CA2466971A1 - Benzimidazol- or indol-aminoacetonitrile derivatives for parasite control - Google Patents
Benzimidazol- or indol-aminoacetonitrile derivatives for parasite control Download PDFInfo
- Publication number
- CA2466971A1 CA2466971A1 CA002466971A CA2466971A CA2466971A1 CA 2466971 A1 CA2466971 A1 CA 2466971A1 CA 002466971 A CA002466971 A CA 002466971A CA 2466971 A CA2466971 A CA 2466971A CA 2466971 A1 CA2466971 A1 CA 2466971A1
- Authority
- CA
- Canada
- Prior art keywords
- halo
- alkyl
- och3
- alkoxy
- thiazol
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
- C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
- C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
- C07D235/06—Benzimidazoles; Hydrogenated benzimidazoles with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 2
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/10—Anthelmintics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/14—Ectoparasiticides, e.g. scabicides
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/04—Indoles; Hydrogenated indoles
- C07D209/08—Indoles; Hydrogenated indoles with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, directly attached to carbon atoms of the hetero ring
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
- C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
- C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
- C07D235/06—Benzimidazoles; Hydrogenated benzimidazoles with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 2
- C07D235/10—Radicals substituted by halogen atoms or nitro radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
- C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
- C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
- C07D235/24—Benzimidazoles; Hydrogenated benzimidazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
- C07D235/28—Sulfur atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Life Sciences & Earth Sciences (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- General Chemical & Material Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Tropical Medicine & Parasitology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Plural Heterocyclic Compounds (AREA)
- Indole Compounds (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CH2103/01 | 2001-11-14 | ||
| CH21032001 | 2001-11-14 | ||
| PCT/EP2002/012709 WO2003042184A1 (en) | 2001-11-14 | 2002-11-13 | Benzimidazol- or indol-aminoacetonitrile derivatives for parasite control |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CA2466971A1 true CA2466971A1 (en) | 2003-05-22 |
Family
ID=4567523
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CA002466971A Abandoned CA2466971A1 (en) | 2001-11-14 | 2002-11-13 | Benzimidazol- or indol-aminoacetonitrile derivatives for parasite control |
Country Status (16)
| Country | Link |
|---|---|
| US (1) | US7279495B2 (https=) |
| EP (1) | EP1446386A1 (https=) |
| JP (1) | JP2005518351A (https=) |
| KR (1) | KR20050044451A (https=) |
| CN (1) | CN1304378C (https=) |
| AR (1) | AR037363A1 (https=) |
| AU (1) | AU2002351995B2 (https=) |
| BR (1) | BR0214151A (https=) |
| CA (1) | CA2466971A1 (https=) |
| CO (1) | CO5390082A1 (https=) |
| MX (1) | MXPA04004605A (https=) |
| NZ (1) | NZ532864A (https=) |
| RU (1) | RU2004118247A (https=) |
| TW (1) | TW200300140A (https=) |
| WO (1) | WO2003042184A1 (https=) |
| ZA (1) | ZA200403459B (https=) |
Families Citing this family (21)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AR042420A1 (es) | 2002-09-11 | 2005-06-22 | Novartis Ag | Benzotriazolil- aminoacetonitril compuestos, proceso para su preparacion, metodo y uso de los mismos en el control de endo- y ecto-parasitos dentro y sobre ganado productor de sangre caliente y animales domesticos y plantas, y en la preparacion de una composicion farmaceutica |
| US20040192738A1 (en) * | 2003-03-18 | 2004-09-30 | Aventis Pharma Deutschland Gmbh | 2-(Butyl-1-sulfonylamino)-N-[1(R)-(6-methoxypyridin-3-yl)propyl] benzamide, its use as a medicament, and pharmaceutical preparations comprising it |
| GB0402677D0 (en) * | 2003-11-06 | 2004-03-10 | Novartis Ag | Organic compounds |
| WO2006043654A1 (ja) * | 2004-10-22 | 2006-04-27 | Nihon Nohyaku Co., Ltd. | アセトニトリル誘導体及び有害生物防除剤並びにその使用方法 |
| WO2007006739A1 (en) * | 2005-07-12 | 2007-01-18 | Bayer Cropscience Sa | Benzoheterocyclylethylcarboxamide derivatives |
| PE20070335A1 (es) | 2005-08-30 | 2007-04-21 | Novartis Ag | Benzimidazoles sustituidos y metodos para su preparacion |
| RS55271B1 (sr) | 2007-05-15 | 2017-02-28 | Merial Sas | Ariloazol-2-il cijanoetilamino jedinjenja, postupci dobijanja i postupci njihove primene |
| AR072297A1 (es) | 2008-06-27 | 2010-08-18 | Novartis Ag | Derivados de indol-2-il-piridin-3-ilo, composicion farmaceutica que los comprende y su uso en medicamentos para el tratamiento de enfermedades mediadas por la sintasa aldosterona. |
| MX2011004217A (es) | 2008-10-21 | 2011-06-20 | Merial Ltd | Compuestos de tioamida, metodo de elaboracion y metodo para usarlos. |
| AR074024A1 (es) | 2008-11-14 | 2010-12-15 | Merial Ltd | Compuesto de arilazol-2-il-cianoetilamino enantiomericamente enriquecidos, composicion plaguicida y su uso para prevenir la infeccion parasitaria |
| GB0905365D0 (en) | 2009-03-27 | 2009-05-13 | Norbrook Lab Ltd | A topical parasiticide composition |
| US20100307542A1 (en) * | 2009-06-05 | 2010-12-09 | Kraft Foods Global Brands Llc | Method of Reducing Surface Oil on Encapsulated Material |
| US9968564B2 (en) * | 2009-06-05 | 2018-05-15 | Intercontinental Great Brands Llc | Delivery of functional compounds |
| US20100310726A1 (en) | 2009-06-05 | 2010-12-09 | Kraft Foods Global Brands Llc | Novel Preparation of an Enteric Release System |
| US8859003B2 (en) * | 2009-06-05 | 2014-10-14 | Intercontinental Great Brands Llc | Preparation of an enteric release system |
| BR122015032741B1 (pt) * | 2012-04-20 | 2019-11-26 | Merial Ltd | composições parasiticídicas compreendendo derivados de benzimidazol, métodos e seus usos |
| US8822689B2 (en) | 2012-09-19 | 2014-09-02 | Merial Limited | Aryloazol-2-yl cyanoethylamino compounds, method of making and method of using thereof |
| US8859005B2 (en) | 2012-12-03 | 2014-10-14 | Intercontinental Great Brands Llc | Enteric delivery of functional ingredients suitable for hot comestible applications |
| US10493416B2 (en) * | 2014-05-08 | 2019-12-03 | Osaka University | Thermal convection generating chip and liquid measuring device |
| EP3157912B1 (en) * | 2014-06-19 | 2019-02-20 | Merial, Inc. | Parasiticidal compositions comprising indole derivatives, methods and uses thereof |
| BR112021024726A2 (pt) * | 2019-06-07 | 2022-01-18 | Elanco Tiergesundheit Ag | Novos derivados bicíclicos |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6239077B1 (en) | 1998-05-01 | 2001-05-29 | Nihon Nohyaku Co., Ltd. | Aminoacetonitrile derivative agricultural and horticultural insecticide containing the same and use thereof |
-
2002
- 2002-11-12 TW TW091133121A patent/TW200300140A/zh unknown
- 2002-11-13 AU AU2002351995A patent/AU2002351995B2/en not_active Ceased
- 2002-11-13 RU RU2004118247/04A patent/RU2004118247A/ru not_active Application Discontinuation
- 2002-11-13 CN CNB028241053A patent/CN1304378C/zh not_active Expired - Fee Related
- 2002-11-13 MX MXPA04004605A patent/MXPA04004605A/es unknown
- 2002-11-13 US US10/494,897 patent/US7279495B2/en not_active Expired - Fee Related
- 2002-11-13 BR BR0214151-5A patent/BR0214151A/pt not_active IP Right Cessation
- 2002-11-13 KR KR1020047007293A patent/KR20050044451A/ko not_active Withdrawn
- 2002-11-13 JP JP2003544020A patent/JP2005518351A/ja not_active Withdrawn
- 2002-11-13 WO PCT/EP2002/012709 patent/WO2003042184A1/en not_active Ceased
- 2002-11-13 NZ NZ532864A patent/NZ532864A/xx unknown
- 2002-11-13 AR ARP020104355A patent/AR037363A1/es not_active Application Discontinuation
- 2002-11-13 EP EP02787667A patent/EP1446386A1/en not_active Withdrawn
- 2002-11-13 CA CA002466971A patent/CA2466971A1/en not_active Abandoned
- 2002-11-14 CO CO02103446A patent/CO5390082A1/es not_active Application Discontinuation
-
2004
- 2004-05-06 ZA ZA200403459A patent/ZA200403459B/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| EP1446386A1 (en) | 2004-08-18 |
| US7279495B2 (en) | 2007-10-09 |
| US20050026972A1 (en) | 2005-02-03 |
| AU2002351995B2 (en) | 2006-08-10 |
| KR20050044451A (ko) | 2005-05-12 |
| AR037363A1 (es) | 2004-11-03 |
| NZ532864A (en) | 2005-11-25 |
| BR0214151A (pt) | 2004-09-14 |
| RU2004118247A (ru) | 2006-01-10 |
| TW200300140A (en) | 2003-05-16 |
| JP2005518351A (ja) | 2005-06-23 |
| WO2003042184A1 (en) | 2003-05-22 |
| MXPA04004605A (es) | 2005-03-07 |
| CN1599725A (zh) | 2005-03-23 |
| CO5390082A1 (es) | 2004-04-30 |
| CN1304378C (zh) | 2007-03-14 |
| ZA200403459B (en) | 2006-11-29 |
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| AU2002351995A1 (en) | Benzimidazol-or indol-aminoacetonitrile derivatives for parasite control | |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FZDE | Discontinued |