CA2340486A1 - Process for preparing resorcinol derivatives - Google Patents

Process for preparing resorcinol derivatives Download PDF

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Publication number
CA2340486A1
CA2340486A1 CA002340486A CA2340486A CA2340486A1 CA 2340486 A1 CA2340486 A1 CA 2340486A1 CA 002340486 A CA002340486 A CA 002340486A CA 2340486 A CA2340486 A CA 2340486A CA 2340486 A1 CA2340486 A1 CA 2340486A1
Authority
CA
Canada
Prior art keywords
alkyl
aryl
formula
compound
acyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
CA002340486A
Other languages
English (en)
French (fr)
Inventor
John Kitchin
Graham Michael Wynne
Stuart Edward Bradley
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pfizer Products Inc
Original Assignee
Pfizer Products Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Products Inc filed Critical Pfizer Products Inc
Publication of CA2340486A1 publication Critical patent/CA2340486A1/en
Abandoned legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C37/00—Preparation of compounds having hydroxy or O-metal groups bound to a carbon atom of a six-membered aromatic ring
    • C07C37/06—Preparation of compounds having hydroxy or O-metal groups bound to a carbon atom of a six-membered aromatic ring by conversion of non-aromatic six-membered rings or of such rings formed in situ into aromatic six-membered rings, e.g. by dehydrogenation
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D317/00—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms
    • C07D317/08—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3
    • C07D317/72—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 spiro-condensed with carbocyclic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C37/00—Preparation of compounds having hydroxy or O-metal groups bound to a carbon atom of a six-membered aromatic ring
    • C07C37/06—Preparation of compounds having hydroxy or O-metal groups bound to a carbon atom of a six-membered aromatic ring by conversion of non-aromatic six-membered rings or of such rings formed in situ into aromatic six-membered rings, e.g. by dehydrogenation
    • C07C37/07—Preparation of compounds having hydroxy or O-metal groups bound to a carbon atom of a six-membered aromatic ring by conversion of non-aromatic six-membered rings or of such rings formed in situ into aromatic six-membered rings, e.g. by dehydrogenation with simultaneous reduction of C=O group in that ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C45/00—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
    • C07C45/56—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds from heterocyclic compounds
    • C07C45/57—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds from heterocyclic compounds with oxygen as the only heteroatom
    • C07C45/59—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds from heterocyclic compounds with oxygen as the only heteroatom in five-membered rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C45/00—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
    • C07C45/61—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups
    • C07C45/67—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton
    • C07C45/68—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton by increase in the number of carbon atoms
    • C07C45/70—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton by increase in the number of carbon atoms by reaction with functional groups containing oxygen only in singly bound form
    • C07C45/71—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton by increase in the number of carbon atoms by reaction with functional groups containing oxygen only in singly bound form being hydroxy groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C49/00—Ketones; Ketenes; Dimeric ketenes; Ketonic chelates
    • C07C49/587—Unsaturated compounds containing a keto groups being part of a ring
    • C07C49/703—Unsaturated compounds containing a keto groups being part of a ring containing hydroxy groups
    • C07C49/747—Unsaturated compounds containing a keto groups being part of a ring containing hydroxy groups containing six-membered aromatic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2601/00—Systems containing only non-condensed rings
    • C07C2601/12—Systems containing only non-condensed rings with a six-membered ring
    • C07C2601/14—The ring being saturated
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2601/00—Systems containing only non-condensed rings
    • C07C2601/18—Systems containing only non-condensed rings with a ring being at least seven-membered
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y10—TECHNICAL SUBJECTS COVERED BY FORMER USPC
    • Y10S—TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y10S977/00—Nanotechnology
    • Y10S977/902—Specified use of nanostructure
    • Y10S977/904—Specified use of nanostructure for medical, immunological, body treatment, or diagnosis
    • Y10S977/926—Topical chemical, e.g. cosmetic or sunscreen

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Plural Heterocyclic Compounds (AREA)
CA002340486A 2000-03-15 2001-03-13 Process for preparing resorcinol derivatives Abandoned CA2340486A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US18970400P 2000-03-15 2000-03-15
US60/189,704 2000-03-15

Publications (1)

Publication Number Publication Date
CA2340486A1 true CA2340486A1 (en) 2001-09-15

Family

ID=22698426

Family Applications (1)

Application Number Title Priority Date Filing Date
CA002340486A Abandoned CA2340486A1 (en) 2000-03-15 2001-03-13 Process for preparing resorcinol derivatives

Country Status (18)

Country Link
US (3) US6504037B2 (US20070244113A1-20071018-C00087.png)
EP (1) EP1134207A1 (US20070244113A1-20071018-C00087.png)
JP (1) JP2001294549A (US20070244113A1-20071018-C00087.png)
KR (1) KR100432303B1 (US20070244113A1-20071018-C00087.png)
CN (1) CN1325838A (US20070244113A1-20071018-C00087.png)
AR (1) AR030055A1 (US20070244113A1-20071018-C00087.png)
AU (1) AU782397B2 (US20070244113A1-20071018-C00087.png)
BR (1) BR0100982A (US20070244113A1-20071018-C00087.png)
CA (1) CA2340486A1 (US20070244113A1-20071018-C00087.png)
CZ (1) CZ2001930A3 (US20070244113A1-20071018-C00087.png)
HK (1) HK1040987A1 (US20070244113A1-20071018-C00087.png)
ID (1) ID29673A (US20070244113A1-20071018-C00087.png)
IL (1) IL141915A0 (US20070244113A1-20071018-C00087.png)
IN (1) IN192530B (US20070244113A1-20071018-C00087.png)
PL (1) PL346463A1 (US20070244113A1-20071018-C00087.png)
RU (1) RU2213087C2 (US20070244113A1-20071018-C00087.png)
YU (1) YU18601A (US20070244113A1-20071018-C00087.png)
ZA (1) ZA200102070B (US20070244113A1-20071018-C00087.png)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN111909012A (zh) * 2020-08-24 2020-11-10 浙江工业大学台州研究院 一种高选择性、高转化制备1,3-环己二酮的方法

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6828460B2 (en) * 1999-03-22 2004-12-07 Pfizer Inc. Resorcinol derivatives
US6863897B2 (en) * 2002-03-22 2005-03-08 Unilever Home & Personal Care Usa, Division Of Conopco, Inc. Stabilization of resorcinol derivatives in cosmetic compositions
JP4228605B2 (ja) 2002-07-02 2009-02-25 住友化学株式会社 改変型還元酵素、その遺伝子及びそれらの利用
JP4228606B2 (ja) 2002-07-03 2009-02-25 住友化学株式会社 改変型還元酵素、その遺伝子及びそれらの利用
US6852310B2 (en) 2002-08-23 2005-02-08 Unilever Home & Personal Care Usa Division Of Conopco, Inc. Skin lightening agents, compositions and methods
US7163327B2 (en) * 2002-12-02 2007-01-16 3M Innovative Properties Company Illumination system using a plurality of light sources
US6875425B2 (en) 2002-12-12 2005-04-05 Unilever Home & Personal Care Usa Skin lightening agents, compositions and methods
US7524485B2 (en) 2002-12-12 2009-04-28 Unilever Home & Personal Care, Usa, Division Of Conopco, Inc. Skin lightening agents, compositions and methods
US7338979B2 (en) 2003-02-11 2008-03-04 Warner-Lambert Company Depigmentation agents
US7300646B2 (en) * 2004-02-27 2007-11-27 Unilever Home & Personal Care Usa, Division Of Conopco, Inc. Skin lightening agents, compositions and methods
US20060062865A1 (en) * 2004-09-17 2006-03-23 Nebojsa Ilic Tyrosinase inhibitor and method for preparation
US20060210498A1 (en) 2005-03-18 2006-09-21 Unilever Home & Personal Care Usa, Division Of Conopco, Inc. Novel resorcinol derivatives for skin
US20060210497A1 (en) * 2005-03-18 2006-09-21 Unilever Home & Personal Care Usa, Division Of Conopco, Inc. Novel resorcinol derivatives
US7270805B1 (en) 2006-03-30 2007-09-18 Conopco, Inc. Skin lightening agents, compositions and methods
US7247294B1 (en) 2006-03-30 2007-07-24 Conopco, Inc. Skin lightening agents, compositions and methods
US7250158B1 (en) 2006-03-30 2007-07-31 Conopco, Inc. Skin lightening agents, compositions and methods
US20140256830A1 (en) 2013-03-08 2014-09-11 Ampere Life Sciences, Inc. Resorcinol compounds for dermatological use
MX369987B (es) 2016-06-15 2019-11-27 Unilever Nv Metodo y composicion cosmetica para un suministro transdermico mejorado de resorcinol alquilo sustituido.

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PA8469601A1 (es) * 1998-04-10 2000-09-29 Pfizer Prod Inc Procedimiento para alquilar sulfonamidas impedidas estericamente
CA2362698C (en) * 1999-03-22 2005-02-01 Pfizer Inc. Resorcinol derivatives

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN111909012A (zh) * 2020-08-24 2020-11-10 浙江工业大学台州研究院 一种高选择性、高转化制备1,3-环己二酮的方法
CN111909012B (zh) * 2020-08-24 2022-10-21 浙江工业大学台州研究院 一种高选择性、高转化制备1,3-环己二酮的方法

Also Published As

Publication number Publication date
ID29673A (id) 2001-09-20
US6861564B2 (en) 2005-03-01
US20020032352A1 (en) 2002-03-14
KR20010096608A (ko) 2001-11-07
CZ2001930A3 (cs) 2001-10-17
JP2001294549A (ja) 2001-10-23
BR0100982A (pt) 2001-12-04
EP1134207A1 (en) 2001-09-19
US20030088113A1 (en) 2003-05-08
CN1325838A (zh) 2001-12-12
RU2213087C2 (ru) 2003-09-27
YU18601A (sh) 2003-07-07
ZA200102070B (en) 2002-09-13
IL141915A0 (en) 2002-03-10
AR030055A1 (es) 2003-08-13
US6504037B2 (en) 2003-01-07
KR100432303B1 (ko) 2004-05-20
AU782397B2 (en) 2005-07-21
IN192530B (US20070244113A1-20071018-C00087.png) 2004-04-24
PL346463A1 (en) 2001-09-24
HK1040987A1 (zh) 2002-06-28
US20050143594A1 (en) 2005-06-30
AU2647701A (en) 2001-09-20

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Legal Events

Date Code Title Description
EEER Examination request
FZDE Discontinued