CN100526310C - 用作杀真菌剂的环丙基-噻吩基-甲酰胺 - Google Patents
用作杀真菌剂的环丙基-噻吩基-甲酰胺 Download PDFInfo
- Publication number
- CN100526310C CN100526310C CNB2003801021700A CN200380102170A CN100526310C CN 100526310 C CN100526310 C CN 100526310C CN B2003801021700 A CNB2003801021700 A CN B2003801021700A CN 200380102170 A CN200380102170 A CN 200380102170A CN 100526310 C CN100526310 C CN 100526310C
- Authority
- CN
- China
- Prior art keywords
- sub
- alkyl
- formula
- halogen
- optionally substituted
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Fee Related
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
- C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
- C07D333/26—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D333/30—Hetero atoms other than halogen
- C07D333/36—Nitrogen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D411/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen and sulfur atoms as the only ring hetero atoms
- C07D411/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen and sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D411/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen and sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Plural Heterocyclic Compounds (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Heterocyclic Compounds Containing Sulfur Atoms (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB0225554.5 | 2002-11-01 | ||
| GBGB0225554.5A GB0225554D0 (en) | 2002-11-01 | 2002-11-01 | Chemical compounds |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| CN1708496A CN1708496A (zh) | 2005-12-14 |
| CN100526310C true CN100526310C (zh) | 2009-08-12 |
Family
ID=9947074
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CNB2003801021700A Expired - Fee Related CN100526310C (zh) | 2002-11-01 | 2003-10-24 | 用作杀真菌剂的环丙基-噻吩基-甲酰胺 |
Country Status (23)
| Country | Link |
|---|---|
| US (1) | US7312179B2 (enExample) |
| EP (1) | EP1556377B1 (enExample) |
| JP (1) | JP4673061B2 (enExample) |
| KR (1) | KR101000731B1 (enExample) |
| CN (1) | CN100526310C (enExample) |
| AR (1) | AR041747A1 (enExample) |
| AT (1) | ATE331714T1 (enExample) |
| AU (1) | AU2003286140A1 (enExample) |
| BR (1) | BR0315857A (enExample) |
| CA (1) | CA2501739C (enExample) |
| CO (1) | CO5550397A2 (enExample) |
| DE (1) | DE60306540T2 (enExample) |
| DK (1) | DK1556377T3 (enExample) |
| EC (1) | ECSP055770A (enExample) |
| ES (1) | ES2266881T3 (enExample) |
| GB (1) | GB0225554D0 (enExample) |
| GT (1) | GT200300236A (enExample) |
| MX (1) | MXPA05004463A (enExample) |
| PT (1) | PT1556377E (enExample) |
| RU (1) | RU2005116974A (enExample) |
| TW (1) | TW200412848A (enExample) |
| WO (1) | WO2004039799A1 (enExample) |
| ZA (1) | ZA200502644B (enExample) |
Families Citing this family (18)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB0418047D0 (en) | 2004-08-12 | 2004-09-15 | Syngenta Participations Ag | Fungicidal compositions |
| DE102005025989A1 (de) * | 2005-06-07 | 2007-01-11 | Bayer Cropscience Ag | Carboxamide |
| US7723371B2 (en) | 2005-11-15 | 2010-05-25 | Syngenta Crop Protection, Inc. | Microbiocides |
| EA013354B1 (ru) * | 2005-11-15 | 2010-04-30 | Синджента Партисипейшнс Аг | Способ получения карбоксанилидов |
| HUE029570T2 (en) | 2010-04-27 | 2017-03-28 | Calcimedica Inc | Intracellular calcium modifying compounds |
| US10703722B2 (en) | 2010-04-27 | 2020-07-07 | Calcimedica, Inc. | Compounds that modulate intracellular calcium |
| EP2563759B1 (en) | 2010-04-27 | 2022-04-06 | Calcimedica, Inc. | Compounds that modulate intracellular calcium |
| CN103180316A (zh) | 2010-08-27 | 2013-06-26 | 钙医学公司 | 调节细胞内钙的化合物 |
| BR112013012081A2 (pt) * | 2010-11-15 | 2016-07-19 | Bayer Ip Gmbh | 5-halogenopirazol (tio) carboxamidas |
| US20120316182A1 (en) | 2011-06-10 | 2012-12-13 | Calcimedica, Inc. | Compounds that modulate intracellular calcium |
| US9856240B2 (en) | 2011-10-19 | 2018-01-02 | Calcimedica, Inc. | Compounds that modulate intracellular calcium |
| US9512116B2 (en) | 2012-10-12 | 2016-12-06 | Calcimedica, Inc. | Compounds that modulate intracellular calcium |
| CN114712513B (zh) | 2015-02-27 | 2026-02-10 | 钙医学公司 | 胰腺炎治疗 |
| AU2016306301B2 (en) | 2015-08-07 | 2021-02-11 | Calcimedica, Inc. | Use of CRAC channel inhibitors for the treatment of stroke and traumatic brain injury |
| CN106977457A (zh) * | 2016-12-22 | 2017-07-25 | 浙江海正化工股份有限公司 | 一种3‑二氟甲基‑1‑甲基‑吡唑‑4‑甲酸及其合成方法 |
| MA53085B1 (fr) * | 2018-07-05 | 2022-12-30 | Bayer Ag | Thiophènecarboxamides substitués et analogues comme agents antibactériens |
| US12544371B2 (en) | 2020-03-20 | 2026-02-10 | Calcimedica, Inc. | Methods and compositions for treating acute lung injury and acute respiratory distress syndrome |
| US12522589B2 (en) | 2020-11-13 | 2026-01-13 | Calcimedica, Inc. | Synthesis of CRAC channel inhibitors |
Citations (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB2126587A (en) * | 1982-09-13 | 1984-03-28 | Sandoz Ltd | Fungicidal thiophene derivatives |
| US4743602A (en) * | 1986-07-16 | 1988-05-10 | Imperial Chemical Industries Plc | Thiophene cyclopropyl amine compounds, compositions and fungicidal use |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2385721A1 (fr) * | 1977-03-31 | 1978-10-27 | Hexachimie | Cyclopropyl-6 dihydro-1,3 methyl-1 phenyl-5 oxo-2 2 h-thieno (2,3-e) diazepine, son procede de preparation et son application en therapeutique |
| GB8617378D0 (en) * | 1986-07-16 | 1986-08-20 | Ici Plc | Tertiary amine compounds |
| ES2169773T3 (es) | 1995-04-11 | 2002-07-16 | Mitsui Chemicals Inc | Derivados de tiofeno sustituido y fungicidas agricolas y horticolas que contienen dichos derivados como ingrediente activo. |
| GB9817548D0 (en) * | 1998-08-12 | 1998-10-07 | Novartis Ag | Organic compounds |
| GB9930750D0 (en) * | 1999-12-29 | 2000-02-16 | Novartis Ag | Organic compounds |
| DK1480955T3 (da) | 2002-03-05 | 2007-10-29 | Syngenta Participations Ag | O-cyclopropyl-carboxanilider og deres anvendelse som fungicider |
| EP2258690B1 (en) | 2002-08-22 | 2013-02-20 | Syngenta Participations AG | Tricyclic amines as intermediates in the synthesis of fungicidal carboxamide derivatives |
-
2002
- 2002-11-01 GB GBGB0225554.5A patent/GB0225554D0/en not_active Ceased
-
2003
- 2003-10-24 DE DE60306540T patent/DE60306540T2/de not_active Expired - Lifetime
- 2003-10-24 KR KR1020057007633A patent/KR101000731B1/ko not_active Expired - Fee Related
- 2003-10-24 PT PT03776869T patent/PT1556377E/pt unknown
- 2003-10-24 WO PCT/EP2003/011805 patent/WO2004039799A1/en not_active Ceased
- 2003-10-24 RU RU2005116974/04A patent/RU2005116974A/ru not_active Application Discontinuation
- 2003-10-24 EP EP03776869A patent/EP1556377B1/en not_active Expired - Lifetime
- 2003-10-24 US US10/532,847 patent/US7312179B2/en not_active Expired - Fee Related
- 2003-10-24 AU AU2003286140A patent/AU2003286140A1/en not_active Abandoned
- 2003-10-24 CA CA2501739A patent/CA2501739C/en not_active Expired - Fee Related
- 2003-10-24 MX MXPA05004463A patent/MXPA05004463A/es active IP Right Grant
- 2003-10-24 DK DK03776869T patent/DK1556377T3/da active
- 2003-10-24 BR BR0315857-8A patent/BR0315857A/pt not_active Application Discontinuation
- 2003-10-24 CN CNB2003801021700A patent/CN100526310C/zh not_active Expired - Fee Related
- 2003-10-24 AT AT03776869T patent/ATE331714T1/de not_active IP Right Cessation
- 2003-10-24 JP JP2004547558A patent/JP4673061B2/ja not_active Expired - Fee Related
- 2003-10-24 ES ES03776869T patent/ES2266881T3/es not_active Expired - Lifetime
- 2003-10-27 TW TW092129757A patent/TW200412848A/zh unknown
- 2003-10-30 GT GT200300236A patent/GT200300236A/es unknown
- 2003-10-31 AR ARP030104010A patent/AR041747A1/es unknown
-
2005
- 2005-04-01 ZA ZA200502644A patent/ZA200502644B/en unknown
- 2005-04-29 EC EC2005005770A patent/ECSP055770A/es unknown
- 2005-04-29 CO CO05040972A patent/CO5550397A2/es not_active Application Discontinuation
Patent Citations (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB2126587A (en) * | 1982-09-13 | 1984-03-28 | Sandoz Ltd | Fungicidal thiophene derivatives |
| US4743602A (en) * | 1986-07-16 | 1988-05-10 | Imperial Chemical Industries Plc | Thiophene cyclopropyl amine compounds, compositions and fungicidal use |
Also Published As
| Publication number | Publication date |
|---|---|
| DE60306540T2 (de) | 2007-06-28 |
| AR041747A1 (es) | 2005-05-26 |
| CO5550397A2 (es) | 2005-08-31 |
| WO2004039799A1 (en) | 2004-05-13 |
| KR101000731B1 (ko) | 2010-12-14 |
| KR20050071648A (ko) | 2005-07-07 |
| AU2003286140A1 (en) | 2004-05-25 |
| JP2006508089A (ja) | 2006-03-09 |
| US20060030567A1 (en) | 2006-02-09 |
| PT1556377E (pt) | 2006-10-31 |
| MXPA05004463A (es) | 2005-07-26 |
| ZA200502644B (en) | 2005-11-23 |
| TW200412848A (en) | 2004-08-01 |
| DE60306540D1 (en) | 2006-08-10 |
| BR0315857A (pt) | 2005-09-20 |
| ATE331714T1 (de) | 2006-07-15 |
| EP1556377B1 (en) | 2006-06-28 |
| GT200300236A (es) | 2004-06-23 |
| ECSP055770A (es) | 2005-08-11 |
| ES2266881T3 (es) | 2007-03-01 |
| CA2501739C (en) | 2011-04-12 |
| CA2501739A1 (en) | 2004-05-13 |
| DK1556377T3 (da) | 2006-10-23 |
| EP1556377A1 (en) | 2005-07-27 |
| GB0225554D0 (en) | 2002-12-11 |
| JP4673061B2 (ja) | 2011-04-20 |
| RU2005116974A (ru) | 2006-03-27 |
| CN1708496A (zh) | 2005-12-14 |
| US7312179B2 (en) | 2007-12-25 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| C06 | Publication | ||
| PB01 | Publication | ||
| C10 | Entry into substantive examination | ||
| SE01 | Entry into force of request for substantive examination | ||
| C14 | Grant of patent or utility model | ||
| GR01 | Patent grant | ||
| C17 | Cessation of patent right | ||
| CF01 | Termination of patent right due to non-payment of annual fee |
Granted publication date: 20090812 Termination date: 20131024 |