CL2021001177A1 - Compuestos químicos - Google Patents
Compuestos químicosInfo
- Publication number
- CL2021001177A1 CL2021001177A1 CL2021001177A CL2021001177A CL2021001177A1 CL 2021001177 A1 CL2021001177 A1 CL 2021001177A1 CL 2021001177 A CL2021001177 A CL 2021001177A CL 2021001177 A CL2021001177 A CL 2021001177A CL 2021001177 A1 CL2021001177 A1 CL 2021001177A1
- Authority
- CL
- Chile
- Prior art keywords
- compounds
- atopic dermatitis
- chemical compounds
- inhibitors
- pruritus
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/4985—Pyrazines or piperazines ortho- or peri-condensed with heterocyclic ring systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
- A61K31/52—Purines, e.g. adenine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D473/00—Heterocyclic compounds containing purine ring systems
- C07D473/26—Heterocyclic compounds containing purine ring systems with an oxygen, sulphur, or nitrogen atom directly attached in position 2 or 6, but not in both
- C07D473/32—Nitrogen atom
- C07D473/34—Nitrogen atom attached in position 6, e.g. adenine
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Dermatology (AREA)
- Engineering & Computer Science (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Abstract
La presente invención describe nuevos compuestos, o sales farmacéuticamente aceptables de los mismos, composiciones farmacéuticas que los contienen y sus usos médicos. Los compuestos de la invención tienen actividad como inhibidores de Janus Kinase y son útiles en el tratamiento o control del prurito asociado con dermatitis alérgica, dermatitis atópica en animales y otros trastornos e indicaciones en las que sería deseable la inmunosupresión/inmunomodulación. También se describen en este documento métodos para tratar el prurito y la dermatitis atópica mediante la administración de los compuestos de la invención, los cuales son inhibidores de JAK 1.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US201862755679P | 2018-11-05 | 2018-11-05 |
Publications (1)
Publication Number | Publication Date |
---|---|
CL2021001177A1 true CL2021001177A1 (es) | 2022-05-27 |
Family
ID=70458378
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CL2021001177A CL2021001177A1 (es) | 2018-11-05 | 2021-05-05 | Compuestos químicos |
Country Status (11)
Country | Link |
---|---|
US (1) | US10744136B2 (es) |
EP (1) | EP3877389A4 (es) |
JP (1) | JP2022506682A (es) |
KR (1) | KR20210072125A (es) |
CN (1) | CN113272306A (es) |
AU (1) | AU2019375412A1 (es) |
BR (1) | BR112021008742A2 (es) |
CA (1) | CA3118488A1 (es) |
CL (1) | CL2021001177A1 (es) |
MX (1) | MX2021005334A (es) |
WO (1) | WO2020096948A1 (es) |
Families Citing this family (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US20090053786A1 (en) | 2007-07-09 | 2009-02-26 | Yung-Hsiang Kao | Prevention of disulfide bond reduction during recombinant production of polypeptides |
Family Cites Families (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
KR100415791B1 (ko) * | 1998-06-19 | 2004-01-24 | 화이자 프로덕츠 인코포레이티드 | 피롤로[2,3-디]피리미딘 화합물 |
BRPI0809992A2 (pt) * | 2007-04-02 | 2014-10-14 | Palau Pharma Sa | Derivados de pirrolopirimidina |
RU2493157C2 (ru) * | 2008-08-20 | 2013-09-20 | Пфайзер Инк. | ПРОИЗВОДНЫЕ ПИРРОЛО[2,3-d]ПИРИМИДИНА |
DK2958921T3 (da) * | 2013-02-22 | 2017-11-06 | Pfizer | Pyrrolo[2,3-D]pyrimidin-derivater som hæmmere af Janus kinaser (JAK) |
KR102275326B1 (ko) * | 2013-06-07 | 2021-07-12 | 지앙수 헨그루이 메디슨 컴퍼니 리미티드 | 야누스 키나제(jak) 억제제의 바이설페이트 및 그의 제조 방법 |
EP3180344B1 (en) * | 2014-08-12 | 2019-09-18 | Pfizer Inc | Pyrrolo[2,3-d]pyrimidine derivatives useful for inhibiting janus kinase |
JP7462951B2 (ja) * | 2018-03-21 | 2024-04-08 | リャオ,シビン | Jak阻害剤 |
-
2019
- 2019-11-04 MX MX2021005334A patent/MX2021005334A/es unknown
- 2019-11-04 JP JP2021524221A patent/JP2022506682A/ja active Pending
- 2019-11-04 AU AU2019375412A patent/AU2019375412A1/en active Pending
- 2019-11-04 CN CN201980087712.2A patent/CN113272306A/zh active Pending
- 2019-11-04 BR BR112021008742-7A patent/BR112021008742A2/pt unknown
- 2019-11-04 US US16/673,014 patent/US10744136B2/en active Active
- 2019-11-04 WO PCT/US2019/059634 patent/WO2020096948A1/en unknown
- 2019-11-04 KR KR1020217016999A patent/KR20210072125A/ko unknown
- 2019-11-04 CA CA3118488A patent/CA3118488A1/en active Pending
- 2019-11-04 EP EP19882784.2A patent/EP3877389A4/en active Pending
-
2021
- 2021-05-05 CL CL2021001177A patent/CL2021001177A1/es unknown
Also Published As
Publication number | Publication date |
---|---|
JP2022506682A (ja) | 2022-01-17 |
MX2021005334A (es) | 2021-06-23 |
WO2020096948A1 (en) | 2020-05-14 |
US10744136B2 (en) | 2020-08-18 |
AU2019375412A1 (en) | 2021-06-03 |
BR112021008742A2 (pt) | 2021-08-10 |
KR20210072125A (ko) | 2021-06-16 |
EP3877389A1 (en) | 2021-09-15 |
CN113272306A (zh) | 2021-08-17 |
CA3118488A1 (en) | 2020-05-14 |
US20200138811A1 (en) | 2020-05-07 |
EP3877389A4 (en) | 2022-07-13 |
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