CA2240404A1 - Naphtylglyoxamides en tant qu'inhibiteurs de spla2 - Google Patents

Naphtylglyoxamides en tant qu'inhibiteurs de spla2 Download PDF

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Publication number
CA2240404A1
CA2240404A1 CA 2240404 CA2240404A CA2240404A1 CA 2240404 A1 CA2240404 A1 CA 2240404A1 CA 2240404 CA2240404 CA 2240404 CA 2240404 A CA2240404 A CA 2240404A CA 2240404 A1 CA2240404 A1 CA 2240404A1
Authority
CA
Canada
Prior art keywords
compound
formula
acid
compounds
naphthyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
CA 2240404
Other languages
English (en)
Inventor
David Kent Herron
Theodore Goodson Jr.
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Eli Lilly and Co
Original Assignee
Individual
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GBGB9602268.6A external-priority patent/GB9602268D0/en
Application filed by Individual filed Critical Individual
Priority claimed from PCT/US1996/019529 external-priority patent/WO1997021716A1/fr
Publication of CA2240404A1 publication Critical patent/CA2240404A1/fr
Abandoned legal-status Critical Current

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  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

L'invention concerne une catégorie de nouveaux composés de naphtylglyoxamides ainsi qu'un procédé relatif à la fabrication de ces composés et à leur utilisation pour inhiber la libération d'acides gras, induite par sPLA¿2?, pour le traitement d'affections telle que le choc septique.
CA 2240404 1995-12-13 1996-12-09 Naphtylglyoxamides en tant qu'inhibiteurs de spla2 Abandoned CA2240404A1 (fr)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US855795P 1995-12-13 1995-12-13
US60/008,557 1995-12-13
GBGB9602268.6A GB9602268D0 (en) 1996-02-05 1996-02-05 Naphthyl glyoxamides as sPLA2 inhibitors
GB9602268.6 1996-02-05
PCT/US1996/019529 WO1997021716A1 (fr) 1995-12-13 1996-12-09 NAPHTYLGLYOXAMIDES EN TANT QU'INHIBITEURS DE sPLA¿2?

Publications (1)

Publication Number Publication Date
CA2240404A1 true CA2240404A1 (fr) 1997-06-19

Family

ID=29407348

Family Applications (1)

Application Number Title Priority Date Filing Date
CA 2240404 Abandoned CA2240404A1 (fr) 1995-12-13 1996-12-09 Naphtylglyoxamides en tant qu'inhibiteurs de spla2

Country Status (1)

Country Link
CA (1) CA2240404A1 (fr)

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