CA2393452A1 - Utilisation de l'histamine comme compose ameliorant la liberation de medicaments dans l'administration par voie transmuqueuse ou transdermique - Google Patents
Utilisation de l'histamine comme compose ameliorant la liberation de medicaments dans l'administration par voie transmuqueuse ou transdermique Download PDFInfo
- Publication number
- CA2393452A1 CA2393452A1 CA002393452A CA2393452A CA2393452A1 CA 2393452 A1 CA2393452 A1 CA 2393452A1 CA 002393452 A CA002393452 A CA 002393452A CA 2393452 A CA2393452 A CA 2393452A CA 2393452 A1 CA2393452 A1 CA 2393452A1
- Authority
- CA
- Canada
- Prior art keywords
- histamine
- composition
- transmucosally
- enhancing agent
- transmucosal
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
- A61K47/22—Heterocyclic compounds, e.g. ascorbic acid, tocopherol or pyrrolidones
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0014—Skin, i.e. galenical aspects of topical compositions
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Public Health (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Animal Behavior & Ethology (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Engineering & Computer Science (AREA)
- Oil, Petroleum & Natural Gas (AREA)
- Dermatology (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
La présente invention concerne une composition à administration transmuqueuse à pénétration améliorée comprenant: entre environ 0,001 % et environ 25 % d'un agent améliorant la perméation choisi dans le groupe composé de l'histamine, du dichlorhydrate d'histamine, du phosphate d'histamine, d'un sel pharmaceutiquement acceptable de ces derniers, d'autres agonistes de l'histamine; entre environ 0,2 % et environ 90 % d'un médicament pharmaceutiquement actif; entre environ 0 % et environ 99,8 % d'un solvant; et entre environ 0 % et environ 50 % d'un agent gélifiant.
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US14664199P | 1999-07-30 | 1999-07-30 | |
US60/146,641 | 1999-07-30 | ||
PCT/US2000/020757 WO2001008706A1 (fr) | 1999-07-30 | 2000-07-28 | Utilisation de l'histamine comme compose ameliorant la liberation de medicaments dans l'administration par voie transmuqueuse ou transdermique |
Publications (1)
Publication Number | Publication Date |
---|---|
CA2393452A1 true CA2393452A1 (fr) | 2001-02-08 |
Family
ID=22518302
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CA002393452A Abandoned CA2393452A1 (fr) | 1999-07-30 | 2000-07-28 | Utilisation de l'histamine comme compose ameliorant la liberation de medicaments dans l'administration par voie transmuqueuse ou transdermique |
Country Status (5)
Country | Link |
---|---|
EP (1) | EP1229939A1 (fr) |
AU (1) | AU6751000A (fr) |
CA (1) | CA2393452A1 (fr) |
HK (1) | HK1048770A1 (fr) |
WO (1) | WO2001008706A1 (fr) |
Cited By (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2015089661A1 (fr) * | 2013-12-17 | 2015-06-25 | Contech Enterprises Inc. | Composés, compositions et procédés pour attirer et/ou retenir des punaises des lits |
Families Citing this family (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2016068336A1 (fr) * | 2014-10-30 | 2016-05-06 | 旭化成ケミカルズ株式会社 | Agent et agent auxiliaire de promotion d'absorption transdermique |
CN110075063A (zh) * | 2019-05-27 | 2019-08-02 | 合肥亿帆生物医药有限公司 | 一种二盐酸组胺注射液及其制备方法 |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4521405A (en) * | 1982-05-17 | 1985-06-04 | John McMichael | Methods and materials for treatment of disease states involving immunological factors |
HU223205B1 (hu) * | 1996-12-03 | 2004-03-29 | Zoltán Dárdai | Helyileg alkalmazható készítmény peptidszerű gyógyhatású vegyületek élő szervezetbe vitelére |
US6270781B1 (en) * | 1999-01-08 | 2001-08-07 | Maxim Pharmaceuticals, Inc. | Method and compositions for topical treatment of damaged tissue using reactive oxygen metabolite production or release inhibitors |
-
2000
- 2000-07-28 WO PCT/US2000/020757 patent/WO2001008706A1/fr not_active Application Discontinuation
- 2000-07-28 AU AU67510/00A patent/AU6751000A/en not_active Abandoned
- 2000-07-28 CA CA002393452A patent/CA2393452A1/fr not_active Abandoned
- 2000-07-28 EP EP00955284A patent/EP1229939A1/fr not_active Withdrawn
-
2003
- 2003-02-12 HK HK03101024.5A patent/HK1048770A1/zh unknown
Cited By (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2015089661A1 (fr) * | 2013-12-17 | 2015-06-25 | Contech Enterprises Inc. | Composés, compositions et procédés pour attirer et/ou retenir des punaises des lits |
CN105899074A (zh) * | 2013-12-17 | 2016-08-24 | 西蒙弗雷泽大学 | 用于吸引和/或捕捉臭虫的化合物、组合物和方法 |
AU2014366768B2 (en) * | 2013-12-17 | 2017-10-12 | Simon Fraser University | Compounds, compositions and methods for attracting and/or arresting bed bugs |
RU2678226C1 (ru) * | 2013-12-17 | 2019-01-24 | Саймон Фрейзер Юниверсити | Соединения, композиции и способы приманивания и/или поимки постельных клопов |
CN105899074B (zh) * | 2013-12-17 | 2019-09-24 | 西蒙弗雷泽大学 | 用于吸引和/或捕捉臭虫的化合物、组合物和方法 |
US11553717B2 (en) | 2013-12-17 | 2023-01-17 | Simon Fraser University | Compounds, compositions and methods for attracting and/or arresting bed bugs |
Also Published As
Publication number | Publication date |
---|---|
AU6751000A (en) | 2001-02-19 |
WO2001008706A1 (fr) | 2001-02-08 |
EP1229939A1 (fr) | 2002-08-14 |
HK1048770A1 (zh) | 2003-04-17 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
EEER | Examination request | ||
FZDE | Dead |