CL2009001009A1 - Metodo para inhibir la espermatogenesis en un hombre que comprende administrarle un agonista del receptor de androgenos y una composicion que comprende un compuesto derivado de 19-norpregnanos 21 sustituidos. - Google Patents

Metodo para inhibir la espermatogenesis en un hombre que comprende administrarle un agonista del receptor de androgenos y una composicion que comprende un compuesto derivado de 19-norpregnanos 21 sustituidos.

Info

Publication number
CL2009001009A1
CL2009001009A1 CL2009001009A CL2009001009A CL2009001009A1 CL 2009001009 A1 CL2009001009 A1 CL 2009001009A1 CL 2009001009 A CL2009001009 A CL 2009001009A CL 2009001009 A CL2009001009 A CL 2009001009A CL 2009001009 A1 CL2009001009 A1 CL 2009001009A1
Authority
CL
Chile
Prior art keywords
man
administering
substituted
composition
receptor agonist
Prior art date
Application number
CL2009001009A
Other languages
English (en)
Inventor
Joseph S Podolski
Ronald D Wiehle
Original Assignee
Repros Therapeutics Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Repros Therapeutics Inc filed Critical Repros Therapeutics Inc
Publication of CL2009001009A1 publication Critical patent/CL2009001009A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/565Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
    • A61K31/568Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol substituted in positions 10 and 13 by a chain having at least one carbon atom, e.g. androstanes, e.g. testosterone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/565Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
    • A61K31/568Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol substituted in positions 10 and 13 by a chain having at least one carbon atom, e.g. androstanes, e.g. testosterone
    • A61K31/5685Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol substituted in positions 10 and 13 by a chain having at least one carbon atom, e.g. androstanes, e.g. testosterone having an oxo group in position 17, e.g. androsterone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/58Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids containing heterocyclic rings, e.g. danazol, stanozolol, pancuronium or digitogenin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • A61P15/16Masculine contraceptives

Abstract

Método para inhibir la espermatogénesis en un hombre que comprende administrarle un agonista del receptor de andrógenos y una composición que comprende un compuesto derivado de 19-norpregnanos 21 sustituidos.
CL2009001009A 2008-04-28 2009-04-28 Metodo para inhibir la espermatogenesis en un hombre que comprende administrarle un agonista del receptor de androgenos y una composicion que comprende un compuesto derivado de 19-norpregnanos 21 sustituidos. CL2009001009A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US4844408P 2008-04-28 2008-04-28

Publications (1)

Publication Number Publication Date
CL2009001009A1 true CL2009001009A1 (es) 2009-06-19

Family

ID=40756947

Family Applications (1)

Application Number Title Priority Date Filing Date
CL2009001009A CL2009001009A1 (es) 2008-04-28 2009-04-28 Metodo para inhibir la espermatogenesis en un hombre que comprende administrarle un agonista del receptor de androgenos y una composicion que comprende un compuesto derivado de 19-norpregnanos 21 sustituidos.

Country Status (4)

Country Link
AR (1) AR072781A1 (es)
CL (1) CL2009001009A1 (es)
TW (1) TW200950788A (es)
WO (1) WO2009134713A1 (es)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2016054197A1 (en) * 2014-09-30 2016-04-07 University Of Tennessee Research Foundation In situ gelling form for long-acting drug delivery

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US8173626B2 (en) * 2006-03-08 2012-05-08 Danco Laboratories Llc Methods, dosing regimens and medications using anti-progestational agents for the treatment of disorders

Also Published As

Publication number Publication date
AR072781A1 (es) 2010-09-22
WO2009134713A1 (en) 2009-11-05
TW200950788A (en) 2009-12-16

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