CA2903276A1 - Muscarinic agonists - Google Patents
Muscarinic agonists Download PDFInfo
- Publication number
- CA2903276A1 CA2903276A1 CA2903276A CA2903276A CA2903276A1 CA 2903276 A1 CA2903276 A1 CA 2903276A1 CA 2903276 A CA2903276 A CA 2903276A CA 2903276 A CA2903276 A CA 2903276A CA 2903276 A1 CA2903276 A1 CA 2903276A1
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Classifications
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- C07D451/00—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof
- C07D451/02—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof
- C07D451/04—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof with hetero atoms directly attached in position 3 of the 8-azabicyclo [3.2.1] octane or in position 7 of the 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring system
- C07D451/06—Oxygen atoms
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Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201361790364P | 2013-03-15 | 2013-03-15 | |
| US61/790,364 | 2013-03-15 | ||
| PCT/US2014/026998 WO2014152144A1 (en) | 2013-03-15 | 2014-03-14 | Muscarinic agonists |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CA2903276A1 true CA2903276A1 (en) | 2014-09-25 |
Family
ID=50439523
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CA2903276A Abandoned CA2903276A1 (en) | 2013-03-15 | 2014-03-14 | Muscarinic agonists |
Country Status (13)
| Country | Link |
|---|---|
| US (1) | US9670209B2 (enExample) |
| EP (1) | EP2976079A1 (enExample) |
| JP (1) | JP2016513677A (enExample) |
| KR (1) | KR20150143439A (enExample) |
| CN (1) | CN105120865A (enExample) |
| AU (1) | AU2014240139A1 (enExample) |
| BR (1) | BR112015021271A2 (enExample) |
| CA (1) | CA2903276A1 (enExample) |
| IL (1) | IL241001A0 (enExample) |
| MX (1) | MX2015012043A (enExample) |
| RU (1) | RU2015144155A (enExample) |
| TW (1) | TW201446761A (enExample) |
| WO (1) | WO2014152144A1 (enExample) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US9670209B2 (en) | 2013-03-15 | 2017-06-06 | Acadia Pharmaceuticals Inc. | Muscarinic agonists |
| KR101613245B1 (ko) | 2015-04-27 | 2016-04-18 | 주식회사 대웅제약 | 신규의 4-메톡시 피롤 유도체 또는 이의 염 및 이를 포함하는 약학 조성물 |
| US9822122B2 (en) | 2016-03-31 | 2017-11-21 | Oncternal Therapeutics, Inc. | Indoline analogs and uses thereof |
Family Cites Families (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5707798A (en) | 1993-07-13 | 1998-01-13 | Novo Nordisk A/S | Identification of ligands by selective amplification of cells transfected with receptors |
| JPH10152470A (ja) * | 1996-09-25 | 1998-06-09 | Yoshitomi Pharmaceut Ind Ltd | ピペラジン化合物 |
| EP1535912A1 (en) | 2000-04-28 | 2005-06-01 | Arcadia Pharmaceuticals Inc. | Muscarinic agonists |
| RU2269523C2 (ru) * | 2000-04-28 | 2006-02-10 | Акадиа Фармасьютикалз, Инк. | Мускариновые агонисты |
| US7550459B2 (en) * | 2001-12-28 | 2009-06-23 | Acadia Pharmaceuticals, Inc. | Tetrahydroquinoline analogues as muscarinic agonists |
| BRPI0409523A (pt) * | 2003-03-28 | 2006-04-18 | Acadia Pharm Inc | método para o tratamento da dor neuropática, método de identificação de um composto e composição farmacêutica |
| US7931909B2 (en) | 2005-05-10 | 2011-04-26 | Allergan, Inc. | Ocular therapy using alpha-2 adrenergic receptor compounds having enhanced anterior clearance rates |
| US9670209B2 (en) | 2013-03-15 | 2017-06-06 | Acadia Pharmaceuticals Inc. | Muscarinic agonists |
-
2014
- 2014-03-14 US US14/774,685 patent/US9670209B2/en not_active Expired - Fee Related
- 2014-03-14 EP EP14715518.8A patent/EP2976079A1/en not_active Withdrawn
- 2014-03-14 JP JP2016502306A patent/JP2016513677A/ja active Pending
- 2014-03-14 CA CA2903276A patent/CA2903276A1/en not_active Abandoned
- 2014-03-14 WO PCT/US2014/026998 patent/WO2014152144A1/en not_active Ceased
- 2014-03-14 MX MX2015012043A patent/MX2015012043A/es unknown
- 2014-03-14 RU RU2015144155A patent/RU2015144155A/ru not_active Application Discontinuation
- 2014-03-14 TW TW103109294A patent/TW201446761A/zh unknown
- 2014-03-14 AU AU2014240139A patent/AU2014240139A1/en not_active Abandoned
- 2014-03-14 BR BR112015021271A patent/BR112015021271A2/pt not_active IP Right Cessation
- 2014-03-14 CN CN201480015640.8A patent/CN105120865A/zh active Pending
- 2014-03-14 KR KR1020157025205A patent/KR20150143439A/ko not_active Withdrawn
-
2015
- 2015-09-01 IL IL241001A patent/IL241001A0/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| US9670209B2 (en) | 2017-06-06 |
| KR20150143439A (ko) | 2015-12-23 |
| WO2014152144A1 (en) | 2014-09-25 |
| TW201446761A (zh) | 2014-12-16 |
| EP2976079A1 (en) | 2016-01-27 |
| BR112015021271A2 (pt) | 2017-08-22 |
| JP2016513677A (ja) | 2016-05-16 |
| US20160039819A1 (en) | 2016-02-11 |
| AU2014240139A1 (en) | 2015-09-17 |
| CN105120865A (zh) | 2015-12-02 |
| MX2015012043A (es) | 2016-03-17 |
| IL241001A0 (en) | 2015-11-30 |
| RU2015144155A (ru) | 2017-04-24 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FZDE | Discontinued |
Effective date: 20200831 |
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| FZDE | Discontinued |
Effective date: 20200831 |