CA2878009A1 - Single dose oral formulations and methods for treatment of cats with ectoparasiticidal spinosad - Google Patents
Single dose oral formulations and methods for treatment of cats with ectoparasiticidal spinosad Download PDFInfo
- Publication number
- CA2878009A1 CA2878009A1 CA2878009A CA2878009A CA2878009A1 CA 2878009 A1 CA2878009 A1 CA 2878009A1 CA 2878009 A CA2878009 A CA 2878009A CA 2878009 A CA2878009 A CA 2878009A CA 2878009 A1 CA2878009 A1 CA 2878009A1
- Authority
- CA
- Canada
- Prior art keywords
- spinosad
- formulation
- dose
- treatment
- cats
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
Links
- JFLRKDZMHNBDQS-UCQUSYKYSA-N CC[C@H]1CCC[C@@H]([C@H](C(=O)C2=C[C@H]3[C@@H]4C[C@@H](C[C@H]4C(=C[C@H]3[C@@H]2CC(=O)O1)C)O[C@H]5[C@@H]([C@@H]([C@H]([C@@H](O5)C)OC)OC)OC)C)O[C@H]6CC[C@@H]([C@H](O6)C)N(C)C.CC[C@H]1CCC[C@@H]([C@H](C(=O)C2=C[C@H]3[C@@H]4C[C@@H](C[C@H]4C=C[C@H]3C2CC(=O)O1)O[C@H]5[C@@H]([C@@H]([C@H]([C@@H](O5)C)OC)OC)OC)C)O[C@H]6CC[C@@H]([C@H](O6)C)N(C)C Chemical compound CC[C@H]1CCC[C@@H]([C@H](C(=O)C2=C[C@H]3[C@@H]4C[C@@H](C[C@H]4C(=C[C@H]3[C@@H]2CC(=O)O1)C)O[C@H]5[C@@H]([C@@H]([C@H]([C@@H](O5)C)OC)OC)OC)C)O[C@H]6CC[C@@H]([C@H](O6)C)N(C)C.CC[C@H]1CCC[C@@H]([C@H](C(=O)C2=C[C@H]3[C@@H]4C[C@@H](C[C@H]4C=C[C@H]3C2CC(=O)O1)O[C@H]5[C@@H]([C@@H]([C@H]([C@@H](O5)C)OC)OC)OC)C)O[C@H]6CC[C@@H]([C@H](O6)C)N(C)C JFLRKDZMHNBDQS-UCQUSYKYSA-N 0.000 title claims abstract description 118
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- 230000000694 effects Effects 0.000 description 7
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- ATJFFYVFTNAWJD-UHFFFAOYSA-N Tin Chemical compound [Sn] ATJFFYVFTNAWJD-UHFFFAOYSA-N 0.000 description 1
- VXSIXFKKSNGRRO-MXOVTSAMSA-N [(1s)-2-methyl-4-oxo-3-[(2z)-penta-2,4-dienyl]cyclopent-2-en-1-yl] (1r,3r)-2,2-dimethyl-3-(2-methylprop-1-enyl)cyclopropane-1-carboxylate;[(1s)-2-methyl-4-oxo-3-[(2z)-penta-2,4-dienyl]cyclopent-2-en-1-yl] (1r,3r)-3-[(e)-3-methoxy-2-methyl-3-oxoprop-1-enyl Chemical class CC1(C)[C@H](C=C(C)C)[C@H]1C(=O)O[C@@H]1C(C)=C(C\C=C/C=C)C(=O)C1.CC1(C)[C@H](/C=C(\C)C(=O)OC)[C@H]1C(=O)O[C@@H]1C(C)=C(C\C=C/C=C)C(=O)C1 VXSIXFKKSNGRRO-MXOVTSAMSA-N 0.000 description 1
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Classifications
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- A61K9/0056—Mouth soluble or dispersible forms; Suckable, eatable, chewable coherent forms; Forms rapidly disintegrating in the mouth; Lozenges; Lollipops; Bite capsules; Baked products; Baits or other oral forms for animals
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- A61K31/7042—Compounds having saccharide radicals and heterocyclic rings
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- A01N25/00—Biocides, pest repellants or attractants, or plant growth regulators, characterised by their forms, or by their non-active ingredients or by their methods of application, e.g. seed treatment or sequential application; Substances for reducing the noxious effect of the active ingredients to organisms other than pests
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- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/02—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one or more oxygen or sulfur atoms as the only ring hetero atoms
- A01N43/04—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one or more oxygen or sulfur atoms as the only ring hetero atoms with one hetero atom
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- A61P33/00—Antiparasitic agents
- A61P33/10—Anthelmintics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/14—Ectoparasiticides, e.g. scabicides
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N2300/00—Combinations or mixtures of active ingredients covered by classes A01N27/00 - A01N65/48 with other active or formulation relevant ingredients, e.g. specific carrier materials or surfactants, covered by classes A01N25/00 - A01N65/48
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Public Health (AREA)
- Epidemiology (AREA)
- Zoology (AREA)
- Polymers & Plastics (AREA)
- Engineering & Computer Science (AREA)
- Food Science & Technology (AREA)
- Animal Husbandry (AREA)
- Molecular Biology (AREA)
- Plant Pathology (AREA)
- Environmental Sciences (AREA)
- Agronomy & Crop Science (AREA)
- Pest Control & Pesticides (AREA)
- Dentistry (AREA)
- Wood Science & Technology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Chemistry (AREA)
- Physiology (AREA)
- Inorganic Chemistry (AREA)
- Nutrition Science (AREA)
- Tropical Medicine & Parasitology (AREA)
- Birds (AREA)
- Biophysics (AREA)
- Toxicology (AREA)
- Communicable Diseases (AREA)
- Oncology (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201261676023P | 2012-07-26 | 2012-07-26 | |
| US61/676,023 | 2012-07-26 | ||
| PCT/US2013/050987 WO2014018352A1 (en) | 2012-07-26 | 2013-07-18 | Single dose oral formulations and methods for treatment of cats with ectoparasiticidal spinosad |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CA2878009A1 true CA2878009A1 (en) | 2014-01-30 |
Family
ID=48877579
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CA2878009A Abandoned CA2878009A1 (en) | 2012-07-26 | 2013-07-18 | Single dose oral formulations and methods for treatment of cats with ectoparasiticidal spinosad |
Country Status (14)
| Country | Link |
|---|---|
| US (2) | US9220719B2 (enExample) |
| EP (1) | EP2877005A1 (enExample) |
| JP (1) | JP2015523388A (enExample) |
| KR (1) | KR20150023831A (enExample) |
| CN (1) | CN104703474A (enExample) |
| AR (1) | AR091769A1 (enExample) |
| AU (1) | AU2013293350B2 (enExample) |
| BR (1) | BR112015001152A2 (enExample) |
| CA (1) | CA2878009A1 (enExample) |
| EA (1) | EA201590097A1 (enExample) |
| IN (1) | IN2014MN02599A (enExample) |
| MX (1) | MX2015001137A (enExample) |
| TW (1) | TW201416077A (enExample) |
| WO (1) | WO2014018352A1 (enExample) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2018183512A1 (en) * | 2017-03-28 | 2018-10-04 | Piedmont Animal Health, Llc | Combinations of acaricides and insect growth regulators for control of fleas without emesis in animals |
| WO2020012406A1 (en) * | 2018-07-11 | 2020-01-16 | Jubilant Generics Limited | Veterinary dosage forms |
| CN118055703A (zh) * | 2021-06-25 | 2024-05-17 | 碗中动物健康公司 | 猫科动物口服饲料和在猫科动物中控制蚤侵袭的方法 |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2001011963A1 (en) * | 1999-08-12 | 2001-02-22 | Eli Lilly And Company | Oral treatment of companion animals with ectoparasiticidal spinosyns |
| KR100904941B1 (ko) * | 2001-03-21 | 2009-06-29 | 다우 아그로사이언시즈 엘엘씨 | 살충성 스피노신 유도체 |
| US20080311191A1 (en) * | 2004-08-27 | 2008-12-18 | Avinash Nangia | Multi-Layer Tablets and Bioadhesive Dosage Forms |
| US20070149464A1 (en) * | 2005-06-15 | 2007-06-28 | Pfizer Inc. | Combination |
| EP2248422A1 (en) * | 2009-05-08 | 2010-11-10 | Novartis AG | Ectoparasiticidal compositions |
| US20120003661A1 (en) | 2010-07-05 | 2012-01-05 | C3 Jian, Inc. | Methods and devices for the selective detection of microorganisms |
| CA2817001C (en) * | 2010-11-05 | 2015-09-29 | Eli Lilly And Company | Methods for inhibiting insect infestations |
-
2013
- 2013-07-15 AR ARP130102512 patent/AR091769A1/es unknown
- 2013-07-15 TW TW102125296A patent/TW201416077A/zh unknown
- 2013-07-18 KR KR1020157001565A patent/KR20150023831A/ko not_active Ceased
- 2013-07-18 BR BR112015001152A patent/BR112015001152A2/pt not_active IP Right Cessation
- 2013-07-18 US US13/944,904 patent/US9220719B2/en not_active Expired - Fee Related
- 2013-07-18 WO PCT/US2013/050987 patent/WO2014018352A1/en not_active Ceased
- 2013-07-18 AU AU2013293350A patent/AU2013293350B2/en not_active Ceased
- 2013-07-18 JP JP2015524327A patent/JP2015523388A/ja not_active Withdrawn
- 2013-07-18 CN CN201380039678.4A patent/CN104703474A/zh active Pending
- 2013-07-18 CA CA2878009A patent/CA2878009A1/en not_active Abandoned
- 2013-07-18 IN IN2599MUN2014 patent/IN2014MN02599A/en unknown
- 2013-07-18 EP EP13742365.3A patent/EP2877005A1/en not_active Withdrawn
- 2013-07-18 MX MX2015001137A patent/MX2015001137A/es unknown
- 2013-07-18 EA EA201590097A patent/EA201590097A1/ru unknown
-
2015
- 2015-12-18 US US14/974,961 patent/US20160101127A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| EP2877005A1 (en) | 2015-06-03 |
| AU2013293350A1 (en) | 2015-02-05 |
| AU2013293350B2 (en) | 2015-07-23 |
| BR112015001152A2 (pt) | 2017-06-27 |
| US20140031306A1 (en) | 2014-01-30 |
| JP2015523388A (ja) | 2015-08-13 |
| CN104703474A (zh) | 2015-06-10 |
| EA201590097A1 (ru) | 2015-06-30 |
| AR091769A1 (es) | 2015-02-25 |
| MX2015001137A (es) | 2015-10-14 |
| IN2014MN02599A (enExample) | 2015-07-24 |
| WO2014018352A1 (en) | 2014-01-30 |
| US20160101127A1 (en) | 2016-04-14 |
| TW201416077A (zh) | 2014-05-01 |
| KR20150023831A (ko) | 2015-03-05 |
| US9220719B2 (en) | 2015-12-29 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| EEER | Examination request |
Effective date: 20141223 |
|
| FZDE | Discontinued |
Effective date: 20180612 |