CN105153232B - 一种用于治疗骨质疏松的米诺膦酸的制备方法 - Google Patents
一种用于治疗骨质疏松的米诺膦酸的制备方法 Download PDFInfo
- Publication number
- CN105153232B CN105153232B CN201510677560.5A CN201510677560A CN105153232B CN 105153232 B CN105153232 B CN 105153232B CN 201510677560 A CN201510677560 A CN 201510677560A CN 105153232 B CN105153232 B CN 105153232B
- Authority
- CN
- China
- Prior art keywords
- formula
- reaction
- compound shown
- minodronic acid
- acid
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Fee Related
Links
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Abstract
Description
Claims (8)
Priority Applications (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
CN201510677560.5A CN105153232B (zh) | 2015-10-17 | 2015-10-17 | 一种用于治疗骨质疏松的米诺膦酸的制备方法 |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
CN201510677560.5A CN105153232B (zh) | 2015-10-17 | 2015-10-17 | 一种用于治疗骨质疏松的米诺膦酸的制备方法 |
Publications (2)
Publication Number | Publication Date |
---|---|
CN105153232A CN105153232A (zh) | 2015-12-16 |
CN105153232B true CN105153232B (zh) | 2017-12-15 |
Family
ID=54794316
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CN201510677560.5A Expired - Fee Related CN105153232B (zh) | 2015-10-17 | 2015-10-17 | 一种用于治疗骨质疏松的米诺膦酸的制备方法 |
Country Status (1)
Country | Link |
---|---|
CN (1) | CN105153232B (zh) |
Families Citing this family (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN107033187A (zh) * | 2017-04-28 | 2017-08-11 | 江苏笃诚医药科技股份有限公司 | 一种米诺膦酸的制备方法 |
CN109456363A (zh) * | 2018-11-01 | 2019-03-12 | 南京海纳医药科技股份有限公司 | 一种米诺膦酸工艺杂质的制备方法 |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US6514969B2 (en) * | 2000-08-16 | 2003-02-04 | Boehringer Ingelheim Pharma Kg | β-amyloid inhibitors, processes for preparing them, and their use in pharmaceutical compositions |
CN101531681B (zh) * | 2008-03-10 | 2013-06-05 | 北京德众万全医药科技有限公司 | 一种高纯度的米诺膦酸及其制备方法 |
CN101973993A (zh) * | 2010-11-05 | 2011-02-16 | 天津药物研究院 | 一种制备2-[咪唑并(1,2-a)吡啶-3-基]乙酸的方法 |
CN102875602B (zh) * | 2012-10-25 | 2015-05-20 | 江苏神龙药业有限公司 | 一种米诺膦酸水合物的制备方法 |
-
2015
- 2015-10-17 CN CN201510677560.5A patent/CN105153232B/zh not_active Expired - Fee Related
Also Published As
Publication number | Publication date |
---|---|
CN105153232A (zh) | 2015-12-16 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
CA2340180A1 (en) | 1-aryl,-3-arylmethyl-1,8-naphthyridn-2(1h)-ones | |
WO2010111934A1 (zh) | 吡咯喹啉醌锂盐衍生物及其制备方法 | |
EP2743259B1 (en) | Method for purifying (s)-oxiracetam | |
CN103360425A (zh) | 替诺福韦酯及其富马酸盐的合成方法 | |
CN101885725A (zh) | 吡咯喹啉醌钠盐衍生物及其制备方法 | |
CN105153232B (zh) | 一种用于治疗骨质疏松的米诺膦酸的制备方法 | |
KR20080109088A (ko) | 로수바스타틴 아연 염 | |
CN105175446B (zh) | 一种治疗骨质疏松的米诺膦酸的制备方法 | |
CN102875602B (zh) | 一种米诺膦酸水合物的制备方法 | |
CN102718829A (zh) | 牛磺熊去氧胆酸钠的制备方法 | |
US4073895A (en) | Isopropylamino pyrimidine orthophosphate | |
EP2743258A1 (en) | Method for purifying levo-oxiracetam | |
CN102911234A (zh) | 以鸡胆汁为原料生产鹅去氧胆酸 | |
CN104974057B (zh) | 一种溴芬酸钠的制备方法和重要中间体 | |
CN106699812A (zh) | 替诺福韦前药的制备和纯化方法 | |
CN103159673B (zh) | 一种制备吉美嘧啶的精制方法 | |
CN105837635B (zh) | 一种用于治疗骨质疏松的米诺膦酸的制备方法 | |
CN104356065A (zh) | 一种氢溴酸依他佐辛的制备方法 | |
CA1132562A (en) | Halogeno derivatives of isopropylamino pyrimidine, their preparation and therapeutic use | |
CN106632483B (zh) | 一种替诺福韦二吡呋酯的制备方法 | |
CN110684066B (zh) | 胞二磷胆碱药物制剂及其脑梗塞急性期意识障碍的新用途 | |
CN102516301A (zh) | 用于治疗的汉黄芩素衍生物 | |
CN110981801B (zh) | 一锅法制备盐酸辛可卡因的生产工艺 | |
CN108047272B (zh) | 一种富马酸替诺福韦二吡呋酯的制备方法 | |
CN110746461A (zh) | 一种替诺福韦衍生物盐及其制备方法和一种药物组合物 |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
C06 | Publication | ||
PB01 | Publication | ||
C10 | Entry into substantive examination | ||
SE01 | Entry into force of request for substantive examination | ||
CB03 | Change of inventor or designer information |
Inventor after: Nie Hongmei Inventor after: Li Jianai Inventor after: Yu Jianmei Inventor before: Lv Yanhua |
|
CB03 | Change of inventor or designer information | ||
TA01 | Transfer of patent application right |
Effective date of registration: 20171117 Address after: 276399 No. 2, unit 14, building 70, building 401, Yuquanlu Road, Linyi, Shandong, Yinan Applicant after: Nie Hongmei Applicant after: Li Jianai Applicant after: Yu Jianmei Address before: 1 residential building, No. 443 Changjiang East Road, Huangdao District, Shandong, China, 1708, China, 266520 Applicant before: Chen Da bio tech ltd, Qingdao |
|
TA01 | Transfer of patent application right | ||
GR01 | Patent grant | ||
GR01 | Patent grant | ||
CF01 | Termination of patent right due to non-payment of annual fee |
Granted publication date: 20171215 Termination date: 20181017 |
|
CF01 | Termination of patent right due to non-payment of annual fee |