CA2819106C - Kat ii inhibitors - Google Patents
Kat ii inhibitors Download PDFInfo
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- CA2819106C CA2819106C CA2819106A CA2819106A CA2819106C CA 2819106 C CA2819106 C CA 2819106C CA 2819106 A CA2819106 A CA 2819106A CA 2819106 A CA2819106 A CA 2819106A CA 2819106 C CA2819106 C CA 2819106C
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- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/16—Otologicals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Veterinary Medicine (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Pain & Pain Management (AREA)
- Psychiatry (AREA)
- Cardiology (AREA)
- Hospice & Palliative Care (AREA)
- Heart & Thoracic Surgery (AREA)
- Urology & Nephrology (AREA)
- Psychology (AREA)
- Addiction (AREA)
- Oncology (AREA)
- Ophthalmology & Optometry (AREA)
- Immunology (AREA)
- Anesthesiology (AREA)
- Rheumatology (AREA)
- Communicable Diseases (AREA)
- Vascular Medicine (AREA)
- Otolaryngology (AREA)
- Gastroenterology & Hepatology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Physical Education & Sports Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Quinoline Compounds (AREA)
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US41879110P | 2010-12-01 | 2010-12-01 | |
| US61/418,791 | 2010-12-01 | ||
| US41923210P | 2010-12-02 | 2010-12-02 | |
| US61/419,232 | 2010-12-02 | ||
| PCT/IB2011/055190 WO2012073146A1 (en) | 2010-12-01 | 2011-11-18 | Kat ii inhibitors |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| CA2819106A1 CA2819106A1 (en) | 2012-06-07 |
| CA2819106C true CA2819106C (en) | 2015-12-29 |
Family
ID=45315857
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CA2819106A Expired - Fee Related CA2819106C (en) | 2010-12-01 | 2011-11-18 | Kat ii inhibitors |
Country Status (13)
| Country | Link |
|---|---|
| US (1) | US8487104B2 (OSRAM) |
| EP (1) | EP2646417A1 (OSRAM) |
| JP (1) | JP5868994B2 (OSRAM) |
| KR (1) | KR101522803B1 (OSRAM) |
| CN (1) | CN103228631B (OSRAM) |
| AR (1) | AR084051A1 (OSRAM) |
| AU (1) | AU2011336217B2 (OSRAM) |
| CA (1) | CA2819106C (OSRAM) |
| IL (1) | IL226668A (OSRAM) |
| MX (1) | MX2013005915A (OSRAM) |
| SG (1) | SG190246A1 (OSRAM) |
| WO (1) | WO2012073146A1 (OSRAM) |
| ZA (1) | ZA201303412B (OSRAM) |
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| SG11201407389QA (en) * | 2012-06-15 | 2015-02-27 | Pfizer | Tricyclic compounds as kat ii inhibitors |
| JP6440625B2 (ja) | 2012-11-14 | 2018-12-19 | ザ・ジョンズ・ホプキンス・ユニバーシティー | 精神分裂病を処置するための方法および組成物 |
| AU2015251207B2 (en) * | 2014-04-23 | 2019-08-22 | Mitsubishi Tanabe Pharma Corporation | Novel bicyclic or tricyclic heterocyclic compound |
| NZ738682A (en) | 2015-05-22 | 2022-01-28 | Agenebio Inc | Extended release pharmaceutical compositions of levetiracetam |
| US10793582B2 (en) | 2015-10-22 | 2020-10-06 | Mitsubishi Tanabe Pharma Corporation | Bicyclic heterocyclic compound |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE4208304A1 (de) * | 1992-03-16 | 1993-09-23 | Merck Patent Gmbh | 2-oxochinolinderivate |
| JPH0881443A (ja) * | 1994-09-12 | 1996-03-26 | Otsuka Pharmaceut Co Ltd | 細胞外マトリックス金属プロテアーゼ阻害剤 |
| US5594006A (en) * | 1993-03-18 | 1997-01-14 | Otsuka Pharmaceutical Co., Ltd. | Carbostyril derivatives as matrix metalloproteinases inhibitors |
| US7276608B2 (en) * | 2003-07-11 | 2007-10-02 | Bristol-Myers Squibb Company | Tetrahydroquinoline derivatives as cannabinoid receptor modulators |
| US20100273787A1 (en) * | 2007-11-15 | 2010-10-28 | Robert Schwarcz | Kynurenine-aminotransferase inhibitors |
| SG176288A1 (en) * | 2009-06-18 | 2012-01-30 | Pfizer | Bicyclic and tricyclic compounds as kat ii inhibitors |
| CA2819102A1 (en) | 2010-12-01 | 2012-06-07 | Pfizer Inc. | Kat ii inhibitors |
-
2011
- 2011-11-18 CN CN201180057792.0A patent/CN103228631B/zh not_active Expired - Fee Related
- 2011-11-18 JP JP2013541447A patent/JP5868994B2/ja not_active Expired - Fee Related
- 2011-11-18 WO PCT/IB2011/055190 patent/WO2012073146A1/en not_active Ceased
- 2011-11-18 SG SG2013036314A patent/SG190246A1/en unknown
- 2011-11-18 MX MX2013005915A patent/MX2013005915A/es not_active Application Discontinuation
- 2011-11-18 AU AU2011336217A patent/AU2011336217B2/en not_active Ceased
- 2011-11-18 EP EP11794240.9A patent/EP2646417A1/en not_active Withdrawn
- 2011-11-18 CA CA2819106A patent/CA2819106C/en not_active Expired - Fee Related
- 2011-11-18 KR KR1020137016959A patent/KR101522803B1/ko not_active Expired - Fee Related
- 2011-11-30 AR ARP110104458A patent/AR084051A1/es not_active Application Discontinuation
- 2011-11-30 US US13/307,140 patent/US8487104B2/en not_active Expired - Fee Related
-
2013
- 2013-05-10 ZA ZA2013/03412A patent/ZA201303412B/en unknown
- 2013-05-30 IL IL226668A patent/IL226668A/en not_active IP Right Cessation
Also Published As
| Publication number | Publication date |
|---|---|
| CA2819106A1 (en) | 2012-06-07 |
| MX2013005915A (es) | 2013-07-03 |
| IL226668A (en) | 2016-07-31 |
| US8487104B2 (en) | 2013-07-16 |
| AU2011336217B2 (en) | 2015-10-01 |
| JP2014500885A (ja) | 2014-01-16 |
| AR084051A1 (es) | 2013-04-17 |
| AU2011336217A1 (en) | 2013-06-06 |
| KR20130098421A (ko) | 2013-09-04 |
| HK1187611A1 (en) | 2014-04-11 |
| SG190246A1 (en) | 2013-06-28 |
| WO2012073146A1 (en) | 2012-06-07 |
| JP5868994B2 (ja) | 2016-02-24 |
| KR101522803B1 (ko) | 2015-05-26 |
| US20120142729A1 (en) | 2012-06-07 |
| CN103228631B (zh) | 2015-04-29 |
| EP2646417A1 (en) | 2013-10-09 |
| CN103228631A (zh) | 2013-07-31 |
| ZA201303412B (en) | 2014-07-30 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| EEER | Examination request |
Effective date: 20130527 |
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| MKLA | Lapsed |
Effective date: 20181119 |