CL2022001888A1 - Nuevo derivado de pirazol - Google Patents
Nuevo derivado de pirazolInfo
- Publication number
- CL2022001888A1 CL2022001888A1 CL2022001888A CL2022001888A CL2022001888A1 CL 2022001888 A1 CL2022001888 A1 CL 2022001888A1 CL 2022001888 A CL2022001888 A CL 2022001888A CL 2022001888 A CL2022001888 A CL 2022001888A CL 2022001888 A1 CL2022001888 A1 CL 2022001888A1
- Authority
- CL
- Chile
- Prior art keywords
- pyrazole derivative
- new pyrazole
- new
- salt
- pharmaceutical composition
- Prior art date
Links
- 150000003217 pyrazoles Chemical class 0.000 title 1
- 239000008194 pharmaceutical composition Substances 0.000 abstract 1
- -1 pyrazole derivative compound Chemical class 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
- 239000000126 substance Substances 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
- A61K31/437—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
- A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/02—Antineoplastic agents specific for leukemia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/04—Antineoplastic agents specific for metastasis
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D519/00—Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Epidemiology (AREA)
- Neurosurgery (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Oncology (AREA)
- Rheumatology (AREA)
- Psychiatry (AREA)
- Psychology (AREA)
- Hospice & Palliative Care (AREA)
- Hematology (AREA)
- Pain & Pain Management (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Abstract
La presente invención proporciona un compuesto derivado de pirazol novedoso representado por la fórmula química I o una sal del mismo, y una composición farmacéutica que comprende el mismo.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
KR20200004471 | 2020-01-13 |
Publications (1)
Publication Number | Publication Date |
---|---|
CL2022001888A1 true CL2022001888A1 (es) | 2023-02-24 |
Family
ID=76864348
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CL2022001888A CL2022001888A1 (es) | 2020-01-13 | 2022-07-12 | Nuevo derivado de pirazol |
Country Status (13)
Country | Link |
---|---|
US (1) | US20230067461A1 (es) |
EP (1) | EP4105206A1 (es) |
JP (1) | JP2023511302A (es) |
KR (1) | KR102333863B1 (es) |
CN (1) | CN114945561A (es) |
AU (1) | AU2021208915B2 (es) |
BR (1) | BR112022013849A2 (es) |
CA (1) | CA3167675A1 (es) |
CL (1) | CL2022001888A1 (es) |
CO (1) | CO2022010431A2 (es) |
IL (1) | IL294674A (es) |
MX (1) | MX2022008665A (es) |
WO (1) | WO2021145655A1 (es) |
Families Citing this family (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JP2023536764A (ja) * | 2021-02-25 | 2023-08-29 | アプタバイオ セラピューティクス インコーポレイテッド | 新規なピラゾール誘導体 |
TW202334109A (zh) * | 2022-02-25 | 2023-09-01 | 南韓商阿普塔生物治療公司 | 新穎吡唑衍生物 |
Family Cites Families (15)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DK574976A (da) * | 1976-01-16 | 1977-07-17 | Du Pont | Substituerede cycloalkanpyrazoler samt deres fremstilling og anvendelse |
AR045037A1 (es) * | 2003-07-10 | 2005-10-12 | Aventis Pharma Sa | Tetrahidro-1h-pirazolo [3,4-c] piridinas sustituidas, composiciones que las contienen y su utilizacion. |
KR100863692B1 (ko) * | 2006-12-08 | 2008-10-15 | 울산대학교 산학협력단 | 퇴행성질환 및 염증질환에 대한 예방치료 효과를 갖는7-하이드록시-6-메톡시-1,2,3,4-테트라하이드로이소퀴놀린유도체 |
EP2151433A1 (en) * | 2008-08-05 | 2010-02-10 | Institut Pasteur | Alkoxypyrazoles and the process for their preparation |
TWI389913B (zh) * | 2008-09-08 | 2013-03-21 | Lg Life Sciences Ltd | 并合雜環化合物 |
FR2953839A1 (fr) * | 2009-12-14 | 2011-06-17 | Sanofi Aventis | Nouveaux derives d'(heterocycle-piperidine condensee)-(piperazinyl)-1alcanone ou d'(heterocycle-pyrrolidine condensee)-(piperazinyl)-1alcanone et leur utilisation comme inhibiteurs de p75 |
EP2361911A1 (en) * | 2010-02-18 | 2011-08-31 | GenKyoTex SA | Pyrazolo piperidine derivatives as NADPH oxidase inhibitors |
EP2361912A1 (en) * | 2010-02-18 | 2011-08-31 | GenKyoTex SA | Pyrazolo piperidine derivatives as NADPH oxidase inhibitors |
KR20120098462A (ko) * | 2011-02-28 | 2012-09-05 | 이화여자대학교 산학협력단 | 피라졸 유도체, 이의 제조방법 및 이를 포함하는 골다공증 예방 및 치료용 조성물 |
TWI599567B (zh) * | 2013-03-14 | 2017-09-21 | 健生藥品公司 | P2x7調節劑 |
JP6527167B2 (ja) | 2014-03-27 | 2019-06-05 | ヤンセン ファーマシューティカ エヌ.ベー. | ROS1阻害剤としての置換4,5,6,7−テトラヒドロ−ピラゾロ[1,5−a]ピリミジン誘導体および2,3−ジヒドロ−1H−イミダゾ[1,2−b]ピラゾール誘導体 |
EP3134406A1 (en) * | 2014-04-24 | 2017-03-01 | Dart Neuroscience (Cayman) Ltd | Substituted 2,4,5,6-tetrahydropyrrolo[3,4-c]pyrazole and 4,5,6,7-tetrahydro-2h-pyrazolo [4,3-c]pyridine compounds as glyt1 inhibitors |
US10584118B2 (en) | 2015-06-22 | 2020-03-10 | Actelion Pharmaceuticals Ltd | NADPH oxidase 4 inhibitors |
JP6508721B2 (ja) | 2015-09-28 | 2019-05-08 | 株式会社Screenホールディングス | 基板処理方法および基板処理装置 |
WO2019141957A1 (en) * | 2018-01-19 | 2019-07-25 | Cado Biotechnology Ivs | N-pyrimidinyl hydroxy pyrazole derivatives and uses thereof |
-
2021
- 2021-01-12 WO PCT/KR2021/000425 patent/WO2021145655A1/ko unknown
- 2021-01-12 CA CA3167675A patent/CA3167675A1/en active Pending
- 2021-01-12 CN CN202180009272.6A patent/CN114945561A/zh active Pending
- 2021-01-12 JP JP2022543171A patent/JP2023511302A/ja active Pending
- 2021-01-12 AU AU2021208915A patent/AU2021208915B2/en active Active
- 2021-01-12 BR BR112022013849A patent/BR112022013849A2/pt not_active Application Discontinuation
- 2021-01-12 KR KR1020210004079A patent/KR102333863B1/ko active IP Right Grant
- 2021-01-12 US US17/791,983 patent/US20230067461A1/en active Pending
- 2021-01-12 MX MX2022008665A patent/MX2022008665A/es unknown
- 2021-01-12 IL IL294674A patent/IL294674A/en unknown
- 2021-01-12 EP EP21740932.5A patent/EP4105206A1/en active Pending
-
2022
- 2022-07-12 CL CL2022001888A patent/CL2022001888A1/es unknown
- 2022-07-26 CO CONC2022/0010431A patent/CO2022010431A2/es unknown
Also Published As
Publication number | Publication date |
---|---|
EP4105206A1 (en) | 2022-12-21 |
JP2023511302A (ja) | 2023-03-17 |
AU2021208915B2 (en) | 2024-02-22 |
US20230067461A1 (en) | 2023-03-02 |
IL294674A (en) | 2022-09-01 |
WO2021145655A1 (ko) | 2021-07-22 |
KR102333863B1 (ko) | 2021-12-03 |
AU2021208915A1 (en) | 2022-09-01 |
MX2022008665A (es) | 2022-08-10 |
KR20210091063A (ko) | 2021-07-21 |
CN114945561A (zh) | 2022-08-26 |
CA3167675A1 (en) | 2021-07-22 |
BR112022013849A2 (pt) | 2022-09-13 |
CO2022010431A2 (es) | 2022-08-09 |
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