CH637644A5 - 3-(Alkoxycarbonyl)benzodiazepine derivatives, process for their preparation and their application in therapeutics - Google Patents

3-(Alkoxycarbonyl)benzodiazepine derivatives, process for their preparation and their application in therapeutics Download PDF

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Publication number
CH637644A5
CH637644A5 CH18779A CH18779A CH637644A5 CH 637644 A5 CH637644 A5 CH 637644A5 CH 18779 A CH18779 A CH 18779A CH 18779 A CH18779 A CH 18779A CH 637644 A5 CH637644 A5 CH 637644A5
Authority
CH
Switzerland
Prior art keywords
formula
product
action
preparation
hydrogen atom
Prior art date
Application number
CH18779A
Other languages
English (en)
French (fr)
Inventor
Henri Demarne
Jean-Charles Molimard
Original Assignee
Sanofi Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sanofi Sa filed Critical Sanofi Sa
Publication of CH637644A5 publication Critical patent/CH637644A5/fr

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D243/00—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
    • C07D243/06—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
    • C07D243/10—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D243/14—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines
    • C07D243/16—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals
    • C07D243/18—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals substituted in position 2 by nitrogen, oxygen or sulfur atoms
    • C07D243/24—Oxygen atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Biomedical Technology (AREA)
  • Public Health (AREA)
  • Anesthesiology (AREA)
  • Pain & Pain Management (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
CH18779A 1978-01-10 1979-01-09 3-(Alkoxycarbonyl)benzodiazepine derivatives, process for their preparation and their application in therapeutics CH637644A5 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB95078 1978-01-10

Publications (1)

Publication Number Publication Date
CH637644A5 true CH637644A5 (en) 1983-08-15

Family

ID=9713371

Family Applications (1)

Application Number Title Priority Date Filing Date
CH18779A CH637644A5 (en) 1978-01-10 1979-01-09 3-(Alkoxycarbonyl)benzodiazepine derivatives, process for their preparation and their application in therapeutics

Country Status (8)

Country Link
JP (1) JPS54151992A (US20080094685A1-20080424-C00004.png)
BE (1) BE877567A (US20080094685A1-20080424-C00004.png)
CA (1) CA1126730A (US20080094685A1-20080424-C00004.png)
CH (1) CH637644A5 (US20080094685A1-20080424-C00004.png)
DE (1) DE2900017A1 (US20080094685A1-20080424-C00004.png)
FR (1) FR2414043A1 (US20080094685A1-20080424-C00004.png)
IT (1) IT1118271B (US20080094685A1-20080424-C00004.png)
NL (1) NL7900192A (US20080094685A1-20080424-C00004.png)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9911152D0 (en) * 1999-05-14 1999-07-14 Glaxo Group Ltd Short-acting benzodiazepines
US7160880B1 (en) 1999-05-14 2007-01-09 Cenes Limited Short-acting benzodiazepines
ATE480532T1 (de) 2006-07-10 2010-09-15 Paion Uk Ltd Benzodiazepinsalze mit kurzzeitwirkung und polymorphe formen davon
EP2450039A1 (en) 2010-11-08 2012-05-09 PAION UK Ltd. Dosing regimen for sedation with CNS 7056 (Remimazolam)
AR094963A1 (es) 2013-03-04 2015-09-09 Ono Pharmaceutical Co Reacción de oxidación excelente en el índice de conversión

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3678043A (en) * 1966-03-14 1972-07-18 American Home Prod 2,3-dihydro-2-oxo-1h-1,4-benzodiazepine-3-carboxylic acid esters and related compounds
CH500997A (de) * 1967-08-09 1970-12-31 Hoffmann La Roche Verfahren zur Herstellung von Benzodiazepin-Derivaten
GB1538164A (en) * 1976-05-05 1979-01-10 Clin Midy Benzodiazepine derivatives

Also Published As

Publication number Publication date
FR2414043A1 (fr) 1979-08-03
NL7900192A (nl) 1979-07-12
DE2900017A1 (de) 1979-07-12
CA1126730A (fr) 1982-06-29
FR2414043B1 (US20080094685A1-20080424-C00004.png) 1982-03-26
IT1118271B (it) 1986-02-24
JPS54151992A (en) 1979-11-29
IT7967037A0 (it) 1979-01-09
BE877567A (fr) 1979-11-05

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PL Patent ceased