CA3001903A1 - Therapeutic targeting of casein kinase 1.delta. in breast cancer - Google Patents
Therapeutic targeting of casein kinase 1.delta. in breast cancer Download PDFInfo
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- CA3001903A1 CA3001903A1 CA3001903A CA3001903A CA3001903A1 CA 3001903 A1 CA3001903 A1 CA 3001903A1 CA 3001903 A CA3001903 A CA 3001903A CA 3001903 A CA3001903 A CA 3001903A CA 3001903 A1 CA3001903 A1 CA 3001903A1
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- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
- A61K31/5375—1,4-Oxazines, e.g. morpholine
- A61K31/5377—1,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
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- C—CHEMISTRY; METALLURGY
- C12—BIOCHEMISTRY; BEER; SPIRITS; WINE; VINEGAR; MICROBIOLOGY; ENZYMOLOGY; MUTATION OR GENETIC ENGINEERING
- C12Q—MEASURING OR TESTING PROCESSES INVOLVING ENZYMES, NUCLEIC ACIDS OR MICROORGANISMS; COMPOSITIONS OR TEST PAPERS THEREFOR; PROCESSES OF PREPARING SUCH COMPOSITIONS; CONDITION-RESPONSIVE CONTROL IN MICROBIOLOGICAL OR ENZYMOLOGICAL PROCESSES
- C12Q1/00—Measuring or testing processes involving enzymes, nucleic acids or microorganisms; Compositions therefor; Processes of preparing such compositions
- C12Q1/68—Measuring or testing processes involving enzymes, nucleic acids or microorganisms; Compositions therefor; Processes of preparing such compositions involving nucleic acids
- C12Q1/6876—Nucleic acid products used in the analysis of nucleic acids, e.g. primers or probes
- C12Q1/6883—Nucleic acid products used in the analysis of nucleic acids, e.g. primers or probes for diseases caused by alterations of genetic material
- C12Q1/6886—Nucleic acid products used in the analysis of nucleic acids, e.g. primers or probes for diseases caused by alterations of genetic material for cancer
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- C—CHEMISTRY; METALLURGY
- C12—BIOCHEMISTRY; BEER; SPIRITS; WINE; VINEGAR; MICROBIOLOGY; ENZYMOLOGY; MUTATION OR GENETIC ENGINEERING
- C12Q—MEASURING OR TESTING PROCESSES INVOLVING ENZYMES, NUCLEIC ACIDS OR MICROORGANISMS; COMPOSITIONS OR TEST PAPERS THEREFOR; PROCESSES OF PREPARING SUCH COMPOSITIONS; CONDITION-RESPONSIVE CONTROL IN MICROBIOLOGICAL OR ENZYMOLOGICAL PROCESSES
- C12Q2600/00—Oligonucleotides characterized by their use
- C12Q2600/136—Screening for pharmacological compounds
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- Life Sciences & Earth Sciences (AREA)
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Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201562240689P | 2015-10-13 | 2015-10-13 | |
| US62/240,689 | 2015-10-13 | ||
| PCT/US2016/055436 WO2017066055A1 (en) | 2015-10-13 | 2016-10-05 | THERAPEUTIC TARGETING OF CASEIN KINASE 1δ IN BREAST CANCER |
Publications (1)
| Publication Number | Publication Date |
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| CA3001903A1 true CA3001903A1 (en) | 2017-04-20 |
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| CA3001903A Abandoned CA3001903A1 (en) | 2015-10-13 | 2016-10-05 | Therapeutic targeting of casein kinase 1.delta. in breast cancer |
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| US (2) | US10603322B2 (enExample) |
| EP (1) | EP3362452A4 (enExample) |
| JP (1) | JP2018538241A (enExample) |
| CN (1) | CN108431006A (enExample) |
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| CA (1) | CA3001903A1 (enExample) |
| HK (1) | HK1259409A1 (enExample) |
| WO (1) | WO2017066055A1 (enExample) |
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| US20200078387A1 (en) * | 2016-12-16 | 2020-03-12 | The Johns Hopkins University | Chemical inhibitors against kinases to block telomere elongation in cancer |
| WO2019145386A1 (en) | 2018-01-26 | 2019-08-01 | Roche Innovation Center Copenhagen A/S | Oligonucleotides for modulating csnk1d expression |
| US11666578B2 (en) | 2018-05-08 | 2023-06-06 | The University Of Florida Research Foundation, Inc. | Small molecule inhibitors of CDK12/CDK13 |
| AU2019325593A1 (en) * | 2018-08-22 | 2021-03-18 | Merck Patent Gmbh | Treatment of triple negative breast cancer with targeted TGF-B inhibition |
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| US9493464B2 (en) * | 2012-02-29 | 2016-11-15 | The Scripps Research Institute | Wee1 degradation inhibitors |
| ES2638179T3 (es) * | 2013-01-16 | 2017-10-19 | Signal Pharmaceuticals, Llc | Compuestos de pirrolopirimidina sustituidos, composiciones de los mismos, y métodos de tratamiento con los mismos |
-
2016
- 2016-10-05 EP EP16855974.8A patent/EP3362452A4/en not_active Withdrawn
- 2016-10-05 US US15/768,257 patent/US10603322B2/en not_active Expired - Fee Related
- 2016-10-05 AU AU2016338639A patent/AU2016338639A1/en not_active Abandoned
- 2016-10-05 CN CN201680071705.XA patent/CN108431006A/zh active Pending
- 2016-10-05 CA CA3001903A patent/CA3001903A1/en not_active Abandoned
- 2016-10-05 WO PCT/US2016/055436 patent/WO2017066055A1/en not_active Ceased
- 2016-10-05 HK HK19101778.5A patent/HK1259409A1/zh unknown
- 2016-10-05 JP JP2018519027A patent/JP2018538241A/ja active Pending
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2019
- 2019-11-25 US US16/694,380 patent/US20200163972A1/en not_active Abandoned
Also Published As
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|---|---|
| CN108431006A (zh) | 2018-08-21 |
| EP3362452A4 (en) | 2019-06-12 |
| EP3362452A1 (en) | 2018-08-22 |
| JP2018538241A (ja) | 2018-12-27 |
| AU2016338639A1 (en) | 2018-05-10 |
| WO2017066055A1 (en) | 2017-04-20 |
| US10603322B2 (en) | 2020-03-31 |
| US20200163972A1 (en) | 2020-05-28 |
| HK1259409A1 (zh) | 2019-11-29 |
| US20180311252A1 (en) | 2018-11-01 |
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