistry (AREA)
- Epidemiology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Virology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Pulmonology (AREA)
- Zoology (AREA)
- Physiology (AREA)
- Nutrition Science (AREA)
- Oncology (AREA)
- Communicable Diseases (AREA)
- Molecular Biology (AREA)
- Inorganic Chemistry (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (3)
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| GB2006074.5 | 2020-04-24 | ||
| GBGB2006074.5A GB202006074D0 (en) | 2020-04-24 | 2020-04-24 | New composition |
| PCT/GB2021/050993 WO2021214487A1 (en) | 2020-04-24 | 2021-04-23 | New delayed release composition for peroral administration |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CN115811971A true CN115811971A (zh) | 2023-03-17 |
Family
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| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CN202180042664.2A Pending CN115811971A (zh) | 2020-04-24 | 2021-04-23 | 用于口服施用的新型延迟释放组合物 |
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| LT (1) | LT4138789T (enExample) |
| MA (1) | MA59397B1 (enExample) |
| MD (1) | MD4138789T2 (enExample) |
| MX (1) | MX2022013069A (enExample) |
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| SM (1) | SMT202300289T1 (enExample) |
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| GB202004094D0 (en) * | 2020-03-20 | 2020-05-06 | Vicore Pharma Ab | New compounds and uses |
| GB202006074D0 (en) | 2020-04-24 | 2020-06-10 | Vicore Pharma Ab | New composition |
| WO2023152503A1 (en) * | 2022-02-10 | 2023-08-17 | Vicore Pharma Ab | Use of buloxibutid for the treatment of idiopathic pulmonary fibrosis |
| GB202201723D0 (en) * | 2022-02-10 | 2022-03-30 | Vicore Pharma Ab | New use |
Citations (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2005123072A1 (en) * | 2004-06-14 | 2005-12-29 | Sepracor Inc. | Methods and compositions for the treatment of pulmonary diseases |
| WO2016139475A1 (en) * | 2015-03-02 | 2016-09-09 | Vicore Pharma Ab | Angiotensin ii receptor agonist for treating pulmonary fibrosis |
| WO2019183513A1 (en) * | 2018-03-22 | 2019-09-26 | University Of Iowa Research Foundation | Compositions and methods for the treatment and prevention of muscular dystrophy |
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| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS59139317A (ja) * | 1983-01-31 | 1984-08-10 | Teisan Seiyaku Kk | 持続性のニフエジピン製剤 |
| SE9800550D0 (sv) | 1998-02-24 | 1998-02-24 | A & Science Invest Ab | A pharmaceutical preparation comprising an angiotensin II type 2 receptor agonist, and use thereof |
| EP1395566B1 (en) | 2001-05-31 | 2007-09-12 | Vicore Pharma AB | Tricyclic compounds useful as angiotensin ii agonists |
| JP2003325642A (ja) * | 2002-05-09 | 2003-11-18 | Sansho Pharmaceutical Co Ltd | 腸溶性皮膜付き硬質空カプセルと、腸溶性皮膜付き硬質空カプセルの製造方法と、腸溶性皮膜付き硬質カプセル剤 |
| KR101137084B1 (ko) * | 2003-10-10 | 2012-04-24 | 애보트 프러덕츠 게엠베하 | 셀렉티브 ⅰ１ 이미다졸린 수용체 작용제 및 엔지오텐신 ⅱ수용체 차단제를 포함하는 약학적 조성물 |
| PE20060777A1 (es) | 2004-12-24 | 2006-10-06 | Boehringer Ingelheim Int | Derivados de indolinona para el tratamiento o la prevencion de enfermedades fibroticas |
| EP2946773A1 (en) * | 2014-05-19 | 2015-11-25 | Tillotts Pharma AG | Modified release coated capsules |
| EP2946774B1 (en) | 2014-05-19 | 2020-04-22 | Tillotts Pharma AG | Modified release coated capsules |
| EP3332775A4 (en) * | 2015-08-04 | 2019-05-29 | Fuji Capsule Co., Ltd. | ENTERIC CAPSULE |
| WO2017221012A1 (en) | 2016-06-21 | 2017-12-28 | Vicore Pharma Ab | Methods and compositions for preventing or reducing the risk of cancer treatment-related cardiotoxicity |
| GB201710906D0 (en) | 2017-07-06 | 2017-08-23 | Vicore Pharma Ab | Compounds and methods for treating peripheral neuropathy |
| JP7044360B2 (ja) * | 2018-04-02 | 2022-03-30 | 三生医薬株式会社 | ハードカプセル用コーティング剤及びそれを用いたハードカプセル剤の製造方法 |
| GB201818164D0 (en) | 2018-11-07 | 2018-12-19 | Vicore Pharma Ab | New composition |
| GB202006074D0 (en) | 2020-04-24 | 2020-06-10 | Vicore Pharma Ab | New composition |
| GB202006079D0 (en) | 2020-04-24 | 2020-06-10 | Vicore Pharma Ab | New composition |
| GB202201723D0 (en) | 2022-02-10 | 2022-03-30 | Vicore Pharma Ab | New use |
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2020
- 2020-04-24 GB GBGB2006074.5A patent/GB202006074D0/en not_active Ceased
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2021
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- 2021-04-23 HU HUE21724011A patent/HUE062897T2/hu unknown
- 2021-04-23 FI FIEP21724011.8T patent/FI4138789T3/fi active
- 2021-04-23 WO PCT/GB2021/050993 patent/WO2021214487A1/en not_active Ceased
- 2021-04-23 CN CN202180042664.2A patent/CN115811971A/zh active Pending
- 2021-04-23 BR BR112022021520A patent/BR112022021520A2/pt unknown
- 2021-04-23 MD MDE20230229T patent/MD4138789T2/ro unknown
- 2021-04-23 DK DK21724011.8T patent/DK4138789T3/da active
- 2021-04-23 CA CA3180850A patent/CA3180850A1/en active Pending
- 2021-04-23 EP EP23177726.9A patent/EP4218737A1/en active Pending
- 2021-04-23 SI SI202130057T patent/SI4138789T1/sl unknown
- 2021-04-23 PL PL21724011.8T patent/PL4138789T3/pl unknown
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2022
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2023
- 2023-04-14 US US18/300,739 patent/US12121614B2/en active Active
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2024
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2025
- 2025-04-04 JP JP2025062545A patent/JP2025106410A/ja active Pending
Patent Citations (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2005123072A1 (en) * | 2004-06-14 | 2005-12-29 | Sepracor Inc. | Methods and compositions for the treatment of pulmonary diseases |
| WO2016139475A1 (en) * | 2015-03-02 | 2016-09-09 | Vicore Pharma Ab | Angiotensin ii receptor agonist for treating pulmonary fibrosis |
| WO2019183513A1 (en) * | 2018-03-22 | 2019-09-26 | University Of Iowa Research Foundation | Compositions and methods for the treatment and prevention of muscular dystrophy |
Non-Patent Citations (1)
| Title |
|---|
| DURRIYA HASHMAT等: "Development of enteric coated flurbiprofen tablets using opadry/acryl-ezesystem-A technical note", 《AAPS PHARMSCITECH》, vol. 9, no. 1, pages 116 - 121, XP055055554, DOI: 10.1208/s12249-007-9005-9 * |
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