CN110101734A - 一种治疗气滞血瘀型骨关节病的精油及其制备方法 - Google Patents

一种治疗气滞血瘀型骨关节病的精油及其制备方法 Download PDF

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CN110101734A
CN110101734A CN201910520555.1A CN201910520555A CN110101734A CN 110101734 A CN110101734 A CN 110101734A CN 201910520555 A CN201910520555 A CN 201910520555A CN 110101734 A CN110101734 A CN 110101734A
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郭珈宜
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    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K36/00Medicinal preparations of undetermined constitution containing material from algae, lichens, fungi or plants, or derivatives thereof, e.g. traditional herbal medicines
    • A61K36/18Magnoliophyta (angiosperms)
    • A61K36/185Magnoliopsida (dicotyledons)
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    • A61K36/232Angelica
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K36/00Medicinal preparations of undetermined constitution containing material from algae, lichens, fungi or plants, or derivatives thereof, e.g. traditional herbal medicines
    • A61K36/18Magnoliophyta (angiosperms)
    • A61K36/185Magnoliopsida (dicotyledons)
    • A61K36/23Apiaceae or Umbelliferae (Carrot family), e.g. dill, chervil, coriander or cumin
    • A61K36/236Ligusticum (licorice-root)
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K36/00Medicinal preparations of undetermined constitution containing material from algae, lichens, fungi or plants, or derivatives thereof, e.g. traditional herbal medicines
    • A61K36/18Magnoliophyta (angiosperms)
    • A61K36/185Magnoliopsida (dicotyledons)
    • A61K36/25Araliaceae (Ginseng family), e.g. ivy, aralia, schefflera or tetrapanax
    • A61K36/258Panax (ginseng)
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K36/00Medicinal preparations of undetermined constitution containing material from algae, lichens, fungi or plants, or derivatives thereof, e.g. traditional herbal medicines
    • A61K36/18Magnoliophyta (angiosperms)
    • A61K36/185Magnoliopsida (dicotyledons)
    • A61K36/26Aristolochiaceae (Birthwort family), e.g. heartleaf
    • A61K36/268Asarum (wild ginger)
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K36/00Medicinal preparations of undetermined constitution containing material from algae, lichens, fungi or plants, or derivatives thereof, e.g. traditional herbal medicines
    • A61K36/18Magnoliophyta (angiosperms)
    • A61K36/185Magnoliopsida (dicotyledons)
    • A61K36/32Burseraceae (Frankincense family)
    • A61K36/324Boswellia, e.g. frankincense
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K36/00Medicinal preparations of undetermined constitution containing material from algae, lichens, fungi or plants, or derivatives thereof, e.g. traditional herbal medicines
    • A61K36/18Magnoliophyta (angiosperms)
    • A61K36/185Magnoliopsida (dicotyledons)
    • A61K36/32Burseraceae (Frankincense family)
    • A61K36/328Commiphora, e.g. mecca myrrh or balm of Gilead
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0014Skin, i.e. galenical aspects of topical compositions
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • A61P19/02Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • CCHEMISTRY; METALLURGY
    • C11ANIMAL OR VEGETABLE OILS, FATS, FATTY SUBSTANCES OR WAXES; FATTY ACIDS THEREFROM; DETERGENTS; CANDLES
    • C11BPRODUCING, e.g. BY PRESSING RAW MATERIALS OR BY EXTRACTION FROM WASTE MATERIALS, REFINING OR PRESERVING FATS, FATTY SUBSTANCES, e.g. LANOLIN, FATTY OILS OR WAXES; ESSENTIAL OILS; PERFUMES
    • C11B9/00Essential oils; Perfumes
    • C11B9/02Recovery or refining of essential oils from raw materials
    • C11B9/022Refining
    • CCHEMISTRY; METALLURGY
    • C11ANIMAL OR VEGETABLE OILS, FATS, FATTY SUBSTANCES OR WAXES; FATTY ACIDS THEREFROM; DETERGENTS; CANDLES
    • C11BPRODUCING, e.g. BY PRESSING RAW MATERIALS OR BY EXTRACTION FROM WASTE MATERIALS, REFINING OR PRESERVING FATS, FATTY SUBSTANCES, e.g. LANOLIN, FATTY OILS OR WAXES; ESSENTIAL OILS; PERFUMES
    • C11B9/00Essential oils; Perfumes
    • C11B9/02Recovery or refining of essential oils from raw materials
    • C11B9/025Recovery by solvent extraction
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K2236/00Isolation or extraction methods of medicinal preparations of undetermined constitution containing material from algae, lichens, fungi or plants, or derivatives thereof, e.g. traditional herbal medicine
    • A61K2236/30Extraction of the material
    • A61K2236/33Extraction of the material involving extraction with hydrophilic solvents, e.g. lower alcohols, esters or ketones
    • A61K2236/331Extraction of the material involving extraction with hydrophilic solvents, e.g. lower alcohols, esters or ketones using water, e.g. cold water, infusion, tea, steam distillation, decoction
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K2236/00Isolation or extraction methods of medicinal preparations of undetermined constitution containing material from algae, lichens, fungi or plants, or derivatives thereof, e.g. traditional herbal medicine
    • A61K2236/30Extraction of the material
    • A61K2236/35Extraction with lipophilic solvents, e.g. Hexane or petrol ether

Abstract

本发明提供了一种治疗气滞血瘀型骨关节病的精油及其制备方法,所述精油包括以下成分:人参精油、当归精油、乳香精油、没药精油、细辛精油及川芎精油。本发明提供的一种治疗气滞血瘀型骨关节病的精油及其制备方法,制备方法简单,该精油配方具有活血行气,舒筋通络止痛之功效,能有效治疗气滞血瘀引起的骨关节病,对骨关节疼痛固定不移,痛如针刺,局部压痛明显而拒按,关节活动不利,舌紫暗或有瘀斑,苔薄,脉弦涩等症效果显著。

Description

一种治疗气滞血瘀型骨关节病的精油及其制备方法
技术领域
本发明涉及中医药领域,具体是指一种治疗气滞血瘀型骨关节病的精油及其制备方法。
背景技术
骨关节病是中老年常见的多发病,是一种慢性退行性疾病,以关节软骨局灶损伤,伴有骨赘形成、韧带松弛、关节周围肌肉萎缩、和滑膜炎症等为特征的关节退变。其病理机理是外伤或劳损引起的骨关节周围肌肉、韧带的痉挛、松弛等病变,关节的稳定及受力平衡遭到破坏,关节软骨间的应力改变,产生无菌性炎症,进一步破坏关节软骨。临床表现为关节疼痛肿胀,屈伸不利,肌肉微缩无力,这些症状给患者带来极大的痛苦,也给生活带来许多不便,保守治疗时,服用西药,如非甾体抗炎药,乙酰氨基酚等,对肠胃功能有损害,长期疗效不佳。手术治疗成本高,创伤大,患者不易接受。
发明内容
以解决上述背景技术中提出的问题,本发明的目的在于提供一种治疗气滞血瘀型骨关节病的精油及其制备方法,该精油配方具有活血行气,舒筋通络止痛之功效,能有效治疗气滞血瘀引起的骨关节病,对骨关节疼痛固定不移,痛如针刺,局部压痛明显而拒按,关节活动不利,舌紫暗或有瘀斑,苔薄,脉弦涩等症效果显著。
为解决上述技术问题,本发明提供的技术方案为:
一种治疗气滞血瘀型骨关节病的精油及其制备方法,所述精油包括以下成分:人参、当归、乳香、没药、细辛及川芎;
所述的制备方法包括以下步骤:
1)将人参磨成细粉,其大小不超过200目,将人参细粉放入蒸馏锅内,蒸馏锅锅里灌入清水,清水和人参细粉的质量比为5-6:1,进行加热蒸馏,温度为120-140℃,加热时间为0.5-1小时,制成浆糊状;
2)将步骤1)制得的糊状液体进行沉淀2-4小时,过滤出上部液体为粗精油;
3)将乙醚按照与粗精油1:1的体积比进行萃取,添加10g/L无机盐进行盐析,搅拌萃取得精油成品;
4)当归、乳香、没药、细辛及川芎按照人参相同的方式进行提取精油;
5)提取好各个材料的精油装入玻璃瓶,备用;
6)取人参精油4-6份、当归精油4-6份、乳香精油5份、没药精油4-6份、细辛精油2-4份及川芎精油5-7份,将各个精油进行搅拌混合均匀即得。
作为改进,所述步骤6)中制备好的精油使用玻璃瓶或陶瓷瓶进行盛放。
本发明的有益效果是:
本发明提供的一种治疗治疗气滞血瘀型骨关节病的精油配方,能有效治疗风、寒、湿引起的骨关节病及痹症,表现由气滞血瘀造成的关节疼痛固定不移,痛如针刺,局部压痛明显而拒按,关节活动不利,舌紫暗或有瘀斑,苔薄,脉弦涩等症疗效显著,对防止血瘀气滞不通,经脉痹阻,关节不利效果明显。
本发明的制备工艺简单,工艺中所有药物按照不同方法提取精油,全面提取药材中的有效成分,相互配伍,乳香、没药、川芎活血化瘀;当归活血养血;细辛发散风寒,祛风止痛;人参,大补元气,加强以上药物效力,通过玄府入药,使制备得到的精油配方药物生物利用度高、疗效更加显著,适用推广应用。
具体实施方式
下面用具体实施例说明本发明,并不是对本发明的限制。
实施例一
一种治疗气滞血瘀型骨关节病的精油及其制备方法,所述精油包括以下成分:人参、当归、乳香、没药、细辛及川芎;
所述的制备方法包括以下步骤:
1)将人参磨成细粉,其大小不超过200目,将人参细粉放入蒸馏锅内,蒸馏锅锅里灌入清水,清水和人参细粉的质量比为5-6:1,进行加热蒸馏,温度为130℃,加热时间为1小时,制成浆糊状;
2)将步骤1)制得的糊状液体进行沉淀3小时,过滤出上部液体为粗精油;
3)将乙醚按照与粗精油1:1的体积比进行萃取,添加10g/L无机盐进行盐析,搅拌萃取得精油成品;
4)当归、乳香、没药、细辛及川芎按照人参相同的方式进行提取精油;
5)提取好各个材料的精油装入玻璃瓶,备用;
6)取人参精油6份、当归精油4份、乳香精油5份、没药精油4份、细辛精油4份及川芎精油5份,将各个精油进行搅拌混合均匀即得。
所述步骤6)中制备好的精油使用玻璃瓶或陶瓷瓶进行盛放。
使用时,将自己的患处清洗干净(最好使用酒精擦拭),然后取3-5ml的精油进行涂抹患处,手朝同一方向进行画圆涂抹,直至精油被完全吸收。
实施例二
一种治疗气滞血瘀型骨关节病的精油及其制备方法,其特征在于,所述精油包括以下成分:人参、当归、乳香、没药、细辛及川芎;
所述的制备方法包括以下步骤:
1)将人参磨成细粉,其大小不超过200目,将人参细粉放入蒸馏锅内,蒸馏锅锅里灌入清水,清水和人参细粉的质量比为5:1,进行加热蒸馏,温度为120℃,加热时间为半小时,制成浆糊状;
2)将步骤1)制得的糊状液体进行沉淀3小时,过滤出上部液体为粗精油;
3)将乙醚按照与粗精油1:1的体积比进行萃取,添加10g/L无机盐进行盐析,搅拌萃取得精油成品;
4)当归、乳香、没药、细辛及川芎按照人参相同的方式进行提取精油;
5)提取好各个材料的精油装入玻璃瓶,备用;
6)取人参精油5份、当归精油5份、乳香精油5份、没药精油5份、细辛精油3份及川芎精油6份,将各个精油进行搅拌混合均匀即得。
所述步骤6)中制备好的精油使用玻璃瓶或陶瓷瓶进行盛放。
使用时,将自己的患处清洗干净(最好使用酒精擦拭),然后取3-5ml的精油进行涂抹患处,手朝同一方向进行画圆涂抹,直至精油被完全吸收。
以上所述,仅为本发明较佳的具体实施方式,但本发明的保护范围并不局限于此,任何熟悉本技术领域的技术人员在本发明揭露的技术范围内,根据本发明的技术方案及其发明构思加以等同替换或改变,都应涵盖在本发明的保护范围之内。

Claims (2)

1.一种治疗气滞血瘀型骨关节病的精油及其制备方法,其特征在于,所述精油包括以下成分:人参、当归、乳香、没药、细辛及川芎;
所述的制备方法包括以下步骤:
1)将人参磨成细粉,其大小不超过200目,将人参细粉放入蒸馏锅内,蒸馏锅锅里灌入清水,清水和人参细粉的质量比为5-6:1,进行加热蒸馏,温度为120-140℃,加热时间为0.5-1小时,制成浆糊状;
2)将步骤1)制得的糊状液体进行沉淀2-4小时,过滤出上部液体为粗精油;
3)将乙醚按照与粗精油1:1的体积比进行萃取,添加10g/L无机盐进行盐析,搅拌萃取得精油成品;
4)当归、乳香、没药、细辛及川芎按照人参相同的方式进行提取精油;
5)提取好各个材料的精油装入玻璃瓶,备用;
6)取人参精油4-6份、当归精油4-6份、乳香精油5份、没药精油4-6份、细辛精油2-4份及川芎精油5-7份,将各个精油进行搅拌混合均匀即得。
2.根据权利要求1所述的一种治疗气滞血瘀型骨关节病的精油及其制备方法,其特征在于,所述步骤6)中制备好的精油使用玻璃瓶或陶瓷瓶进行盛放。
CN201910520555.1A 2019-06-17 2019-06-17 一种治疗气滞血瘀型骨关节病的精油及其制备方法 Withdrawn CN110101734A (zh)

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