CL2023001195A1 - Compuestos bicíclicos y usos de los mismos para el tratamiento de enfermedades. - Google Patents

Compuestos bicíclicos y usos de los mismos para el tratamiento de enfermedades.

Info

Publication number
CL2023001195A1
CL2023001195A1 CL2023001195A CL2023001195A CL2023001195A1 CL 2023001195 A1 CL2023001195 A1 CL 2023001195A1 CL 2023001195 A CL2023001195 A CL 2023001195A CL 2023001195 A CL2023001195 A CL 2023001195A CL 2023001195 A1 CL2023001195 A1 CL 2023001195A1
Authority
CL
Chile
Prior art keywords
diseases
treatment
bicyclic compounds
compounds
compositions
Prior art date
Application number
CL2023001195A
Other languages
English (en)
Spanish (es)
Inventor
Leen Kawas
Kevin Church
Robert Taylor
Jewel Johnston
Douglas Boatman
Original Assignee
Athira Pharma Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Athira Pharma Inc filed Critical Athira Pharma Inc
Publication of CL2023001195A1 publication Critical patent/CL2023001195A1/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Neurosurgery (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Hospice & Palliative Care (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Psychiatry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
CL2023001195A 2020-11-02 2023-04-26 Compuestos bicíclicos y usos de los mismos para el tratamiento de enfermedades. CL2023001195A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US202063108660P 2020-11-02 2020-11-02

Publications (1)

Publication Number Publication Date
CL2023001195A1 true CL2023001195A1 (es) 2023-10-20

Family

ID=81384389

Family Applications (2)

Application Number Title Priority Date Filing Date
CL2023001195A CL2023001195A1 (es) 2020-11-02 2023-04-26 Compuestos bicíclicos y usos de los mismos para el tratamiento de enfermedades.
CL2024000340A CL2024000340A1 (es) 2020-11-02 2024-02-02 Compuestos bicíclicos y usos de los mismos para el tratamiento de enfermedades

Family Applications After (1)

Application Number Title Priority Date Filing Date
CL2024000340A CL2024000340A1 (es) 2020-11-02 2024-02-02 Compuestos bicíclicos y usos de los mismos para el tratamiento de enfermedades

Country Status (12)

Country Link
US (1) US20240025903A1 (https=)
EP (1) EP4236944A4 (https=)
JP (1) JP2023550543A (https=)
KR (1) KR20230104191A (https=)
CN (2) CN119684295A (https=)
AR (1) AR124637A1 (https=)
AU (1) AU2021371026A1 (https=)
CA (1) CA3196582A1 (https=)
CL (2) CL2023001195A1 (https=)
IL (1) IL302465A (https=)
MX (1) MX2023004942A (https=)
WO (1) WO2022094400A1 (https=)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR20240121239A (ko) * 2021-12-17 2024-08-08 아티라 파마, 인코포레이티드 질환 치료를 위한 이환식 화합물의 용도
EP4518864A1 (en) * 2022-05-04 2025-03-12 Athira Pharma, Inc. Methods of treating neuropathies
JP2025515045A (ja) * 2022-05-04 2025-05-13 アティラ・ファーマ・インコーポレイテッド 神経炎症病態を治療する方法
EP4618996A1 (en) 2022-11-18 2025-09-24 Athira Pharma, Inc. Methods of treating inflammatory conditions

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6184223B1 (en) * 1995-10-27 2001-02-06 Molecumetics Ltd. Reverse-turn mimetics and methods relating thereto
AU2003284120A1 (en) * 2002-10-17 2004-05-04 Myriad Genetics, Inc. Reverse-turn mimetics and composition and methods relating thereto
US7192976B2 (en) * 2002-12-21 2007-03-20 Angion Biomedica Corporation Small molecule modulators of hepatocyte growth factor (scatter factor) activity
AU2005289560A1 (en) * 2004-09-28 2006-04-06 Angion Biomedica Corp. Small molecule modulators of cytokine activity
US7879898B1 (en) * 2006-02-14 2011-02-01 Angion Biomedica Corp. Hepatocyte growth factor pathway activators in chronic obstructive pulmonary disease
EP1947085A1 (en) * 2007-01-19 2008-07-23 Laboratorios del Dr. Esteve S.A. Substituted indole sulfonamide compounds, their preparation and use as medicaments
CN102186853A (zh) * 2008-10-14 2011-09-14 株式会社棱镜生物实验室 治疗癌症α-螺旋模拟物
WO2014025832A1 (en) * 2012-08-06 2014-02-13 University Of Southern California Wnt modulators for the protection, mitigation and treatment of radiation injury
WO2017047762A1 (ja) * 2015-09-18 2017-03-23 国立大学法人鳥取大学 低分子化合物による癌と線維化の抑制と再生促進の効果

Also Published As

Publication number Publication date
EP4236944A4 (en) 2024-09-04
TW202233622A (zh) 2022-09-01
US20240025903A1 (en) 2024-01-25
WO2022094400A1 (en) 2022-05-05
MX2023004942A (es) 2023-07-06
EP4236944A1 (en) 2023-09-06
JP2023550543A (ja) 2023-12-01
CA3196582A1 (en) 2022-05-05
AR124637A1 (es) 2023-04-19
CN116568301A (zh) 2023-08-08
AU2021371026A9 (en) 2024-04-18
KR20230104191A (ko) 2023-07-07
IL302465A (en) 2023-06-01
CL2024000340A1 (es) 2024-08-16
CN119684295A (zh) 2025-03-25
AU2021371026A1 (en) 2023-06-15

Similar Documents

Publication Publication Date Title
CL2024000340A1 (es) Compuestos bicíclicos y usos de los mismos para el tratamiento de enfermedades
CO2021007993A2 (es) Compuestos de 2‐formil‐3‐hidroxifeniloximetilo capaces de modular la hemoglobina
MX2021007468A (es) Compuestos que participan en la union cooperativa y usos de los mismos.
ECSP20018487A (es) Activadores de piruvato quinasas para usar en el tratamiento de trastornos en la sangre
CO2022010547A2 (es) Compuestos y usos de los mismos
DOP2020000040A (es) Compuestos espirocíclicos y sus métodos de preparación y uso
PA8570701A1 (es) Compuestos que modulan la actividad de ppar y procedimientos para su preparacion
DOP2024000028A (es) Degradadores bifuncionales de quinasas asociadas al receptor de interleucina 1 y usos terapéuticos de los mismos
MX2020012158A (es) Inhibidores de magl.
MX2022000550A (es) Imidazopirimidinas como inhibidores de eed y uso de estas.
NI202000014A (es) Compuestos espirocíclicos y sus métodos de preparación y uso
MX350890B (es) Agentes para tratar trastornos que implican la modulación de receptores de rianodina.
MX2022006862A (es) Inhibidores duales de magl y faah.
CO2023010940A2 (es) Compuestos moduladores de gcn2 y usos de los mismos
CL2021001656A1 (es) Compuestos de imidazopiridina e imidazopiridina y sus usos.
CL2021002521A1 (es) Compuestos heteocíclicos y sus usos.
MX2024013040A (es) Pirfenidona enriquecida con deuterio y metodos para su uso
CL2024003870A1 (es) Compuestos de degradación de wee1 y usos de los mismos
DOP2022000127A (es) Triterpenoides sintéticos con sustituyentes a base de nitrógeno en c-17 y métodos de uso de los mismos.
MX2018009189A (es) Compuestos de anillo de siete miembros de pirimidina.
CL2025003186A1 (es) Moduladores de nk3 y usos de los mismos.
CL2024001748A1 (es) Usos de compuestos biciclicos para el tratamiento de enfermedades.
CL2022002589A1 (es) Tratamiento de trastornos respiratorios
CO2023003078A2 (es) Compuestos como moduladores de bis-fosfoglicerato mutasa para el tratamiento de la anemia de células falciforme
ECSP22019177A (es) Proteínas de fusión nkg2d y sus usos