CA2485166A1 - Substituted pyrimidinone and pyridinone compounds - Google Patents

Substituted pyrimidinone and pyridinone compounds Download PDF

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Publication number
CA2485166A1
CA2485166A1 CA002485166A CA2485166A CA2485166A1 CA 2485166 A1 CA2485166 A1 CA 2485166A1 CA 002485166 A CA002485166 A CA 002485166A CA 2485166 A CA2485166 A CA 2485166A CA 2485166 A1 CA2485166 A1 CA 2485166A1
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CA
Canada
Prior art keywords
methyl
substituted
pyrrolidin
naphthalen
groups
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
CA002485166A
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English (en)
French (fr)
Inventor
Celia Dominguez
Dawei Zhang
Guo-Qiang Cao
Martin H. Goldberg
Fang-Tsao Hong
Kelvin K. C. Sham
Seifu Tadesse
Nuria A. Tamayo
Kurt E. Weiler
Hongyu Liao
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Amgen Inc
Original Assignee
Individual
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Filing date
Publication date
Application filed by Individual filed Critical Individual
Publication of CA2485166A1 publication Critical patent/CA2485166A1/en
Abandoned legal-status Critical Current

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
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    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
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  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
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  • Molecular Biology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Hematology (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Dermatology (AREA)
  • Neurosurgery (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Pain & Pain Management (AREA)
  • Cardiology (AREA)
  • Biotechnology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Hospice & Palliative Care (AREA)
  • Transplantation (AREA)
  • Emergency Medicine (AREA)
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CA002485166A 2002-05-21 2003-05-13 Substituted pyrimidinone and pyridinone compounds Abandoned CA2485166A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US38269902P 2002-05-21 2002-05-21
US60/382,699 2002-05-21
PCT/US2003/015473 WO2003099808A1 (en) 2002-05-21 2003-05-13 Substituted heterocyclic compounds and methods of use

Publications (1)

Publication Number Publication Date
CA2485166A1 true CA2485166A1 (en) 2003-12-04

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Application Number Title Priority Date Filing Date
CA002485166A Abandoned CA2485166A1 (en) 2002-05-21 2003-05-13 Substituted pyrimidinone and pyridinone compounds

Country Status (10)

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US (1) US7026326B2 (US07094801-20060822-C00173.png)
EP (1) EP1506186A1 (US07094801-20060822-C00173.png)
JP (2) JP4606161B2 (US07094801-20060822-C00173.png)
AR (1) AR039842A1 (US07094801-20060822-C00173.png)
AU (1) AU2003234628B2 (US07094801-20060822-C00173.png)
CA (1) CA2485166A1 (US07094801-20060822-C00173.png)
MX (1) MXPA04011470A (US07094801-20060822-C00173.png)
PL (1) PL376575A1 (US07094801-20060822-C00173.png)
TW (1) TW200406399A (US07094801-20060822-C00173.png)
WO (1) WO2003099808A1 (US07094801-20060822-C00173.png)

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