CA2671632A1 - Novel protein kinase modulators and therapeutic uses thereof - Google Patents
Novel protein kinase modulators and therapeutic uses thereof Download PDFInfo
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- CA2671632A1 CA2671632A1 CA002671632A CA2671632A CA2671632A1 CA 2671632 A1 CA2671632 A1 CA 2671632A1 CA 002671632 A CA002671632 A CA 002671632A CA 2671632 A CA2671632 A CA 2671632A CA 2671632 A1 CA2671632 A1 CA 2671632A1
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Classifications
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- C07C327/40—Amides of thiocarboxylic acids having carbon atoms of thiocarboxamide groups bound to hydrogen atoms or to acyclic carbon atoms
- C07C327/44—Amides of thiocarboxylic acids having carbon atoms of thiocarboxamide groups bound to hydrogen atoms or to acyclic carbon atoms to carbon atoms of an unsaturated carbon skeleton
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Landscapes
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- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
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- Emergency Medicine (AREA)
- Immunology (AREA)
- Heart & Thoracic Surgery (AREA)
- Cardiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Enzymes And Modification Thereof (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US87251106P | 2006-12-04 | 2006-12-04 | |
| US60/872,511 | 2006-12-04 | ||
| PCT/IL2007/001494 WO2008068751A1 (en) | 2006-12-04 | 2007-12-04 | Novel protein kinase modulators and therapeutic uses thereof |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CA2671632A1 true CA2671632A1 (en) | 2008-06-12 |
Family
ID=39111493
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CA002671632A Abandoned CA2671632A1 (en) | 2006-12-04 | 2007-12-04 | Novel protein kinase modulators and therapeutic uses thereof |
Country Status (8)
| Country | Link |
|---|---|
| US (1) | US8058309B2 (https=) |
| EP (1) | EP2125712B1 (https=) |
| JP (1) | JP2010511694A (https=) |
| CN (1) | CN101652345A (https=) |
| AU (1) | AU2007330333A1 (https=) |
| BR (1) | BRPI0719708A2 (https=) |
| CA (1) | CA2671632A1 (https=) |
| WO (1) | WO2008068751A1 (https=) |
Families Citing this family (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP2285774B1 (en) | 2008-06-05 | 2015-02-25 | Yissum Research Development Company of the Hebrew University of Jerusalem Ltd. | Novel modulators of protein kinase signaling |
| EP2658847B1 (en) * | 2010-12-27 | 2015-12-23 | Yissum Research Development Company of the Hebrew University of Jerusalem Ltd. | 2-(2-phenylethenyl)-1,3-benzothiazine derivatives useful for the treatment of cancer |
| WO2012117396A1 (en) | 2011-03-01 | 2012-09-07 | Novotyr Therapeutics Ltd | Tyrphostin derivative in combination with cytotoxic compounds for treating cancer |
| US9770454B2 (en) | 2013-07-14 | 2017-09-26 | Yissum Research Development Company Of The Hebrew University Of Jerusalem, Ltd. | IGF-1R signaling pathway inhibitors useful in the treatment of neurodegenerative diseases |
| CN112353938A (zh) | 2015-02-05 | 2021-02-12 | 特尔诺沃有限公司 | 用于治疗癌症的irs/stat3双重调节剂与抗癌剂的组合 |
| EP3710050A4 (en) * | 2017-11-16 | 2021-06-16 | TyrNovo Ltd. | COMBINATIONS OF IRS / STAT3 DOUBLE MODULATORS AND ANTI-PD-1 / PD-L1 AMBODIES FOR TREATMENT OF CANCER |
| WO2019246273A1 (en) | 2018-06-20 | 2019-12-26 | Progenity, Inc. | Treatment of a disease of the gastrointestinal tract with a jak or other kinase inhibitor |
| CN115466205B (zh) * | 2021-11-04 | 2023-10-24 | 特尔诺沃有限公司 | 分离的3-（2-溴-3,4-二羟基-苯基）-n-（3,4,5-三羟基-苄基）-硫代丙烯酰胺的反式异构体 |
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|---|---|---|---|---|
| US5217999A (en) | 1987-12-24 | 1993-06-08 | Yissum Research Development Company Of The Hebrew University Of Jerusalem | Styryl compounds which inhibit EGF receptor protein tyrosine kinase |
| WO1995024190A2 (en) * | 1994-03-07 | 1995-09-14 | Sugen, Inc. | Receptor tyrosine kinase inhibitors for inhibiting cell proliferative disorders and compositions thereof |
| IL159270A0 (en) * | 2001-06-14 | 2004-06-01 | Yissum Res Dev Co | Non-myeloablative tolerogenic treatment with tyrphostins |
| ATE517617T1 (de) * | 2001-12-10 | 2011-08-15 | Yansheng Dr Du | Behandlung von parkinson erkrankung mit kape |
| PT2527315E (pt) * | 2002-05-31 | 2014-06-24 | Proteotech Inc | Compostos, composições e métodos para o tratamento de doenças da amiloide e sinucleínopatias tais como doença de alzheimer, diabetes do tipo 2, e doença de parkinson |
-
2007
- 2007-12-04 WO PCT/IL2007/001494 patent/WO2008068751A1/en not_active Ceased
- 2007-12-04 EP EP07827467.7A patent/EP2125712B1/en active Active
- 2007-12-04 US US12/517,278 patent/US8058309B2/en active Active
- 2007-12-04 CN CN200780050587A patent/CN101652345A/zh active Pending
- 2007-12-04 BR BRPI0719708-0A2A patent/BRPI0719708A2/pt not_active Application Discontinuation
- 2007-12-04 CA CA002671632A patent/CA2671632A1/en not_active Abandoned
- 2007-12-04 JP JP2009539869A patent/JP2010511694A/ja active Pending
- 2007-12-04 AU AU2007330333A patent/AU2007330333A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| US20100056635A1 (en) | 2010-03-04 |
| EP2125712A1 (en) | 2009-12-02 |
| AU2007330333A1 (en) | 2008-06-12 |
| JP2010511694A (ja) | 2010-04-15 |
| US8058309B2 (en) | 2011-11-15 |
| WO2008068751A1 (en) | 2008-06-12 |
| BRPI0719708A2 (pt) | 2014-02-18 |
| EP2125712B1 (en) | 2014-07-23 |
| CN101652345A (zh) | 2010-02-17 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FZDE | Discontinued |
Effective date: 20131204 |