CA2693024A1 - Synthese catalysee par un metal de transition de 2h-indazoles - Google Patents

Synthese catalysee par un metal de transition de 2h-indazoles Download PDF

Info

Publication number
CA2693024A1
CA2693024A1 CA 2693024 CA2693024A CA2693024A1 CA 2693024 A1 CA2693024 A1 CA 2693024A1 CA 2693024 CA2693024 CA 2693024 CA 2693024 A CA2693024 A CA 2693024A CA 2693024 A1 CA2693024 A1 CA 2693024A1
Authority
CA
Canada
Prior art keywords
unsubstituted
alkyl
phenyl
another
mono
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
CA 2693024
Other languages
English (en)
Inventor
Nis Halland
Marc Nazare
Andreas Lindenschmidt
Jorge Alonso
Omar R'kyek
Matthias Urmann
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Sanofi Aventis France
Original Assignee
Sanofi-Aventis
Nis Halland
Marc Nazare
Andreas Lindenschmidt
Jorge Alonso
Omar R'kyek
Matthias Urmann
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sanofi-Aventis, Nis Halland, Marc Nazare, Andreas Lindenschmidt, Jorge Alonso, Omar R'kyek, Matthias Urmann filed Critical Sanofi-Aventis
Publication of CA2693024A1 publication Critical patent/CA2693024A1/fr
Abandoned legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/54—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings condensed with carbocyclic rings or ring systems
    • C07D231/56—Benzopyrazoles; Hydrogenated benzopyrazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/10—Anthelmintics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/14—Ectoparasiticides, e.g. scabicides

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Catalysts (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Transition And Organic Metals Composition Catalysts For Addition Polymerization (AREA)
CA 2693024 2007-06-26 2008-06-11 Synthese catalysee par un metal de transition de 2h-indazoles Abandoned CA2693024A1 (fr)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP07290799.1 2007-06-26
EP07290799 2007-06-26
PCT/EP2008/004637 WO2009000411A1 (fr) 2007-06-26 2008-06-11 Synthèse catalysée par un métal de transition de 2h-indazoles

Publications (1)

Publication Number Publication Date
CA2693024A1 true CA2693024A1 (fr) 2008-12-31

Family

ID=38577414

Family Applications (1)

Application Number Title Priority Date Filing Date
CA 2693024 Abandoned CA2693024A1 (fr) 2007-06-26 2008-06-11 Synthese catalysee par un metal de transition de 2h-indazoles

Country Status (12)

Country Link
US (1) US8283476B2 (fr)
EP (1) EP2170833B1 (fr)
JP (1) JP5250029B2 (fr)
KR (1) KR20100024963A (fr)
CN (1) CN101687809A (fr)
AT (1) ATE511501T1 (fr)
AU (1) AU2008267442A1 (fr)
BR (1) BRPI0813870A2 (fr)
CA (1) CA2693024A1 (fr)
IL (1) IL202825A0 (fr)
MX (1) MX2009014203A (fr)
WO (1) WO2009000411A1 (fr)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US9487506B2 (en) 2011-04-13 2016-11-08 Merck Sharp & Dohme Corp. Mineralocorticoid receptor antagonists
JP6225356B2 (ja) * 2012-10-31 2017-11-08 ラクオリア創薬株式会社 Ｔｔｘ−ｓ遮断薬としてのピラゾロピリジン誘導体
CN103232462B (zh) * 2013-05-13 2016-03-02 湖北科技学院 香豆素-吡咯类化合物的合成方法
MX2017011579A (es) * 2015-03-12 2018-03-15 Du Pont Pesticidas de tipo azol bicíclicos sustituidos con un heterociclo.
KR101931234B1 (ko) 2016-02-12 2018-12-21 주식회사 엘지화학 신규한 리간드 화합물 및 전이금속 화합물
WO2017138783A1 (fr) * 2016-02-12 2017-08-17 주식회사 엘지화학 Nouveau composé ligand et composé de métal de transition
KR102095007B1 (ko) * 2016-02-12 2020-03-30 주식회사 엘지화학 신규한 리간드 화합물 및 전이금속 화합물의 제조방법
KR102038977B1 (ko) * 2016-12-30 2019-11-01 사빅 에스케이 넥슬렌 컴퍼니 피티이 엘티디 신규한 시클로펜타[ｂ]티오펜일 전이금속 화합물, 이를 포함하는 전이금속 촉매 조성물, 및 이를 이용한 에틸렌 단독중합체 또는 에틸렌과 α-올레핀의 공중합체의 제조방법
KR20210033444A (ko) 2018-06-04 2021-03-26 엑스사이언티아 엘티디 아데노신 수용체 길항제로서 피라졸로피리미딘 화합물
CN110317204B (zh) * 2019-08-02 2022-02-08 安徽农业大学 吡唑并嘧啶酮类衍生物及其制备方法和应用
CN113698349B (zh) * 2021-09-02 2023-08-01 河南师范大学 一种2-(2-苯基-2h-吲唑-3-基)乙酸酯类化合物的水相光催化制备方法
CN114920699B (zh) * 2022-05-31 2024-03-19 甘肃皓天科技股份有限公司 一种制备6-氯-2-甲基-2h-吲唑-5-胺的方法

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP4647780B2 (ja) * 1998-02-26 2011-03-09 マサチューセッツ インスティテュート オブ テクノロジー ヒドラジン、ヒドラゾン、ヒドロキシルアミンおよびオキシムの金属−触媒アリール化およびビニル化

Also Published As

Publication number Publication date
AU2008267442A1 (en) 2008-12-31
WO2009000411A1 (fr) 2008-12-31
KR20100024963A (ko) 2010-03-08
US8283476B2 (en) 2012-10-09
JP2010531311A (ja) 2010-09-24
EP2170833A1 (fr) 2010-04-07
EP2170833B1 (fr) 2011-06-01
JP5250029B2 (ja) 2013-07-31
BRPI0813870A2 (pt) 2015-01-06
US20100234601A1 (en) 2010-09-16
ATE511501T1 (de) 2011-06-15
CN101687809A (zh) 2010-03-31
MX2009014203A (es) 2010-01-28
IL202825A0 (en) 2010-06-30

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Legal Events

Date Code Title Description
FZDE Discontinued

Effective date: 20130611