CN114929703A - 一种溴区结构域蛋白抑制剂的晶型、盐型及其制备方法 - Google Patents
一种溴区结构域蛋白抑制剂的晶型、盐型及其制备方法 Download PDFInfo
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Abstract
一种式(I)所示的溴区结构域蛋白抑制剂的晶型、盐型及其制备方法,以及上述晶型和盐型在制备治疗由BET蛋白介导的疾病的药物中的用途。
Description
PCT国内申请,说明书已公开。
Claims (17)
- PCT国内申请,权利要求书已公开。
Applications Claiming Priority (5)
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CN202010057297 | 2020-01-19 | ||
CN2020100601102 | 2020-01-19 | ||
CN2020100572970 | 2020-01-19 | ||
CN202010060110 | 2020-01-19 | ||
PCT/CN2021/072651 WO2021143922A1 (zh) | 2020-01-19 | 2021-01-19 | 一种溴区结构域蛋白抑制剂的晶型、盐型及其制备方法 |
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CN114929703A true CN114929703A (zh) | 2022-08-19 |
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US (1) | US20240101551A1 (zh) |
EP (1) | EP4092027A4 (zh) |
JP (1) | JP2023510610A (zh) |
CN (1) | CN114929703A (zh) |
WO (1) | WO2021143922A1 (zh) |
Citations (1)
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WO2018130174A1 (zh) * | 2017-01-11 | 2018-07-19 | 江苏豪森药业集团有限公司 | 吡咯并[2,3-c]吡啶类衍生物、其制备方法及其在医药上的应用 |
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WO2013097052A1 (en) * | 2011-12-30 | 2013-07-04 | Abbott Laboratories | Bromodomain inhibitors |
AR096758A1 (es) * | 2013-06-28 | 2016-02-03 | Abbvie Inc | Inhibidores cristalinos de bromodominios |
CN110577526B (zh) * | 2018-06-07 | 2023-10-27 | 上海翰森生物医药科技有限公司 | 溴域结构蛋白抑制剂的盐及其制备方法和应用 |
US20210300923A1 (en) * | 2018-07-25 | 2021-09-30 | Chia Tai Tianqing Pharmaceutical Group Co., Ltd. | Sulfoximine compound as bromodomain protein inhibitor and pharmaceutical composition and medical use thereof |
-
2021
- 2021-01-19 EP EP21742003.3A patent/EP4092027A4/en active Pending
- 2021-01-19 CN CN202180008525.8A patent/CN114929703A/zh active Pending
- 2021-01-19 WO PCT/CN2021/072651 patent/WO2021143922A1/zh unknown
- 2021-01-19 JP JP2022543423A patent/JP2023510610A/ja active Pending
- 2021-01-19 US US17/793,588 patent/US20240101551A1/en active Pending
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WO2018130174A1 (zh) * | 2017-01-11 | 2018-07-19 | 江苏豪森药业集团有限公司 | 吡咯并[2,3-c]吡啶类衍生物、其制备方法及其在医药上的应用 |
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US20240101551A1 (en) | 2024-03-28 |
EP4092027A1 (en) | 2022-11-23 |
JP2023510610A (ja) | 2023-03-14 |
EP4092027A4 (en) | 2024-02-14 |
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