CA2902599C - Pyrimido-diazepinone compounds and methods of treating disorders - Google Patents

Pyrimido-diazepinone compounds and methods of treating disorders Download PDF

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CA2902599C
CA2902599C CA2902599A CA2902599A CA2902599C CA 2902599 C CA2902599 C CA 2902599C CA 2902599 A CA2902599 A CA 2902599A CA 2902599 A CA2902599 A CA 2902599A CA 2902599 C CA2902599 C CA 2902599C
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compound
disease
cancer
kinase
alkyl
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French (fr)
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CA2902599A1 (en
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Nathanael S. Gray
David Waller
Hwan Guen Choi
Jinhua Wang
Xianming Deng
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Dana Farber Cancer Institute Inc
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Dana Farber Cancer Institute Inc
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    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
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CA2902599A 2013-03-15 2014-03-17 Pyrimido-diazepinone compounds and methods of treating disorders Active CA2902599C (en)

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US201361802075P 2013-03-15 2013-03-15
US61/802,075 2013-03-15
PCT/US2014/030760 WO2014145909A2 (en) 2013-03-15 2014-03-17 Pyrimido-diazepinone compounds and methods of treating disorders

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CA2902599A1 CA2902599A1 (en) 2014-09-18
CA2902599C true CA2902599C (en) 2023-03-21

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WO2014145909A2 (en) * 2013-03-15 2014-09-18 Dana-Farber Cancer Institute, Inc. Pyrimido-diazepinone compounds and methods of treating disorders
EP3189051A1 (en) * 2014-09-02 2017-07-12 Pierre Fabre Médicament Isoquinolinone derivatives useful in the treatment of cancer
CN104803914B (zh) * 2015-03-05 2017-11-14 成都理工大学 作为Rho激酶抑制剂的六氢氮杂卓氧基苯甲酰胺类化合物
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