CA2961009A1 - Systems and methods for attenuating opioid-induced euphoria - Google Patents
Systems and methods for attenuating opioid-induced euphoria Download PDFInfo
- Publication number
- CA2961009A1 CA2961009A1 CA2961009A CA2961009A CA2961009A1 CA 2961009 A1 CA2961009 A1 CA 2961009A1 CA 2961009 A CA2961009 A CA 2961009A CA 2961009 A CA2961009 A CA 2961009A CA 2961009 A1 CA2961009 A1 CA 2961009A1
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- CA
- Canada
- Prior art keywords
- buprenorphine
- opioid
- administered
- mcg
- amount
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
Links
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Classifications
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- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
- A61K31/485—Morphinan derivatives, e.g. morphine, codeine
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/13—Amines
- A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
- A61K31/137—Arylalkylamines, e.g. amphetamine, epinephrine, salbutamol, ephedrine or methadone
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- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
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- A—HUMAN NECESSITIES
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- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
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- A61P25/36—Opioid-abuse
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
- A61K9/006—Oral mucosa, e.g. mucoadhesive forms, sublingual droplets; Buccal patches or films; Buccal sprays
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
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- Nutrition Science (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (5)
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| US201462049989P | 2014-09-12 | 2014-09-12 | |
| US62/049,989 | 2014-09-12 | ||
| US201462065393P | 2014-10-17 | 2014-10-17 | |
| US62/065,393 | 2014-10-17 | ||
| PCT/US2015/049948 WO2016040934A1 (en) | 2014-09-12 | 2015-09-14 | Systems and methods for attenuating opioid-induced euphoria |
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| CA2961009A1 true CA2961009A1 (en) | 2016-03-17 |
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| CA2961009A Abandoned CA2961009A1 (en) | 2014-09-12 | 2015-09-14 | Systems and methods for attenuating opioid-induced euphoria |
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| CN (1) | CN107072204A (enExample) |
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| TW (1) | TW201613590A (enExample) |
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| WO2018125716A1 (en) | 2017-01-02 | 2018-07-05 | Purdue Pharma L.P. | Morphinan derivatives and use thereof |
| CA3068036A1 (en) * | 2017-06-30 | 2019-01-03 | Purdue Pharma L.P. | Use to buprenorphine in combination with an opioid to treat pain |
| AU2018351502B2 (en) * | 2017-10-20 | 2024-09-05 | Purdue Pharma L.P. | Pharmaceutical dosage forms |
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| EP1613266A4 (en) * | 2003-04-15 | 2009-05-06 | Theraquest Biosciences Llc | METHOD FOR TREATING PAIN AND COMPOSITIONS FOR USE THEREOF |
| EP1813276A1 (en) * | 2006-01-27 | 2007-08-01 | Euro-Celtique S.A. | Tamper resistant dosage forms |
| US20090246265A1 (en) * | 2008-03-26 | 2009-10-01 | Alltranz Inc. | Abuse deterrent transdermal formulations of opiate agonists and agonist-antagonists |
| WO2011109743A2 (en) * | 2010-03-04 | 2011-09-09 | Rand Jerry N | Synergistic effects of combinations of buprenorphine and opioids for the treatment of pain |
| CA2817071C (en) * | 2010-11-08 | 2018-04-24 | Omeros Corporation | Treatment of addiction and impulse-control disorders using pde7 inhibitors |
| HK1206978A1 (en) * | 2012-04-17 | 2016-01-22 | Purdue Pharma L.P. | Systems and methods for treating an opioid-induced adverse pharmacodynamic response |
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2015
- 2015-09-11 TW TW104130183A patent/TW201613590A/zh unknown
- 2015-09-14 JP JP2017513760A patent/JP2017526719A/ja active Pending
- 2015-09-14 KR KR1020177009493A patent/KR20170052644A/ko not_active Withdrawn
- 2015-09-14 EP EP15840440.0A patent/EP3190890A4/en not_active Withdrawn
- 2015-09-14 CA CA2961009A patent/CA2961009A1/en not_active Abandoned
- 2015-09-14 WO PCT/US2015/049948 patent/WO2016040934A1/en not_active Ceased
- 2015-09-14 US US14/853,151 patent/US20160074387A1/en not_active Abandoned
- 2015-09-14 AU AU2015314714A patent/AU2015314714A1/en not_active Abandoned
- 2015-09-14 MA MA040333A patent/MA40333A/fr unknown
- 2015-09-14 CN CN201580055965.3A patent/CN107072204A/zh active Pending
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2017
- 2017-03-09 IL IL251049A patent/IL251049A0/en unknown
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2020
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Also Published As
| Publication number | Publication date |
|---|---|
| WO2016040934A1 (en) | 2016-03-17 |
| JP2017526719A (ja) | 2017-09-14 |
| IL251049A0 (en) | 2017-04-30 |
| MA40333A (fr) | 2016-03-17 |
| AU2015314714A1 (en) | 2017-03-09 |
| KR20170052644A (ko) | 2017-05-12 |
| EP3190890A4 (en) | 2018-04-25 |
| EP3190890A1 (en) | 2017-07-19 |
| US20200276187A1 (en) | 2020-09-03 |
| US20160074387A1 (en) | 2016-03-17 |
| CN107072204A (zh) | 2017-08-18 |
| TW201613590A (en) | 2016-04-16 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| US20240350479A1 (en) | Systems and Methods for Treating an Opioid-Induced Adverse Pharmacodynamic Response | |
| US20200276187A1 (en) | Systems and methods for attenuating opioid-induced euphoria | |
| US10226457B2 (en) | Systems and methods for treating an opioid-induced adverse pharmacodynamic response |
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| FZDE | Discontinued |
Effective date: 20211207 |