CL2007002491A1 - Compuestos derivados de piridinona sustituida, antagonistas de la hormona concentradora de melanina (mch); composicion farmaceutica; y uso para influir en el comportamiento de alimentacion en un mamifero, trastornos metabolicos, trastornos de la alimentacion como obesidad, bulimia, caquexia, anorexia nerviosa, hiperfagia. - Google Patents
Compuestos derivados de piridinona sustituida, antagonistas de la hormona concentradora de melanina (mch); composicion farmaceutica; y uso para influir en el comportamiento de alimentacion en un mamifero, trastornos metabolicos, trastornos de la alimentacion como obesidad, bulimia, caquexia, anorexia nerviosa, hiperfagia.Info
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- CL2007002491A1 CL2007002491A1 CL2007002491A CL2007002491A CL2007002491A1 CL 2007002491 A1 CL2007002491 A1 CL 2007002491A1 CL 2007002491 A CL2007002491 A CL 2007002491A CL 2007002491 A CL2007002491 A CL 2007002491A CL 2007002491 A1 CL2007002491 A1 CL 2007002491A1
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- mammal
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- hyperphagia
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Abstract
Compuestos derivados de piridinona sustituida, antagonistas de la hormona concentradora de melanina mch; composición farmacéutica; y uso para influir en el comportamiento de alimentación en un mamífero.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP06119523 | 2006-08-25 |
Publications (1)
Publication Number | Publication Date |
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CL2007002491A1 true CL2007002491A1 (es) | 2008-01-18 |
Family
ID=38896082
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CL2007002491A CL2007002491A1 (es) | 2006-08-25 | 2007-08-24 | Compuestos derivados de piridinona sustituida, antagonistas de la hormona concentradora de melanina (mch); composicion farmaceutica; y uso para influir en el comportamiento de alimentacion en un mamifero, trastornos metabolicos, trastornos de la alimentacion como obesidad, bulimia, caquexia, anorexia nerviosa, hiperfagia. |
Country Status (17)
Country | Link |
---|---|
US (2) | US8067590B2 (es) |
EP (2) | EP2383259A1 (es) |
JP (1) | JP5073746B2 (es) |
KR (1) | KR20090047542A (es) |
CN (1) | CN101506195A (es) |
AR (1) | AR062510A1 (es) |
AU (1) | AU2007287601B2 (es) |
BR (1) | BRPI0716579A2 (es) |
CA (1) | CA2657183A1 (es) |
CL (1) | CL2007002491A1 (es) |
IL (1) | IL197128A (es) |
MX (1) | MX2009000334A (es) |
NZ (1) | NZ575520A (es) |
RU (1) | RU2453543C2 (es) |
TW (1) | TW200817366A (es) |
WO (1) | WO2008022979A1 (es) |
ZA (1) | ZA200810404B (es) |
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CN101945872B (zh) | 2008-01-11 | 2014-07-23 | 阿尔巴尼分子研究公司 | 作为mch拮抗剂的(1-吖嗪酮)-取代的吡啶并吲哚 |
WO2009103478A1 (en) * | 2008-02-19 | 2009-08-27 | Boehringer Ingelheim International Gmbh | Pyridone and pyridazinone derivatives as mch antagonists |
CA2967254C (en) | 2008-02-29 | 2019-03-26 | Lantheus Medical Imaging, Inc. | Contrast agents for applications including imaging cancer |
MX2010012848A (es) | 2008-06-03 | 2011-03-01 | Intermune Inc | Compuestos y metodos para tratar trastornos inflamatorios y fibroticos. |
AR075401A1 (es) | 2009-02-13 | 2011-03-30 | Sanofi Aventis | Indanos sustituidos, procesos para su preparacion y uso de los mismos como un medicamento |
UY32443A (es) | 2009-02-13 | 2010-09-30 | Sanofi Aventis | Nuevos tetrahidronaftalenos, procesos para su preparación y uso de los mismos como medicamento. |
US8629158B2 (en) | 2009-07-01 | 2014-01-14 | Albany Molecular Research, Inc. | Azabicycloalkane-indole and azabicycloalkane-pyrrolo-pyridine MCH-1 antagonists, methods of making, and use thereof |
WO2011003021A1 (en) | 2009-07-01 | 2011-01-06 | Albany Molecular Research, Inc. | Azinone-substituted azabicycloalkane-indole and azabicycloalkane-pyrrolo-pyridine mch-1 antagonists, methods of making, and use thereof |
EP2448585B1 (en) | 2009-07-01 | 2014-01-01 | Albany Molecular Research, Inc. | Azinone-substituted azepino[b]indole and pyrido-pyrrolo-azepine mch-1 antagonists, methods of making, and use thereof |
US8618299B2 (en) | 2009-07-01 | 2013-12-31 | Albany Molecular Research, Inc. | Azinone-substituted azapolycycle MCH-1 antagonists, methods of making, and use thereof |
US20110021570A1 (en) | 2009-07-23 | 2011-01-27 | Nancy-Ellen Haynes | Pyridone glucokinase activators |
JP6092628B2 (ja) | 2010-02-08 | 2017-03-08 | ランセウス メディカル イメージング, インコーポレイテッド | 造影剤およびその中間体を合成するための方法および装置 |
WO2012088124A2 (en) | 2010-12-21 | 2012-06-28 | Albany Molecular Research, Inc. | Tetrahydro-azacarboline mch-1 antagonists, methods of making, and uses thereof |
US8697700B2 (en) | 2010-12-21 | 2014-04-15 | Albany Molecular Research, Inc. | Piperazinone-substituted tetrahydro-carboline MCH-1 antagonists, methods of making, and uses thereof |
SG2014013767A (en) | 2011-09-09 | 2014-05-29 | Lantheus Medical Imaging Inc | Compositions, methods, and systems for the synthesis and use of imaging agents |
US9365540B2 (en) | 2012-01-12 | 2016-06-14 | Takeda Pharmaceutical Company Limited | Benzimidazole derivatives as MCH receptor antagonists |
US8933079B2 (en) * | 2012-03-07 | 2015-01-13 | Boehringer Ingelheim International Gmbh | Pyridone and pyridazinone derivatives as anti-obesity agents |
WO2013168760A1 (ja) * | 2012-05-10 | 2013-11-14 | 武田薬品工業株式会社 | 芳香環化合物 |
JP6186434B2 (ja) | 2012-07-18 | 2017-08-23 | サンシャイン・レイク・ファーマ・カンパニー・リミテッドSunshine Lake Pharma Co.,Ltd. | 窒素複素環誘導体及びその医薬品への応用 |
AU2013203000B9 (en) | 2012-08-10 | 2017-02-02 | Lantheus Medical Imaging, Inc. | Compositions, methods, and systems for the synthesis and use of imaging agents |
AR092742A1 (es) | 2012-10-02 | 2015-04-29 | Intermune Inc | Piridinonas antifibroticas |
EP3083584B1 (en) | 2013-12-19 | 2018-02-21 | Sunshine Lake Pharma Co., Ltd. | Nitrogenous heterocyclic derivatives and their application in the treatment of tissue fibrosis |
CN106459042B (zh) | 2014-04-02 | 2019-06-28 | 英特穆恩公司 | 抗纤维化吡啶酮类 |
US10540723B1 (en) | 2014-07-21 | 2020-01-21 | State Farm Mutual Automobile Insurance Company | Methods of providing insurance savings based upon telematics and usage-based insurance |
CN117538462B (zh) * | 2024-01-10 | 2024-03-26 | 地奥集团成都药业股份有限公司 | 一种氨氯地平贝那普利胶囊有关物质的检测方法 |
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CA2386474A1 (en) | 1999-09-20 | 2001-03-29 | Takeda Chemical Industries, Ltd. | Melanin concentrating hormone antagonist |
CA2407149C (en) | 2000-04-28 | 2010-10-12 | Takeda Chemical Industries, Ltd. | Melanin-concentrating hormone antagonist |
MXPA04004830A (es) * | 2001-11-22 | 2004-07-30 | Ono Pharmaceutical Co | Compuestos derivados de piperidin-2-ona, y composiciones farmaceuticas que los contienen como ingredientes activos. |
WO2003059891A1 (en) | 2002-01-18 | 2003-07-24 | Pharmacia Corporation | Substituted pyridazinones as inhibitors of p38 |
ES2334990T3 (es) | 2002-02-14 | 2010-03-18 | Pharmacia Corporation | Piridinonas sustituidas como moduladores de p38 map quinasa. |
DE10238865A1 (de) | 2002-08-24 | 2004-03-11 | Boehringer Ingelheim International Gmbh | Neue Carbonsäureamid-Verbindungen mit MCH-antagonistischer Wirkung, diese Verbindungen enthaltende Arzneimittel und Verfahren zu ihrer Herstellung |
DE10250708A1 (de) | 2002-10-31 | 2004-05-19 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | Neue Alkin-Verbindungen mit MCH-antagonistischer Wirkung und diese Verbindungen enthaltende Arzneimittel |
DE10250743A1 (de) | 2002-10-31 | 2004-05-19 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | Neue Amid-Verbindungen mit MCH-antagonistischer Wirkung und diese Verbindungen enthaltende Arzneimittel |
US7183287B2 (en) | 2003-04-03 | 2007-02-27 | Pharmacia Corporation | Substituted pyrimidinones |
WO2005007632A1 (en) | 2003-07-18 | 2005-01-27 | Pharmacia Corporation | Substituted pyridazinones as inhibitors of p38 |
CL2004002050A1 (es) | 2003-08-13 | 2005-06-03 | Pharmacia Corp Sa Organizada B | Compuestos derivados de piridinonas sustituidas; su uso en el tratamiento de afecciones causadas o exacerbadas por actividad p38 map kinasa y/o tnf no regulada, tales como inflamaciones, tumores, sida y otros. |
DE10360745A1 (de) | 2003-12-23 | 2005-07-28 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | Neue Amid-Verbindungen mit MCH-antagonistischer Wirkung und diese Verbindungen enthaltende Arzneimittel |
CA2558272C (en) | 2004-03-05 | 2011-02-15 | Banyu Pharmaceutical Co., Ltd. | Pyridone derivative |
DE102004010893A1 (de) | 2004-03-06 | 2005-09-22 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | Neue ß-Ketoamid-Verbindungen mit MCH-antagonistischer Wirkung und diese Verbindungen enthaltende Arzneimittel |
DE102004017930A1 (de) | 2004-04-14 | 2005-11-03 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | Neue Alkin-Verbindungen mit MCH-antagonistischer Wirkung und diese Verbindungen enthaltende Arzneimittel |
DE102004017933A1 (de) | 2004-04-14 | 2005-11-03 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | Neue Alkin-Verbindungen mit MCH-antagonistischer Wirkung und diese Verbindungen enthaltende Arzneimittel |
DE102004017935A1 (de) | 2004-04-14 | 2005-11-03 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | Neue Alkin-Verbindungen mit MCH-antagonistischer Wirkung und diese Verbindungen enthaltende Arzneimittel |
DE102004017934A1 (de) | 2004-04-14 | 2005-11-03 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | Neue Alkin-Verbindungen mit MCH-antagonistischer Wirkung und diese Verbindungen enthaltende Arzneimittel |
DE102004017932A1 (de) | 2004-04-14 | 2005-11-03 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | Neue Alkin-Verbindungen mit MCH-antagonistischer Wirkung und diese Verbindungen enthaltende Arzneimittel |
JPWO2007018248A1 (ja) | 2005-08-10 | 2009-02-19 | 萬有製薬株式会社 | ピリドン化合物 |
US7875633B2 (en) | 2005-08-24 | 2011-01-25 | Banyu Pharmaceutical Co., Ltd. | Phenylpyridone derivative |
JPWO2007029847A1 (ja) | 2005-09-07 | 2009-03-19 | 萬有製薬株式会社 | 二環性芳香族置換ピリドン誘導体 |
BRPI0617891A2 (pt) | 2005-10-26 | 2011-08-09 | Boehringer Ingelheim Int | compostos de (hetero)arila com atividade antagonista de mch, sais fisiologicamente aceitáveis dos mesmos, composição, composição farmacêutica bem como uso e preparação dos ditos compostos |
-
2007
- 2007-08-20 AU AU2007287601A patent/AU2007287601B2/en not_active Ceased
- 2007-08-20 EP EP11168245A patent/EP2383259A1/en not_active Withdrawn
- 2007-08-20 CA CA002657183A patent/CA2657183A1/en not_active Abandoned
- 2007-08-20 RU RU2009110446/04A patent/RU2453543C2/ru not_active IP Right Cessation
- 2007-08-20 BR BRPI0716579-0A2A patent/BRPI0716579A2/pt not_active IP Right Cessation
- 2007-08-20 CN CNA2007800316731A patent/CN101506195A/zh active Pending
- 2007-08-20 NZ NZ575520A patent/NZ575520A/en not_active IP Right Cessation
- 2007-08-20 MX MX2009000334A patent/MX2009000334A/es active IP Right Grant
- 2007-08-20 EP EP07819958.5A patent/EP2069327B1/en active Active
- 2007-08-20 JP JP2009525040A patent/JP5073746B2/ja active Active
- 2007-08-20 KR KR1020097006150A patent/KR20090047542A/ko not_active Application Discontinuation
- 2007-08-20 WO PCT/EP2007/058601 patent/WO2008022979A1/en active Application Filing
- 2007-08-24 TW TW096131555A patent/TW200817366A/zh unknown
- 2007-08-24 AR ARP070103758A patent/AR062510A1/es not_active Application Discontinuation
- 2007-08-24 US US11/844,842 patent/US8067590B2/en active Active
- 2007-08-24 CL CL2007002491A patent/CL2007002491A1/es unknown
-
2008
- 2008-12-09 ZA ZA200810404A patent/ZA200810404B/xx unknown
-
2009
- 2009-02-19 IL IL197128A patent/IL197128A/en not_active IP Right Cessation
-
2011
- 2011-09-22 US US13/239,537 patent/US20120010185A1/en not_active Abandoned
Also Published As
Publication number | Publication date |
---|---|
ZA200810404B (en) | 2009-10-28 |
CA2657183A1 (en) | 2008-02-28 |
EP2069327B1 (en) | 2013-10-16 |
MX2009000334A (es) | 2009-01-28 |
CN101506195A (zh) | 2009-08-12 |
NZ575520A (en) | 2012-03-30 |
EP2069327A1 (en) | 2009-06-17 |
BRPI0716579A2 (pt) | 2013-10-08 |
JP2010501518A (ja) | 2010-01-21 |
TW200817366A (en) | 2008-04-16 |
RU2009110446A (ru) | 2010-09-27 |
US8067590B2 (en) | 2011-11-29 |
AU2007287601A1 (en) | 2008-02-28 |
WO2008022979A1 (en) | 2008-02-28 |
JP5073746B2 (ja) | 2012-11-14 |
US20080255083A1 (en) | 2008-10-16 |
KR20090047542A (ko) | 2009-05-12 |
RU2453543C2 (ru) | 2012-06-20 |
IL197128A0 (en) | 2009-11-18 |
US20120010185A1 (en) | 2012-01-12 |
AR062510A1 (es) | 2008-11-12 |
EP2383259A1 (en) | 2011-11-02 |
IL197128A (en) | 2013-04-30 |
AU2007287601B2 (en) | 2012-12-20 |
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