CA3247129A1 - SERPINE PEPTIDES AND THEIR METHODS OF USE - Google Patents

SERPINE PEPTIDES AND THEIR METHODS OF USE

Info

Publication number
CA3247129A1
CA3247129A1 CA3247129A CA3247129A CA3247129A1 CA 3247129 A1 CA3247129 A1 CA 3247129A1 CA 3247129 A CA3247129 A CA 3247129A CA 3247129 A CA3247129 A CA 3247129A CA 3247129 A1 CA3247129 A1 CA 3247129A1
Authority
CA
Canada
Prior art keywords
seq
peptide
serpin
disease
serpin peptide
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
CA3247129A
Other languages
English (en)
French (fr)
Inventor
Dana AUSTIN
Cohava Gelber
Original Assignee
SERPIN PHARMA LLC
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by SERPIN PHARMA LLC filed Critical SERPIN PHARMA LLC
Publication of CA3247129A1 publication Critical patent/CA3247129A1/en
Pending legal-status Critical Current

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • A61K38/16Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • A61K38/55Protease inhibitors
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K14/00Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • C07K14/81Protease inhibitors
    • C07K14/8107Endopeptidase (E.C. 3.4.21-99) inhibitors
    • C07K14/811Serine protease (E.C. 3.4.21) inhibitors
    • C07K14/8121Serpins

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Immunology (AREA)
  • Epidemiology (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Medicinal Preparation (AREA)
CA3247129A 2022-01-05 2022-12-30 SERPINE PEPTIDES AND THEIR METHODS OF USE Pending CA3247129A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US202263266444P 2022-01-05 2022-01-05
US63/266,444 2022-01-05
PCT/US2022/082669 WO2023133078A2 (en) 2022-01-05 2022-12-30 Serpin peptides and methods of using the same

Publications (1)

Publication Number Publication Date
CA3247129A1 true CA3247129A1 (en) 2023-07-13

Family

ID=87074167

Family Applications (1)

Application Number Title Priority Date Filing Date
CA3247129A Pending CA3247129A1 (en) 2022-01-05 2022-12-30 SERPINE PEPTIDES AND THEIR METHODS OF USE

Country Status (8)

Country Link
US (2) US20250161419A1 (https=)
EP (1) EP4460322A4 (https=)
JP (1) JP2025503607A (https=)
CN (1) CN118804758A (https=)
AU (1) AU2022431253A1 (https=)
CA (1) CA3247129A1 (https=)
IL (1) IL314135A (https=)
WO (1) WO2023133078A2 (https=)

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2017040287A1 (en) * 2015-08-28 2017-03-09 Serpin Pharma, Llc Methods for treatment of diseases
WO2017123401A1 (en) * 2016-01-13 2017-07-20 Children's Hospital Medical Center Compositions and methods for treating allergic inflammatory conditions
EP3773727A4 (en) * 2018-04-09 2022-05-04 Yale University BIFUNCTIONAL SMALL MOLECULES TO TARGETING THE SELECTIVE DEGRADATION OF CIRCULATING PROTEINS
KR20220099963A (ko) * 2019-10-10 2022-07-14 예일 유니버시티 세포 수용체를 통한 분자 분해제로서의 조작된 항체
US20210162029A1 (en) * 2019-11-04 2021-06-03 Azitra Inc Compositions and methods for treatment or prevention of skin diseases and disorders with lekti
EP4003391A4 (en) * 2020-07-06 2023-02-22 Serpin Pharma, LLC PEPTIDES AND METHODS OF USE THEREOF
AU2022222778A1 (en) * 2021-02-22 2023-08-31 Yale University Targeted bifunctional degraders and methods using same

Also Published As

Publication number Publication date
US20230406906A1 (en) 2023-12-21
AU2022431253A1 (en) 2024-07-25
WO2023133078A2 (en) 2023-07-13
EP4460322A2 (en) 2024-11-13
US20250161419A1 (en) 2025-05-22
IL314135A (en) 2024-09-01
JP2025503607A (ja) 2025-02-04
CN118804758A (zh) 2024-10-18
EP4460322A4 (en) 2026-02-25
WO2023133078A3 (en) 2023-08-17

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