CA3229079A1 - Flow through cation exchange chromatography purification processes for antibody drug conjugates - Google Patents

Flow through cation exchange chromatography purification processes for antibody drug conjugates Download PDF

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Publication number
CA3229079A1
CA3229079A1 CA3229079A CA3229079A CA3229079A1 CA 3229079 A1 CA3229079 A1 CA 3229079A1 CA 3229079 A CA3229079 A CA 3229079A CA 3229079 A CA3229079 A CA 3229079A CA 3229079 A1 CA3229079 A1 CA 3229079A1
Authority
CA
Canada
Prior art keywords
adc
purification
antibody
cys
purified
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
CA3229079A
Other languages
English (en)
French (fr)
Inventor
Rachel HENDRICKS
Matthew Henry HUTCHINSON
Mark Frederick FEDESCO
Benjamin Phu TRAN
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Genentech Inc
Original Assignee
Genentech Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Genentech Inc filed Critical Genentech Inc
Publication of CA3229079A1 publication Critical patent/CA3229079A1/en
Pending legal-status Critical Current

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Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/50Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates
    • A61K47/51Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent
    • A61K47/68Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent the modifying agent being an antibody, an immunoglobulin or a fragment thereof, e.g. an Fc-fragment
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K1/00General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length
    • C07K1/107General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length by chemical modification of precursor peptides
    • C07K1/1072General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length by chemical modification of precursor peptides by covalent attachment of residues or functional groups
    • C07K1/1077General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length by chemical modification of precursor peptides by covalent attachment of residues or functional groups by covalent attachment of residues other than amino acids or peptide residues, e.g. sugars, polyols, fatty acids
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K1/00General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length
    • C07K1/14Extraction; Separation; Purification
    • C07K1/16Extraction; Separation; Purification by chromatography
    • C07K1/18Ion-exchange chromatography

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Genetics & Genomics (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Biochemistry (AREA)
  • Analytical Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Immunology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Peptides Or Proteins (AREA)
CA3229079A 2021-08-23 2022-08-22 Flow through cation exchange chromatography purification processes for antibody drug conjugates Pending CA3229079A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US202163236170P 2021-08-23 2021-08-23
US63/236,170 2021-08-23
PCT/US2022/075252 WO2023028446A1 (en) 2021-08-23 2022-08-22 Flow through cation exchange chromatography purification processes for antibody drug conjugates

Publications (1)

Publication Number Publication Date
CA3229079A1 true CA3229079A1 (en) 2023-03-02

Family

ID=83271094

Family Applications (1)

Application Number Title Priority Date Filing Date
CA3229079A Pending CA3229079A1 (en) 2021-08-23 2022-08-22 Flow through cation exchange chromatography purification processes for antibody drug conjugates

Country Status (12)

Country Link
US (1) US20240277859A1 (enExample)
EP (1) EP4392433A1 (enExample)
JP (1) JP2024532238A (enExample)
KR (1) KR20240046733A (enExample)
CN (1) CN117881686A (enExample)
AR (1) AR126847A1 (enExample)
AU (1) AU2022332274A1 (enExample)
CA (1) CA3229079A1 (enExample)
IL (1) IL310556A (enExample)
MX (1) MX2024002133A (enExample)
TW (1) TW202323268A (enExample)
WO (1) WO2023028446A1 (enExample)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN118290513B (zh) * 2024-06-05 2025-03-14 东曜药业有限公司 一种去除抗体偶联药物中游离小分子的阴离子柱层析方法及抗体偶联药物

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DK1869065T3 (da) 2005-03-11 2020-06-08 Wyeth Llc Fremgangsmåde til kromatografi med svag opdeling
WO2012059308A1 (en) * 2010-11-01 2012-05-10 Dsm Ip Assets B.V. Single unit ion exchange chromatography antibody purification
SG10201701224UA (en) 2012-03-12 2017-04-27 Merck Patent Gmbh Removal of protein aggregates from biopharmaceutical preparations in a flowthrough mode
CN104208719B (zh) * 2014-09-24 2017-05-03 北京天广实生物技术股份有限公司 一种抗体偶联药物的阳离子交换层析纯化方法
US20180311375A1 (en) * 2017-04-27 2018-11-01 Cadila Healthcare Limited Process of preparing antibody-drug conjugate

Also Published As

Publication number Publication date
AU2022332274A1 (en) 2024-02-15
MX2024002133A (es) 2024-03-06
EP4392433A1 (en) 2024-07-03
IL310556A (en) 2024-03-01
AR126847A1 (es) 2023-11-22
US20240277859A1 (en) 2024-08-22
KR20240046733A (ko) 2024-04-09
TW202323268A (zh) 2023-06-16
CN117881686A (zh) 2024-04-12
WO2023028446A1 (en) 2023-03-02
JP2024532238A (ja) 2024-09-05

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