CA2763207A1 - Cyclosporin derivatives for treating inflammatory diseases and conditions - Google Patents
Cyclosporin derivatives for treating inflammatory diseases and conditions Download PDFInfo
- Publication number
- CA2763207A1 CA2763207A1 CA2763207A CA2763207A CA2763207A1 CA 2763207 A1 CA2763207 A1 CA 2763207A1 CA 2763207 A CA2763207 A CA 2763207A CA 2763207 A CA2763207 A CA 2763207A CA 2763207 A1 CA2763207 A1 CA 2763207A1
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- Prior art keywords
- radical
- cyclosporin
- alkyl
- sar
- alk
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
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- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
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- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
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- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
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Landscapes
- Health & Medical Sciences (AREA)
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- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US18138209P | 2009-05-27 | 2009-05-27 | |
| US61/181,382 | 2009-05-27 | ||
| PCT/US2010/035807 WO2010138423A1 (en) | 2009-05-27 | 2010-05-21 | Cyclosporin derivatives for treating inflammatory diseases and conditions |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CA2763207A1 true CA2763207A1 (en) | 2010-12-02 |
Family
ID=42797341
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CA2763207A Abandoned CA2763207A1 (en) | 2009-05-27 | 2010-05-21 | Cyclosporin derivatives for treating inflammatory diseases and conditions |
Country Status (6)
| Country | Link |
|---|---|
| US (2) | US8524671B2 (https=) |
| EP (1) | EP2435065A1 (https=) |
| JP (1) | JP2012528163A (https=) |
| AU (1) | AU2010254316A1 (https=) |
| CA (1) | CA2763207A1 (https=) |
| WO (1) | WO2010138423A1 (https=) |
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2015519368A (ja) | 2012-06-01 | 2015-07-09 | アラーガン インコーポレイテッドＡｌｌｅｒｇａｎ，Ｉｎｃｏｒｐｏｒａｔｅｄ | シクロスポリンａ類似体 |
| WO2014138425A1 (en) | 2013-03-08 | 2014-09-12 | Allergan, Inc. | Cyclosporine a-steroid conjugates |
| BR112017008433B1 (pt) | 2014-10-31 | 2021-11-03 | Dow Global Technologies Llc | Dispersão de colofônia, processo contínuo para a preparação da dispersão de colofônia e formulação adesiva |
| US9914755B2 (en) | 2015-01-08 | 2018-03-13 | Allergan, Inc. | Cyclosporin derivatives wherein the MeBmt sidechain has been cyclized |
| WO2020037530A1 (en) * | 2018-08-22 | 2020-02-27 | Waterstone Pharmaceuticals (Wuhan) Co., Ltd. | Crystalline form of compound and uses thereof in medicine |
Family Cites Families (13)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP0194972B1 (en) * | 1985-03-11 | 1992-07-29 | Sandoz Ag | Novel cyclosporins |
| JP3034806B2 (ja) * | 1996-08-28 | 2000-04-17 | 富士インジェクタ株式会社 | 回動形切換弁における回動切換機構 |
| FR2757522B1 (fr) * | 1996-12-24 | 1999-01-29 | Rhone Poulenc Rorer Sa | Derives de cyclosporine, leur preparation et les compositions pharmaceutiques qui les contiennent |
| FR2757520B1 (fr) | 1996-12-24 | 1999-01-29 | Rhone Poulenc Rorer Sa | Derive de cyclosporine, sa preparation et les compositions pharmaceutiques qui le contiennent |
| FR2757521B1 (fr) | 1996-12-24 | 1999-01-29 | Rhone Poulenc Rorer Sa | Nouveaux derives de cyclosporine, leur preparation et les compositions pharmaceutiques qui les contiennent |
| FR2762843B1 (fr) * | 1997-04-30 | 1999-12-10 | Rhone Poulenc Rorer Sa | Nouveaux derives de cyclosporine, leur preparation et les compositions pharmaceutiques qui les contiennent |
| US6346511B1 (en) * | 1997-09-08 | 2002-02-12 | Panacea Biotec Limited | Pharmaceutical composition comprising cyclosporin |
| FR2772768B1 (fr) * | 1997-12-19 | 2000-01-14 | Rhone Poulenc Rorer Sa | Nouveau procede de preparation de derives de cyclosporine |
| PT1086124E (pt) * | 1998-06-12 | 2004-04-30 | Chem Ag C | Ciclosporinas novas |
| FR2780061B1 (fr) * | 1998-06-22 | 2001-09-07 | Rhone Poulenc Rorer Sa | Nouveau procede de preparation de derives de cyclosporine |
| US6254860B1 (en) | 1999-04-13 | 2001-07-03 | Allergan Sales, Inc. | Ocular treatment using cyclosporin-A derivatives |
| US20050059583A1 (en) * | 2003-09-15 | 2005-03-17 | Allergan, Inc. | Methods of providing therapeutic effects using cyclosporin components |
| KR20110031973A (ko) | 2008-07-10 | 2011-03-29 | 알러간, 인코포레이티드 | 눈 및 피부의 질환 및 상태를 치료하기 위한 사이클로스포린 유도체 |
-
2010
- 2010-05-21 WO PCT/US2010/035807 patent/WO2010138423A1/en not_active Ceased
- 2010-05-21 CA CA2763207A patent/CA2763207A1/en not_active Abandoned
- 2010-05-21 EP EP10720506A patent/EP2435065A1/en not_active Withdrawn
- 2010-05-21 JP JP2012513144A patent/JP2012528163A/ja active Pending
- 2010-05-21 AU AU2010254316A patent/AU2010254316A1/en not_active Abandoned
- 2010-05-21 US US12/785,133 patent/US8524671B2/en not_active Expired - Fee Related
-
2013
- 2013-08-30 US US14/014,728 patent/US20140005124A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| US8524671B2 (en) | 2013-09-03 |
| JP2012528163A (ja) | 2012-11-12 |
| EP2435065A1 (en) | 2012-04-04 |
| US20140005124A1 (en) | 2014-01-02 |
| AU2010254316A1 (en) | 2011-12-22 |
| US20100305037A1 (en) | 2010-12-02 |
| WO2010138423A1 (en) | 2010-12-02 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| EEER | Examination request |
Effective date: 20150508 |
|
| FZDE | Discontinued |
Effective date: 20170524 |